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P. Schiller · SciRah

Researcher profile · Semantic Scholar

P. Schiller

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P. Schiller — researcher profile on SciRah

h-index: 39
Works: 270
Citations: 6,538

Most-cited papers

A genetically encoded biosensor reveals location bias of opioid drug action
M. Stoeber, Damien Jullié, Braden T. Lobingier, T. Laeremans +4 more
2018bioRxiv272 citations Open access
Semantic Scholar
MicroRNA-195 promotes palmitate-induced apoptosis in cardiomyocytes by down-regulating Sirt1.
Huaqing Zhu, Yi-Xin Yang, Yan-Peng Wang, Jianmin Li +2 more
2011Cardiovascular Research192 citations
Semantic Scholar
Structural basis for bifunctional peptide recognition at human δ-Opioid receptor
G. Fenalti, N. Zatsepin, Cecilia Betti, P. Giguère +32 more
2015Nature Structural &Molecular Biology180 citations Open access
Semantic Scholar
Novel Therapies Targeting Inner Mitochondrial Membrane—From Discovery to Clinical Development
H. Szeto, P. Schiller
2011Pharmaceutical Research171 citations
Semantic Scholar
Bi- or multifunctional peptide drugs
P. Schiller
2009Life Science162 citations Open access
Semantic Scholar
Molecular Pharmacology of δ-Opioid Receptors
L. Gendron, C. Cahill, M. von Zastrow, P. Schiller +1 more
2016Pharmacological Reviews137 citations Open access
Semantic Scholar
Bioluminescence Resonance Energy Transfer Assays Reveal Ligand-specific Conformational Changes within Preformed Signaling Complexes Containing δ-Opioid Receptors and Heterotrimeric G Proteins*
N. Audet, C. Galés, E. Archer-Lahlou, M. Vallières +3 more
2008Journal of Biological Chemistry120 citations Open access
Semantic Scholar
Histone Deacetylase-3 Activation Promotes Tumor Necrosis Factor-α (TNF-α) Expression in Cardiomyocytes during Lipopolysaccharide Stimulation*
Huaqing Zhu, Limei Shan, P. Schiller, A. Mai +1 more
2010Journal of Biological Chemistry87 citations Open access
Semantic Scholar
Internalization and Src Activity Regulate the Time Course of ERK Activation by Delta Opioid Receptor Ligands*
N. Audet, M. Paquin-Gobeil, Olivier Landry-Paquet, P. Schiller +1 more
2005Journal of Biological Chemistry79 citations Open access
Semantic Scholar
Inhibition of calpain reduces oxidative stress and attenuates endothelial dysfunction in diabetes
Bainian Chen, Qing Zhao, R. Ni, Futian Tang +6 more
2014Cardiovascular Diabetology64 citations Open access
Semantic Scholar
Dicarba analogues of the cyclic enkephalin peptides H-Tyr-c[D-Cys-Gly-Phe-D(or L)-Cys]NH(2) retain high opioid activity.
I. Berezowska, N. Chung, C. Lemieux, B. Wilkes +1 more
2007Journal of Medicinal Chemistry51 citations Open access
Semantic Scholar
Conformational Dynamics of Kir3.1/Kir3.2 Channel Activation Via δ-Opioid Receptors
Melissa Richard-Lalonde, Karim Nagi, N. Audet, Rory Sleno +7 more
2013Molecular Pharmacology50 citations Open access
Semantic Scholar
Ligand- and cell-dependent determinants of internalization and cAMP modulation by delta opioid receptor (DOR) agonists
I. Charfi, Karim Nagi, O. Mnie-Filali, Dominic Thibault +4 more
2013Cellular and Molecular Life Sciences47 citations Open access
Semantic Scholar
Synthesis and Characterization of Potent and Selective μ-Opioid Receptor Antagonists, [Dmt1, d-2-Nal4]endomorphin-1 (Antanal-1) and [Dmt1, d-2-Nal4]endomorphin-2 (Antanal-2)
J. Fichna, J. Do Régo, N. Chung, C. Lemieux +5 more
200742 citations Open access
Semantic Scholar
Opioid peptide-derived analgesics
P. Schiller
2005AAPS Journal42 citations Open access
Semantic Scholar
Design of novel neurokinin 1 receptor antagonists based on conformationally constrained aromatic amino acids and discovery of a potent chimeric opioid agonist-neurokinin 1 receptor antagonist
S. Ballet, D. Feytens, K. Buysse, N. Chung +10 more
2011Journal of Medicinal Chemistry41 citations Open access
Semantic Scholar
Bifunctional Peptide-Based Opioid Agonist–Nociceptin Antagonist Ligands for Dual Treatment of Acute and Neuropathic Pain
Karel Guillemyn, Joanna Sarnowska, Camille Lagard, J. Dyniewicz +15 more
2016Journal of Medicinal Chemistry40 citations Open access
Semantic Scholar
Protective Effect of a Mitochondria-Targeted Peptide against the Development of Chemotherapy-Induced Peripheral Neuropathy in Mice
S. Toyama, N. Shimoyama, H. Szeto, P. Schiller +1 more
2018ACS Chemical Neuroscience37 citations Open access
Semantic Scholar
Impact of the prorenin/renin receptor on the development of obesity and associated cardiometabolic risk factors
Paul Tan, Z Shamansurova, Sandra Bisotto, C. Michel +6 more
2014Obesity35 citations Open access
Semantic Scholar
In vivo antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist - neurokinin 1 receptor antagonist chimera
Karel Guillemyn, P. Kleczkowska, A. Novoa, Bart Vandormael +8 more
2012Molecular Brain31 citations Open access
Semantic Scholar
Analgesic Properties of Opioid/NK1 Multitarget Ligands with Distinct in Vitro Profiles in Naive and Chronic Constriction Injury Mice
Joanna Starnowska, Roberto Costante, Karel Guillemyn, K. Popiołek-Barczyk +12 more
2017ACS Chemical Neuroscience30 citations Open access
Semantic Scholar
Variation of the net charge, lipophilicity and side chain flexibility in Dmt1-DALDA: effect on opioid activity and biodistribution
A. Novoa, Sylvia Van Dorpe, E. Wynendaele, M. Spetea +11 more
2012Journal of Medicinal Chemistry30 citations Open access
Semantic Scholar
‘Carba’-Analogues of Fentanyl are Opioid Receptor Agonists
G. Weltrowska, N. Chung, C. Lemieux, Jianxin Guo +3 more
2010Journal of Medicinal Chemistry29 citations Open access
Semantic Scholar
Blood-brain barrier penetration by two dermorphin tetrapeptide analogues: role of lipophilicity vs structural flexibility.
S. Ballet, A. Misicka, P. Kosson, C. Lemieux +4 more
2008Journal of Medicinal Chemistry28 citations Open access
Semantic Scholar
Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - neurokinin-1 antagonist peptidomimetics.
Karel Guillemyn, Patrycia Kleczkowska, A. Leśniak, J. Dyniewicz +18 more
2015European journal of medicinal chemistry27 citations Open access
Semantic Scholar
A New Structural Motif for μ-Opioid Antagonists
Isabelle Van den Eynde, G. Laus, P. Schiller, P. Kosson +3 more
200526 citations Open access
Semantic Scholar
Mast cell degranulation and fibroblast activation in the morphine-induced spinal mass: Role of Mas-related G protein-coupled receptor signaling.
T. Yaksh, Kelly A. Eddinger, Shinichi Kokubu, Zhen-Ping Wang +15 more
2019Anesthesiology25 citations Open access
Semantic Scholar
Synthesis of 4-amino-3-oxo-tetrahydroazepino[3,4-b]indoles: new conformationally constrained Trp analogs
Karolina Pulka, D. Feytens, Isabelle Van den Eynde, R. De Wachter +6 more
200723 citations
Semantic Scholar
Cyclic dermorphin tetrapeptide analogues obtained via ring-closing metathesis.
I. Berezowska, N. Chung, C. Lemieux, B. Wilkes +1 more
2006Acta Biochimica Polonica23 citations Open access
Semantic Scholar
Reciprocal Regulation of Agonist and Inverse Agonist Signaling Efficacy upon Short-Term Treatment of the Human δ-Opioid Receptor with an Inverse Agonist
G. Pineyro, M. Azzi, A. Delean, P. Schiller +1 more
2005Molecular Pharmacology21 citations
Semantic Scholar
Dual Alleviation of Acute and Neuropathic Pain by Fused Opioid Agonist-Neurokinin 1 Antagonist Peptidomimetics.
Cecilia Betti, Joanna Starnowska, J. Mika, J. Dyniewicz +18 more
2015ACS Medicinal Chemistry Letters20 citations Open access
Semantic Scholar
Determination of the intramolecular tyrosine-tryptophan distance in a 7-peptide related to the C-terminal sequence of cholecystokinin.
P. Schiller, S. Natarajan, M. Bodanszky
2009International journal of peptide & protein research20 citations
Semantic Scholar
Cyclic Enkephalins with a Diversely Substituted Guanidine Bridge or a Thiourea Bridge: Synthesis, Biological and Structural Evaluations
Youness Touati-Jallabe, Engin Bojnik, Baptiste Legrand, Elodie Mauchauffée +6 more
2013Journal of Medicinal Chemistry19 citations Open access
Semantic Scholar
Fluorescence study on the solution conformation to dynorphin in comparison of enkephalin.
P. Schiller
2009International journal of peptide & protein research19 citations
Semantic Scholar
1H n.m.r. investigation of conformational features of cyclic enkephalinamide analogs.
H. Mosberg, P. Schiller
2009International journal of peptide & protein research19 citations
Semantic Scholar
The Bifunctional μ Opioid Agonist/Antioxidant [Dmt1]DALDA Is a Superior Analgesic in an Animal Model of Complex Regional Pain Syndrome-Type I
P. Schiller, Thi M.-D. Nguyen, A. Saray, An-Nie-Wing-Hoi Poon +2 more
2015ACS Chemical Neuroscience18 citations Open access
Semantic Scholar
Influence of new deltorphin analogues on reinstatement of cocaine-induced conditioned place preference in rats
J. Kotlinska, Ewa Gibuła-Bruzda, A. Pachuta, D. Kunce +4 more
2010Behavioural Pharmacology18 citations
Semantic Scholar
β-methyl substitution of cyclohexylalanine in Dmt-Tic-Cha-Phe peptides results in highly potent δ opioid antagonists
G. Tóth, Enikő Ioja, C. Tömböly, S. Ballet +7 more
200718 citations Open access
Semantic Scholar
Mannosylated glycoliposomes for the delivery of a peptide kappa opioid receptor antagonist to the brain.
Jordan D Lewicky, N. Fraleigh, Amanda Boraman, Alexandrine L Martel +6 more
2020European journal of pharmaceutics and biopharmaceutics17 citations Open access
Semantic Scholar
Solid-Phase Azopeptide Diels-Alder Chemistry for Aza-pipecolyl Residue Synthesis To Study Peptide Conformation.
Ramesh M Chingle, Mukandila Mulumba, N. Chung, Thi M.-D. Nguyen +4 more
2019Journal of Organic Chemistry17 citations
Semantic Scholar
Endocytic Profiles of δ-Opioid Receptor Ligands Determine the Duration of Rapid but Not Sustained cAMP Responses
H. B. Tudashki, D. Robertson, P. Schiller, G. Pineyro
2014Molecular Pharmacology17 citations Open access
Semantic Scholar
Agonist vs Antagonist Behavior of δ Opioid Peptides Containing Novel Phenylalanine Analogues in Place of Tyr1
I. Berezowska, N. Chung, C. Lemieux, B. Wilkes +1 more
2009Journal of Medicinal Chemistry17 citations Open access
Semantic Scholar
A novel cyclic enkephalin analogue with potent opioid antagonist activity.
G. Weltrowska, Yi-Xin Lu, C. Lemieux, N. Chung +1 more
2004Bioorganic & Medicinal Chemistry Letters17 citations Open access
Semantic Scholar
[Dmt1]DALDA analogues with enhanced μ opioid agonist potency and with a mixed μ/κ opioid activity profile
Longxiang Bai, Zi-Yuan Li, Jia-Jia Chen, N. Chung +3 more
2014Bioorganic & Medicinal Chemistry16 citations Open access
Semantic Scholar
Novel highly potent mu-opioid receptor antagonist based on endomorphin-2 structure.
J. Fichna, J. Do Régo, T. Janecki, Renata Staniszewska +5 more
2008Bioorganic & Medicinal Chemistry Letters15 citations Open access
Semantic Scholar
Synthesis of 8-L-tryptophan-oxytocin and determination of one of its conformational parameters.
M. Bodanszky, J. Tolle, Maria A. Bednarek, P. Schiller
2009International journal of peptide & protein research14 citations
Semantic Scholar
[Dmt1, d-1-Nal3]morphiceptin, a novel opioid peptide analog with high analgesic activity.
J. Fichna, J. Do Régo, N. Chung, J. Costentin +2 more
2008Peptides12 citations
Semantic Scholar
Novel endomorphin-2 analogs with mu-opioid receptor antagonist activity.
R. Kruszyński, J. Fichna, J. Do Régo, N. Chung +4 more
2005Journal of Peptide Research12 citations
Semantic Scholar
Strengthening peptide-based drug activity with novel glyconanoparticle
Jordan D Lewicky, Alexandrine L Martel, N. Fraleigh, Amanda Boraman +5 more
2018PLoS ONE10 citations Open access
Semantic Scholar
In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt1-DALDA Analogues
S. Ballet, Cecilia Betti, A. Novoa, C. Tömböly +9 more
2014ACS Medicinal Chemistry Letters10 citations Open access
Semantic Scholar

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