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C. Menet · SciRah

Researcher profile · Semantic Scholar

C. Menet

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C. Menet — researcher profile on SciRah

h-index: 17
Works: 43
Citations: 1,024

Most-cited papers

Preclinical Characterization of GLPG0634, a Selective Inhibitor of JAK1, for the Treatment of Inflammatory Diseases
L. van Rompaey, R. Galien, E. M. van der Aar, P. Clément-Lacroix +13 more
2013Journal of Immunology225 citations Open access
Semantic Scholar
Triazolopyridines as selective JAK1 inhibitors: from hit identification to GLPG0634.
C. Menet, S. Fletcher, G. V. Van Lommen, Raphaël Geney +15 more
2014Journal of Medicinal Chemistry108 citations Open access
Semantic Scholar
Type II kinase inhibitors: an opportunity in cancer for rational design.
J. Blanc, Raphaël Geney, C. Menet
2013Anti-Cancer Agents in Medicinal Chemistry96 citations
Semantic Scholar
Advances in the discovery of selective JAK inhibitors.
C. Menet, L. van Rompaey, Raphaël Geney
2013Progress in Medicinal Chemistry74 citations
Semantic Scholar
Synthesis of (-)-kainic acid using chiral lithium amides in an asymmetric dearomatizing cyclization
J. Clayden, C. Menet, K. Tchabanenko
200248 citations
Semantic Scholar
Wandering beyond small molecules: peptides as allosteric protein modulators.
M. Mannes, C. Martin, C. Menet, S. Ballet
2021TIPS - Trends in Pharmacological Sciences42 citations
Semantic Scholar
Accelerating GPCR Drug Discovery With Conformation-Stabilizing VHHs
T. Laeremans, Z. Sands, Pieter Claes, Ann De Blieck +7 more
2022Frontiers in Molecular Biosciences41 citations Open access
Semantic Scholar
Dearomatizing anionic cyclization of substituted N-cumyl-N-benzyl- benzamides on treatment with LDA: synthesis of partially saturated substituted isoindolones
J. Clayden, C. Menet, D. J. Mansfield
2000Organic Letters40 citations
Semantic Scholar
IRAK4 inhibition dampens pathogenic processes driving inflammatory skin diseases
S. Lavazais, M. Jargosch, S. Dupont, Frédéric Labéguère +16 more
2023Science Translational Medicine39 citations
Semantic Scholar
Asymmetric deprotonation and dearomatising cyclisation of N-benzyl benzamides using chiral lithium amides: formal synthesis of (-)-kainic acid.
J. Clayden, C. Menet, D. J. Mansfield
2002Chemical Communications38 citations
Semantic Scholar
2,3-Dihydroisoindolones by cyclisation and rearomatisation of lithiated benzamides
J. Clayden, C. Menet
200334 citations
Semantic Scholar
Discovery of the S1P2 Antagonist GLPG2938 (1-[2-Ethoxy-6-(trifluoromethyl)-4-pyridyl]-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea), a Preclinical Candidate for the Treatment of Idiopathic Pulmonary Fibrosis.
Oscar Mammoliti, Adeline Palisse, Caroline Joannesse, Sandy El Bkassiny +16 more
2021Journal of Medicinal Chemistry28 citations Open access
Semantic Scholar
Synthesis of α-methyl kainic acid by stereospecific lithiation-dearomatizing cyclization of a chiral benzamide
J. Clayden, F. E. Knowles, C. Menet
200327 citations
Semantic Scholar
Progress toward JAK1-selective inhibitors.
C. Menet, Oscar Mammoliti, Miriam López-Ramos
2015Future Medicinal Chemistry26 citations
Semantic Scholar
Stereospecific photochemical ring expansion of lithiated benzamides.
J. Clayden, F. E. Knowles, C. Menet
2003Journal of the American Chemical Society23 citations Open access
Semantic Scholar
Discovery of GLPG2451, a Novel Once Daily Potentiator for the Treatment of Cystic Fibrosis.
S. E. Van der Plas, H. Kelgtermans, Oscar Mammoliti, C. Menet +12 more
2021Journal of Medicinal Chemistry18 citations Open access
Semantic Scholar
Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases.
Oscar Mammoliti, Koen Jansen, Sandy El Bkassiny, Adeline Palisse +30 more
2021Journal of Medicinal Chemistry17 citations Open access
Semantic Scholar
Toward selective TYK2 inhibitors as therapeutic agents for the treatment of inflammatory diseases.
C. Menet
2014Pharmaceutical Patent Analyst16 citations
Semantic Scholar
A Dual Inhibition, a Better Solution: Development of a JAK1/TYK2 inhibitor.
C. Menet
2018Journal of Medicinal Chemistry15 citations
Semantic Scholar
Stereospecific dearomatising cyclisation of tertiary .alpha.-amidoorganolithiums.
J. Clayden, F. E. Knowles, C. Menet
200315 citations
Semantic Scholar
Design and synthesis of APTCs (aminopyrrolidinetricarboxylic acids): identification of a new group III metabotropic glutamate receptor selective agonist.
S. Schann, C. Menet, Paul Arvault, G. Mercier +7 more
2006Bioorganic & Medicinal Chemistry Letters14 citations Open access
Semantic Scholar
Development of Generic G Protein Peptidomimetics Able to Stabilize Active State Gs Protein-Coupled Receptors for Application in Drug Discovery.
M. Mannes, C. Martin, Sarah Triest, Marilisa Pia Dimmito +4 more
2021Angewandte Chemie13 citations
Semantic Scholar
meso-Selective' functionalisation of N-benzyl-α-methylbenzylamine derivatives by α-lithiation and alkylation
R. Bragg, J. Clayden, C. Menet
200211 citations
Semantic Scholar
Modulation of sleep behavior in zebrafish larvae by pharmacological targeting of the orexin receptor
Marie-Christine Pardon, Pieter Claes, Sarah Druwé, M. Martini +4 more
2022Frontiers in Pharmacology7 citations Open access
Semantic Scholar
Expediting drug discovery: recent advances in fast medicinal chemistry--optimization of hits and leads.
P. Edwards, B. Allart, M. Andrews, J. Clase +1 more
2006Current opinion in drug discovery & development6 citations
Semantic Scholar
Design of a potent and selective dual JAK1/TYK2 inhibitor.
Oscar Mammoliti, C. Menet, C. Cottereaux, J. Blanc +19 more
2024Bioorganic & Medicinal Chemistry3 citations Open access
Semantic Scholar
Regio- and Diastereoselective Functionalization of 3-Amino-hexahydrooxazoninones
Ben Schurgers, J. Wouters, Ann De Blieck, G. V. Van Lommen +2 more
2018Annalen der Pharmacie2 citations Open access
Semantic Scholar
Development of a G protein mimetic toolbox to conformationally lock G protein coupled receptors (GPCRs) in the active state
Thijs Vynckier, M. Mannes, Morgane Rivoal, Charlotte Martin +4 more
2026Proceedings of the 38th European Peptide Symposium0 citations Open access
Semantic Scholar
Development of G Protein Peptidomimetics to Stabilize Active State G Protein-Coupled Receptors
M. Mannes, C. Martin, Sarah Triest, Toon Laeremens +2 more
2022Proceedings of the 36th European and the 12th International Peptide Symposium0 citations Open access
Semantic Scholar
Correction to "Discovery of GLPG2451, a Novel Once Daily Potentiator for the Treatment of Cystic Fibrosis".
S. E. Van der Plas, H. Kelgtermans, Oscar Mammoliti, C. Menet +12 more
2021Journal of Medicinal Chemistry0 citations Open access
Semantic Scholar
THU0138 Glpg0634m1, A Major Metabolite of the Jak1-Selective Inhibitor Glpg0634, is Also Jak1-Selective and Efficient in the Rat CIA Model
C. Belleville-Da-Costa, D. Merciris, Béatrice Vayssière, N. Houvenaghel +10 more
20140 citations
Semantic Scholar
Selective Inhibitor of JAK 1 , for the Preclinical Characterization of GLPG 0634 , a Feyen and
C. Menet, Fletcher, R. Brys, Gerben A. van'T Klooster +14 more
20130 citations
Semantic Scholar
Novel compound for the treatment of degenerative and inflammatory diseases.
J. Blanc, C. Menet
20100 citations
Semantic Scholar
New compound useful for the treatment of degenerative and inflammatory diseases
C. Menet, J. Blanc
20100 citations
Semantic Scholar
Novel compound useful for the treatment of inflammatory and degenerative diseases
J. Blanc, C. Menet
20100 citations
Semantic Scholar
Novel compounds which are useful for the treatment of degenerative and inflammatory diseases
Nolwenn Jouannigot, C. Menet, Rompaey Luc Juliaan Corina Van, S. Fletcher +3 more
20090 citations
Semantic Scholar
Novel compounds useful for treating degenerative and inflammatory diseases
C. Menet, J. Blanc
20090 citations
Semantic Scholar
Stereospecific Dearomatizing Cyclization of Tertiary α‐Amidoorganolithiums.
J. Clayden, F. E. Knowles, C. Menet
20040 citations
Semantic Scholar
Synthesis of α-Methyl Kainic Acid (I) by Stereospecific Lithiation—Dearomatizing Cyclization of a Chiral Benzamide.
J. Clayden, F. E. Knowles, C. Menet
20030 citations
Semantic Scholar
2,3‐Dihydroisoindolones by Cyclization and Rearomatization of Lithiated Benzamides.
J. Clayden, C. Menet
20030 citations
Semantic Scholar
“meso-Selective” Functionalization of N-Benzyl-α-methylbenzylamine Derivatives by α-Lithiation and Alkylation.
R. Bragg, J. Clayden, C. Menet
20020 citations
Semantic Scholar
Asymmetric Deprotonation and Dearomatizing Cyclization of N-Benzyl Benzamides Using Chiral Lithium Amides: Formal Synthesis of (-)-Kainic Acid.
J. Clayden, C. Menet, D. J. Mansfield
20020 citations
Semantic Scholar
Dearomatizing Anionic Cyclization of Substituted N-Cumyl-N-benzylbenzamides on Treatment with LDA: Synthesis of Partially Saturated Substituted Isoindolones.
J. Clayden, C. Menet, D. J. Mansfield
20010 citations
Semantic Scholar

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