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S. Colletti · SciRah

Researcher profile · Semantic Scholar

S. Colletti

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S. Colletti — researcher profile on SciRah

h-index: 30
Works: 86
Citations: 3,808

Most-cited papers

Apicidin: a novel antiprotozoal agent that inhibits parasite histone deacetylase.
Sandra J. Darkin-Rattray, A. Gurnett, R. W. Myers, P. Dulski +11 more
1996Proceedings of the National Academy of Sciences of the United States of America562 citations Open access
Semantic Scholar
International Union of Basic and Clinical Pharmacology. LXXXII: Nomenclature and Classification of Hydroxy-carboxylic Acid Receptors (GPR81, GPR109A, and GPR109B)
S. Offermanns, S. Colletti, T. Lovenberg, G. Semple +2 more
2011Pharmacological Reviews424 citations Open access
Semantic Scholar
Photoredox-catalyzed deuteration and tritiation of pharmaceutical compounds
Yong Yao Loh, K. Nagao, Andrew J. Hoover, D. Hesk +4 more
2017Science396 citations Open access
Semantic Scholar
Discovery of platencin, a dual FabF and FabH inhibitor with in vivo antibiotic properties
Jun Wang, S. Kodali, Sang-Ho Lee, Andrew M. Galgoci +19 more
2007Proceedings of the National Academy of Sciences of the United States of America349 citations Open access
Semantic Scholar
Structural basis for the cooperative allosteric activation of the free fatty acid receptor GPR40
Jun Lu, N. Byrne, John Wang, G. Bricogne +30 more
2017Nature Structural &Molecular Biology182 citations
Semantic Scholar
Niacin Lipid Efficacy Is Independent of Both the Niacin Receptor GPR109A and Free Fatty Acid Suppression
Brett Lauring, Andrew K. P. Taggart, J. Tata, Richard L. Dunbar +29 more
2012Science Translational Medicine126 citations
Semantic Scholar
Palladium-catalyzed Suzuki-Miyaura coupling of pyridyl-2-boronic esters with aryl halides using highly active and air-stable phosphine chloride and oxide ligands.
David X. Yang, S. Colletti, K. Wu, Mao-Ying Song +2 more
2009Organic Letters101 citations
Semantic Scholar
Chemoselective Peptide Modification via Photocatalytic Tryptophan β-Position Conjugation.
Younong Yu, Li-Kang Zhang, A. Buevich, Guo-Qing Li +4 more
2018Journal of the American Chemical Society94 citations
Semantic Scholar
Profiling and Application of Photoredox C(sp3)-C(sp2) Cross-Coupling in Medicinal Chemistry.
Rui Zhang, Guo-Qing Li, M. Wismer, Petr Vachal +2 more
2018ACS Medicinal Chemistry Letters78 citations Open access
Semantic Scholar
Broad spectrum antiprotozoal agents that inhibit histone deacetylase: structure-activity relationships of apicidin. Part 1.
S. Colletti, R. W. Myers, Sandra J. Darkin-Rattray, A. Gurnett +12 more
2001Bioorganic & Medicinal Chemistry Letters67 citations Open access
Semantic Scholar
Broad spectrum antiprotozoal agents that inhibit histone deacetylase: structure-activity relationships of apicidin. Part 2.
S. Colletti, R. W. Myers, Sandra J. Darkin-Rattray, A. Gurnett +12 more
2001Bioorganic & Medicinal Chemistry Letters66 citations Open access
Semantic Scholar
Total Synthesis of Bleomycin A2 and Related Agents. 1. Synthesis and DNA Binding Properties of the Extended C-Terminus: Tripeptide S, Tetrapeptide S, Pentapeptide S, and Related Agents
D. Boger, S. Colletti, Takeshi Honda, Royce F. Menezes
199465 citations
Semantic Scholar
Medicinal chemistry of siRNA delivery.
Matthew G. Stanton, S. Colletti
2010Journal of Medicinal Chemistry61 citations
Semantic Scholar
Synthesis of apicidin-derived quinolone derivatives: parasite-selective histone deacetylase inhibitors and antiproliferative agents.
P. Meinke, S. Colletti, G. Doss, R. W. Myers +8 more
2000Journal of Medicinal Chemistry50 citations Open access
Semantic Scholar
Synthesis and biological evaluation of platensimycin analogs.
Hong C. Shen, Fa-Xiang Ding, Sheo B. Singh, G. Parthasarathy +10 more
2009Bioorganic & Medicinal Chemistry Letters46 citations Open access
Semantic Scholar
Discovery of spirocyclic secondary amine-derived tertiary ureas as highly potent, selective and bioavailable soluble epoxide hydrolase inhibitors.
Hong C. Shen, Fa-Xiang Ding, Siyi Wang, Suo-Yu S. Xu +15 more
2009Bioorganic & Medicinal Chemistry Letters44 citations Open access
Semantic Scholar
GPR40 reduces food intake and body weight through GLP-1.
Judith N. Gorski, Michele J Pachanski, Joel Mane, C. Plummer +9 more
2017American Journal of Physiology. Endocrinology and Metabolism42 citations
Semantic Scholar
Total syntheses of (+)-P-3A, epi-(-)-P-3A, and (-)-desacetamido P-3A
D. Boger, Takeshi Honda, Royce F. Menezes, S. Colletti +2 more
199442 citations
Semantic Scholar
Asymmetric synthesis and metalation of a binaphthylcyclopentadiene, a C2-symmetric chiral cyclopentadiene
S. Colletti, R. L. Halterman
199141 citations
Semantic Scholar
Endosomolytic bioreducible poly(amido amine disulfide) polymer conjugates for the in vivo systemic delivery of siRNA therapeutics.
R. Parmar, Marina Busuek, E. Walsh, K. Leander +10 more
2013Bioconjugate chemistry39 citations
Semantic Scholar
Discovery of a highly potent, selective, and bioavailable soluble epoxide hydrolase inhibitor with excellent ex vivo target engagement.
Hong C. Shen, Fa-Xiang Ding, Siyi Wang, Q. Deng +20 more
2009Journal of Medicinal Chemistry38 citations Open access
Semantic Scholar
Cheminformatic Analysis of Natural Product-based Drugs and Chemical Probes
Samantha Stone, D. Newman, S. Colletti, Derek S. Tan
2021Natural product reports (Print)37 citations Open access
Semantic Scholar
Hybrid-designed inhibitors of p38 MAP kinase utilizing N-arylpyridazinones.
S. Colletti, Jessica L. Frie, E. Dixon, Suresh B. Singh +18 more
2003Journal of Medicinal Chemistry35 citations Open access
Semantic Scholar
Total Synthesis of Bleomycin A2 and Related Agents. 3. Synthesis and Comparative Evaluation of Deglycobleomycin A2,Epideglycobleomycin A2, Deglycobleomycin A1, and Desacetamido-, Descarboxamido-, Desmethyl-, and Desimidazolyldeglycobleomycin A2
D. Boger, Takeshi Honda, Royce F. Menezes, S. Colletti
199435 citations
Semantic Scholar
C2-symmetric 2,2'-dimethyl-1,1'-binaphthyl-bridged ansa-bis(1-indenyl)metal complexes
M. Burk, S. Colletti, R. L. Halterman
199135 citations
Semantic Scholar
Discovery of biaryl anthranilides as full agonists for the high affinity niacin receptor.
Hong C. Shen, Fa-Xiang Ding, S. Luell, M. Forrest +19 more
2007Journal of Medicinal Chemistry34 citations Open access
Semantic Scholar
Asymmetric epoxidation of unfunctionalized alkenes using the new C2-symmetrical 1,1′-binaphthyl-2,2′-dimethylene-bridged ansa-Bis(1-indenyl)titanium dichloride catalyst
S. Colletti, R. L. Halterman
199232 citations
Semantic Scholar
A strategy of employing aminoheterocycles as amide mimics to identify novel, potent and bioavailable soluble epoxide hydrolase inhibitors.
Hong C. Shen, Fa-Xiang Ding, Q. Deng, Suo-Yu S. Xu +11 more
2009Bioorganic & Medicinal Chemistry Letters31 citations Open access
Semantic Scholar
Binaphthylcyclopentadiene: a C2-symmetric annulated cyclopentadienyl ligand with axial chirality
S. Colletti, R. L. Halterman
198931 citations
Semantic Scholar
Tryptophan-replacement and indole-modified apicidins: synthesis of potent and selective antiprotozoal agents
S. Colletti, Chunshi Li, M. Fisher, M. Wyvratt +1 more
200030 citations
Semantic Scholar
Novel patent publications on high-affinity nicotinic acid receptor agonists
Hong C. Shen, S. Colletti
2009Expert Opinion on Therapeutic Patents28 citations
Semantic Scholar
Tetrahydro anthranilic acid as a surrogate for anthranilic acid: application to the discovery of potent niacin receptor agonists.
Subharekha Raghavan, G. Tria, Hong C. Shen, Fa-Xiang Ding +10 more
2008Bioorganic & Medicinal Chemistry Letters28 citations Open access
Semantic Scholar
Agonist lead identification for the high affinity niacin receptor GPR109a.
T. Gharbaoui, P. Skinner, Young-Jun Shin, Claudia Averbuj +22 more
2007Bioorganic & Medicinal Chemistry Letters28 citations Open access
Semantic Scholar
Synthesis of side chain modified apicidin derivatives: potent mechanism-based histone deacetylase inhibitors
P. Meinke, S. Colletti, Michelle B. Ayer, Sandra J. Darkin-Rattray +4 more
200028 citations
Semantic Scholar
Design and Synthesis of Novel, Selective GPR40 AgoPAMs.
C. Plummer, Matthew J. Clements, Helen Chen, M. Rajagopalan +23 more
2017ACS Medicinal Chemistry Letters27 citations Open access
Semantic Scholar
Discovery of the development candidate N-tert-butyl nodulisporamide: a safe and efficacious once monthly oral agent for the control of fleas and ticks on companion animals.
P. Meinke, S. Colletti, M. Fisher, M. Wyvratt +15 more
2009Journal of Medicinal Chemistry25 citations
Semantic Scholar
Discovery of pyrazolopyrimidines as the first class of allosteric agonists for the high affinity nicotinic acid receptor GPR109A.
Hong C. Shen, Andrew K. P. Taggart, L. Wilsie, M. Waters +3 more
2008Bioorganic & Medicinal Chemistry Letters23 citations Open access
Semantic Scholar
Discovery of 3,3-disubstituted piperidine-derived trisubstituted ureas as highly potent soluble epoxide hydrolase inhibitors.
Hong C. Shen, Fa-Xiang Ding, Q. Deng, Suo-Yu S. Xu +13 more
2009Bioorganic & Medicinal Chemistry Letters22 citations Open access
Semantic Scholar
Microbial biotransformation – an important tool for the study of drug metabolism
R. Salter, D. Beshore, S. Colletti, L. Evans +12 more
2018Xenobiotica; the fate of foreign compounds in biological systems21 citations
Semantic Scholar
Anthranilic acid replacements in a niacin receptor agonist.
Darby Schmidt, A. Smenton, Subharekha Raghavan, Hong C. Shen +16 more
2010Bioorganic & Medicinal Chemistry Letters20 citations Open access
Semantic Scholar
Improving the in vivo therapeutic index of siRNA polymer conjugates through increasing pH responsiveness.
Erin N. Guidry, J. Farand, A. Soheili, C. Parish +16 more
2014Bioconjugate chemistry19 citations
Semantic Scholar
Discovery of benzimidazole pyrrolidinyl amides as prolylcarboxypeptidase inhibitors.
Hong C. Shen, Fa-Xiang Ding, Changyou Zhou, Y. Xiong +17 more
2011Bioorganic & Medicinal Chemistry Letters19 citations Open access
Semantic Scholar
GPR109a agonists. Part 1: 5-Alkyl and 5-aryl-pyrazole-tetrazoles as agonists of the human orphan G-protein coupled receptor GPR109a.
J. Imbriglio, Sookhee Chang, Rui Liang, Subharekha Raghavan +12 more
2009Bioorganic & Medicinal Chemistry Letters19 citations Open access
Semantic Scholar
Discovery of orally bioavailable and novel urea agonists of the high affinity niacin receptor GPR109A.
Hong C. Shen, M. Szymonifka, Divya Kharbanda, Q. Deng +13 more
2007Bioorganic & Medicinal Chemistry Letters19 citations Open access
Semantic Scholar
Alpha-heteroarylation of esters, lactones, amides, and lactams by nucleophilic aromatic substitution.
Hong C. Shen, Fa-Xiang Ding, S. Colletti
2006Organic Letters19 citations Open access
Semantic Scholar
GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent
Michele J Pachanski, Melissa E Kirkland, Daniel T Kosinski, Joel Mane +20 more
2017PLoS ONE18 citations Open access
Semantic Scholar
Comparison of rat and dog models of vasodilatation and lipolysis for the calculation of a therapeutic index for GPR109A agonists.
E. Carballo-Jane, Lynn S. Gerckens, S. Luell, A. Parlapiano +8 more
2007Journal of pharmacological and toxicological methods18 citations
Semantic Scholar
The discovery of high affinity agonists of GPR109a with reduced serum shift and improved ADME properties.
J. Imbriglio, D. DiRocco, R. Bodner, Subharekha Raghavan +9 more
2011Bioorganic & Medicinal Chemistry Letters17 citations Open access
Semantic Scholar
Design and synthesis of histone deacetylase inhibitors: the development of apicidin transition state analogs
S. Colletti, R. W. Myers, Sandra J. Darkin-Rattray, D. Schmatz +3 more
200017 citations
Semantic Scholar
An in vivo evaluation of amphiphilic, biodegradable peptide copolymers as siRNA delivery agents.
Stephanie E. Barrett, M. Abrams, Rob S. Burke, B. Carr +16 more
2014International journal of pharmaceutics15 citations
Semantic Scholar

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