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Emilie Durieu · SciRah

Researcher profile · Semantic Scholar

Emilie Durieu

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Emilie Durieu — researcher profile on SciRah

h-index: 17
Works: 29
Citations: 912

Most-cited papers

Selectivity, cocrystal structures, and neuroprotective properties of leucettines, a family of protein kinase inhibitors derived from the marine sponge alkaloid leucettamine B.
Tania Tahtouh, J. Elkins, P. Filippakopoulos, M. Soundararajan +12 more
2012Journal of Medicinal Chemistry188 citations Open access
Semantic Scholar
Synthesis, protein kinase inhibitory potencies, and in vitro antiproliferative activities of meridianin derivatives.
F. Giraud, Georges Alves, E. Débiton, L. Nauton +8 more
2011Journal of Medicinal Chemistry101 citations Open access
Semantic Scholar
Novel Inverse Binding Mode of Indirubin Derivatives Yields Improved Selectivity for DYRK Kinases
V. Myrianthopoulos, M. Kritsanida, N. Gaboriaud-Kolar, P. Magiatis +11 more
2012ACS Medicinal Chemistry Letters69 citations Open access
Semantic Scholar
Pharmacological Assessment Defines Leishmania donovani Casein Kinase 1 as a Drug Target and Reveals Important Functions in Parasite Viability and Intracellular Infection
N. Rachidi, Jean-François Taly, Emilie Durieu, Olivier Leclercq +6 more
2013Antimicrobial Agents and Chemotherapy54 citations Open access
Semantic Scholar
Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases
Nadège Loaëc, Eletta Attanasio, Benoît Villiers, Emilie Durieu +13 more
2017Marine Drugs48 citations Open access
Semantic Scholar
Synthesis, resolution, and biological evaluation of atropisomeric (aR)- and (aS)-16-methyllamellarins N: unique effects of the axial chirality on the selectivity of protein kinases inhibition.
K. Yoshida, Ryosuke Itoyama, Masashi Yamahira, Junji Tanaka +7 more
2013Journal of Medicinal Chemistry45 citations Open access
Semantic Scholar
From Drug Screening to Target Deconvolution: a Target-Based Drug Discovery Pipeline Using Leishmania Casein Kinase 1 Isoform 2 To Identify Compounds with Antileishmanial Activity
Emilie Durieu, E. Prina, Olivier Leclercq, Nassima Oumata +11 more
2016Antimicrobial Agents and Chemotherapy42 citations Open access
Semantic Scholar
Identification and structure-activity relationship of 8-hydroxy-quinoline-7-carboxylic acid derivatives as inhibitors of Pim-1 kinase.
Faten Sliman, Mélina Blairvacq, Emilie Durieu, L. Meijer +2 more
2010Bioorganic & Medicinal Chemistry Letters38 citations Open access
Semantic Scholar
cdc-Like/Dual-Specificity Tyrosine Phosphorylation–Regulated Kinases Inhibitor Leucettine L41 Induces mTOR-Dependent Autophagy: Implication for Alzheimer’s Disease
X. Fant, Emilie Durieu, G. Chicanne, B. Payrastre +6 more
2014Molecular Pharmacology33 citations Open access
Semantic Scholar
Library-based Discovery of DYRK1A/CLK1 Inhibitors from Natural Product Extracts
Patrick Grabher, Emilie Durieu, Eirini Kouloura, M. Halabalaki +4 more
2012Planta Medica33 citations
Semantic Scholar
Inhibition of NF-κB–Mediated Signaling by the Cyclin-Dependent Kinase Inhibitor CR8 Overcomes Prosurvival Stimuli to Induce Apoptosis in Chronic Lymphocytic Leukemia Cells
E. Cosimo, Alison M. McCaig, Luke J. M. Carter-Brzezinski, H. Wheadon +8 more
2013Clinical Cancer Research32 citations Open access
Semantic Scholar
Dispacamide E and other bioactive bromopyrrole alkaloids from two Indonesian marine sponges of the genus Stylissa
S. S. Ebada, M. Linh, A. Longeon, N. D. de Voogd +6 more
2015Natural Product Research30 citations
Semantic Scholar
Roscovitine is a proteostasis regulator that corrects the trafficking defect of F508del‐CFTR by a CDK‐independent mechanism
C. Norez, C. Vandebrouck, J. Bertrand, Sabrina Noël +8 more
2014British Journal of Pharmacology29 citations Open access
Semantic Scholar
Chemical synthesis and biological validation of immobilized protein kinase inhibitory Leucettines.
Guillaume Burgy, Tania Tahtouh, Emilie Durieu, Béatrice Foll-Josselin +4 more
2013European journal of medicinal chemistry29 citations Open access
Semantic Scholar
Induction of Amyloid-β42 Production by Fipronil and Other Pyrazole Insecticides
M. Cam, Emilie Durieu, M. Bodin, A. Manousopoulou +25 more
2018Journal of Alzheimer's Disease24 citations Open access
Semantic Scholar
Aftins Increase Amyloid-β42, Lower Amyloid-β38, and Do Not Alter Amyloid-β40 Extracellular Production in vitro: Toward a Chemical Model of Alzheimer’s Disease?
A. Hochard, Nassima Oumata, K. Bettayeb, O. Gloulou +8 more
2013Journal of Alzheimer's Disease20 citations Open access
Semantic Scholar
Structure-Activity Relationship in the Leucettine Family of Kinase Inhibitors.
Tania Tahtouh, Emilie Durieu, Benoît Villiers, Céline Bruyère +18 more
2021Journal of Medicinal Chemistry18 citations Open access
Semantic Scholar
New 5-ylidene rhodanine derivatives based on the dispacamide A model
S. Guiheneuf, L. Paquin, F. Carreaux, Emilie Durieu +3 more
2014Molecular diversity14 citations Open access
Semantic Scholar
Synthesis of N,N'-bis(5-arylidene-4-oxo-3,5-dihydro-4H-imidazol-2-yl)diamines bearing various linkers and biological evaluation as potential inhibitors of kinases.
W. Coulibaly, L. Paquin, Anoubilé Bénié, Y. Bekro +3 more
2012European journal of medicinal chemistry14 citations
Semantic Scholar
An efficient approach to dispacamide A and its derivatives.
S. Guiheneuf, L. Paquin, F. Carreaux, Emilie Durieu +2 more
2012Organic and biomolecular chemistry14 citations
Semantic Scholar
Specific Triazine Herbicides Induce Amyloid-β42 Production
E. Portelius, Emilie Durieu, M. Bodin, M. Cam +24 more
2016Journal of Alzheimer's Disease12 citations Open access
Semantic Scholar
Design and Microwave Synthesis of New (5Z) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5Z) 2-Amino-5-arylidene-1,3-thiazol-4(5H)-one as New Inhibitors of Protein Kinase DYRK1A
Khadidja Bourahla, S. Guiheneuf, Emmanuelle Limanton, L. Paquin +8 more
2021Pharmaceuticals9 citations Open access
Semantic Scholar
A Collection of Bioactive Nitrogen-Containing Molecules from the Marine Sponge Acanthostrongylophora ingens
Germana Esposito, Linh H. Mai, A. Longeon, A. Mangoni +5 more
2019Marine Drugs9 citations Open access
Semantic Scholar
Microwave Assisted Organic Synthesis (MAOS) of New Dispacamide A Derivatives Bearing a Thiazolinone Platform, Biological Assays on Inhibition of Protein Kinases and Cell Effects
S. Guiheneuf, L. Paquin, F. Carreaux, Emilie Durieu +5 more
20136 citations
Semantic Scholar
Exploring the Synthesis of New 1-(4-Substitutedphenylamino) imidazo[1,5-a]indol-3-one Derivatives as Cyclized Analogs of Leucettines
Guillaume Burgy, Emmanuelle Limanton, F. Carreaux, Emilie Durieu +2 more
20142 citations Open access
Semantic Scholar
Intracellular Infection Functions in Parasite Viability and Drug Target and Reveals Important Leishmania donovani Casein Kinase 1 as a Pharmacological Assessment Defines
C. Notredame, L. Meijer, G. Späth, Leclercq +6 more
20140 citations
Semantic Scholar
s and reveals important functions in parasite viability and intracellular infection. t u
N. Rachidi, Jean-François Taly, Emilie Durieu, Olivier Leclercq +6 more
20130 citations
Semantic Scholar
Cosimo, Emilio et al. (2014) Inhibition of NF-κB-mediated signaling by the cyclin-dependent kinase inhibitor CR8 overcomes pro-survival stimuli to induce apoptosis in chronic lymphocytic leukemia cells. Clinical Cancer
E. Cosimo, Alison M. McCaig, Luke J. M. Carter-Brzezinski, H. Wheadon +8 more
20130 citations
Semantic Scholar
Human DYRK1A in complex with Leucettine L41
J. Elkins, M. Soundararajan, J. Muniz, Tania Tahtouh +13 more
20120 citations
Semantic Scholar

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