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F. Giraud · SciRah

Researcher profile · Semantic Scholar

F. Giraud

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F. Giraud — researcher profile on SciRah

h-index: 15
Works: 51
Citations: 652

Most-cited papers

Synthesis, protein kinase inhibitory potencies, and in vitro antiproliferative activities of meridianin derivatives.
F. Giraud, Georges Alves, E. Débiton, L. Nauton +8 more
2011Journal of Medicinal Chemistry101 citations Open access
Semantic Scholar
Alternative RNA splicing modulates ribosomal composition and determines the spatial phenotype of glioblastoma cells
T. Larionova, Soniya Bastola, Tatiana E Aksinina, Ksenia S. Anufrieva +22 more
2022Nature Cell Biology56 citations Open access
Semantic Scholar
Synthesis and structure-activity relationships of 2-phenyl-1-[(pyridinyl- and piperidinylmethyl)amino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents.
F. Giraud, Rémi Guillon, C. Logé, F. Pagniez +3 more
2009Bioorganic & Medicinal Chemistry Letters47 citations
Semantic Scholar
Efficient microwave-assisted synthesis of 1-(1H-indol-1-yl)-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents
N. Lebouvier, F. Giraud, T. Corbin, Young Na +3 more
200639 citations
Semantic Scholar
Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co-crystal structure.
Y. Esvan, Wael Zeinyeh, T. Boibessot, L. Nauton +8 more
2016European journal of medicinal chemistry34 citations Open access
Semantic Scholar
Recent Advances in Pain Management: Relevant Protein Kinases and Their Inhibitors
F. Giraud, Elisabeth Pereira, F. Anizon, P. Moreau
2021Molecules32 citations Open access
Semantic Scholar
Design, synthesis, and evaluation of 1-(N-benzylamino)-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents.
F. Giraud, C. Logé, F. Pagniez, Damien Crépin +2 more
2008Bioorganic & Medicinal Chemistry Letters32 citations
Semantic Scholar
New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis.
H. Tazarki, Wael Zeinyeh, Y. Esvan, S. Knapp +11 more
2019European journal of medicinal chemistry30 citations Open access
Semantic Scholar
Synthesis and biological activities of 4-substituted pyrrolo[2,3-a]carbazole Pim kinase inhibitors.
F. Giraud, Rufine Akué-Gédu, L. Nauton, N. Candelon +4 more
2012European journal of medicinal chemistry28 citations Open access
Semantic Scholar
Design of new antifungal agents: synthesis and evaluation of 1-[(1H-indol-5-ylmethyl)amino]-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.
Rémi Guillon, F. Giraud, C. Logé, M. le Borgne +3 more
2009Bioorganic & Medicinal Chemistry Letters26 citations
Semantic Scholar
Synthesis and biological activity of pyrazole analogues of the staurosporine aglycon K252c.
Y. Esvan, F. Giraud, Elisabeth Pereira, Virginie Suchaud +8 more
2016Bioorganic & Medicinal Chemistry18 citations Open access
Semantic Scholar
New N-1,N-10-bridged pyrrolo[2,3-a]carbazole-3-carbaldehydes: synthesis and biological activities.
F. Giraud, M. Bourhis, L. Nauton, V. Théry +4 more
2014Bioorganic chemistry (Print)18 citations
Semantic Scholar
Design, Synthesis, and in vitro Antifungal Activity of 1‐[(4‐Substituted‐benzyl)methylamino]‐2‐(2,4‐difluorophenyl)‐3‐(1H‐1,2,4‐triazol‐1‐yl)propan‐2‐ols
Rémi Guillon, F. Pagniez, F. Giraud, Damien Crépin +6 more
2011ChemMedChem17 citations
Semantic Scholar
An efficient route from coumarins to highly functionalized N-phenyl-2-quinolinones via Buchwald–Hartwig amination
T. Ullrich, F. Giraud
200317 citations
Semantic Scholar
Synthesis of pyrazolo[4,3-a]phenanthridines, a new scaffold for Pim kinase inhibition.
Virginie Suchaud, Laurent Gavara, F. Giraud, L. Nauton +3 more
2014Bioorganic & Medicinal Chemistry16 citations Open access
Semantic Scholar
A Kinase Inhibitor with Anti-Pim Kinase Activity is a Potent and Selective Cytotoxic Agent Toward Acute Myeloid Leukemia
Ronja Bjørnstad, Reidun Aesoy, Ø. Bruserud, A. Brenner +7 more
2019Molecular Cancer Therapeutics15 citations Open access
Semantic Scholar
Synthesis and preliminary in vitro kinase inhibition evaluation of new diversely substituted pyrido[3,4-g]quinazoline derivatives.
Wael Zeinyeh, Y. Esvan, L. Nauton, Nadège Loaëc +5 more
2016Bioorganic & Medicinal Chemistry Letters14 citations
Semantic Scholar
Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activity.
Wael Zeinyeh, Y. Esvan, B. Josselin, M. Defois +7 more
2022European journal of medicinal chemistry11 citations Open access
Semantic Scholar
Design, synthesis and evaluation of 3-(imidazol- 1-ylmethyl)indoles as antileishmanial agents. Part II
F. Giraud, C. Logé, F. Pagniez, Damien Crépin +4 more
2009Journal of Enzyme Inhibition and Medicinal Chemistry11 citations Open access
Semantic Scholar
Kinase inhibitions in pyrido[4,3-h] and [3,4-g]quinazolines: Synthesis, SAR and molecular modeling studies.
Wael Zeinyeh, Y. Esvan, B. Josselin, B. Baratte +7 more
2019Bioorganic & Medicinal Chemistry10 citations Open access
Semantic Scholar
Synthesis and Applications of Dihydropyrrolocarbazoles
F. Giraud, Elisabeth Pereira, F. Anizon, P. Moreau
2019Annalen der Pharmacie9 citations
Semantic Scholar
Synthesis and activities of new indolopyrrolobenzodiazepine derivatives toward acute myeloid leukemia cells.
F. Giraud, M. Bourhis, E. Ebrahimi, L. Herfindal +5 more
2015Bioorganic & Medicinal Chemistry8 citations Open access
Semantic Scholar
Liposomes loaded with daunorubicin and an emetine prodrug for improved selective cytotoxicity towards acute myeloid leukaemia cells.
Ingeborg Nerbø Reiten, F. Giraud, Tuva Torblå Augedal, Jan-Lukas Førde +6 more
2024International journal of pharmaceutics7 citations Open access
Semantic Scholar
Pyridin-2(1H)one derivatives: A possible new class of therapeutics for mechanical allodynia.
A. Visseq, Amélie Descheemaeker, Nicolas Pinto-Pardo, L. Nauton +7 more
2019European journal of medicinal chemistry7 citations Open access
Semantic Scholar
Synthesis and antiproliferative evaluation of glucosylated pyrazole analogs of K252c
Bachir Douara, Y. Esvan, Elisabeth Pereira, F. Giraud +5 more
20186 citations
Semantic Scholar
Synthesis of N-aryl-3-(indol-3-yl)propanamides and their immunosuppressive activities.
F. Giraud, P. Marchand, D. Carbonnelle, Michael Sartor +2 more
2010Bioorganic & Medicinal Chemistry Letters6 citations Open access
Semantic Scholar
Heteroaromatic Pim Kinase Inhibitors Containing a Pyrazole Moiety.
P. Moreau, F. Anizon, F. Giraud, Y. Esvan
2016Recent Patents on Anti-Cancer Drug Discovery5 citations
Semantic Scholar
Synthesis, kinase inhibition and anti-leukemic activities of diversely substituted indolopyrazolocarbazoles.
Théo Frazier, Elisabeth Pereira, Reidun Aesoy, L. Nauton +4 more
2024European journal of medicinal chemistry4 citations Open access
Semantic Scholar
Synthesis and biological activities of new pyrrolocarbazole-imidazobenzimidazole conjugates
F. Anizon, F. Giraud, E. Ivanova, D. Kaluzhny +3 more
2020Tetrahedron Letters4 citations Open access
Semantic Scholar
A 3D-QSAR CoMSIA study on 3-azolylmethylindoles as anti-leishmanial agents
F. Giraud, C. Logé, M. le Borgne, F. Pagniez +2 more
2006SAR and QSAR in environmental research (Print)4 citations
Semantic Scholar
The Nitro Group Reshapes the Effects of Pyrido[3,4-g]quinazoline Derivatives on DYRK/CLK Activity and RNA Splicing in Glioblastoma Cells
S. Borisevich, Tatiana E Aksinina, M. G. Ilyina, V. Shender +11 more
2024Cancers3 citations Open access
Semantic Scholar
Synthesis and biological evaluation of 1H-pyrrolo[3,2-g]isoquinolines.
M. Defois, B. Josselin, Pierre Brindeau, Andreas Krämer +5 more
2024Bioorganic & Medicinal Chemistry3 citations Open access
Semantic Scholar
Synthesis and Kinase Inhibitory Potencies of Pyrazolo[3,4-g]isoquinolines
M. Defois, Chloé Rémondin, B. Josselin, L. Nauton +5 more
2022Molecules3 citations Open access
Semantic Scholar
Advances in the Synthesis and Kinase Inhibitory Potencies of Non‐fused Indazole Derivatives
F. Giraud, F. Anizon, P. Moreau
20163 citations
Semantic Scholar
Synthesis and biological activity of 1H-pyrrolo[3,2-g]isoquinolines as Haspin kinase inhibitors.
Killian Malosse, Marie Ben Doula, B. Josselin, Thomas Robert +4 more
2025Bioorganic & Medicinal Chemistry2 citations Open access
Semantic Scholar
Synthesis of new pyrazolo[4,3-a]phenanthridine Pim-1 inhibitors and evaluation of their cytotoxic activity towards the MOLM-13 acute myeloid leukemia cell line.
Etienne Auvert, Reidun Aesoy, F. Giraud, L. Herfindal +2 more
2022Bioorganic & Medicinal Chemistry Letters2 citations Open access
Semantic Scholar
Improved potency of pyridin-2(1H)one derivatives for the treatment of mechanical allodynia.
A. Visseq, Amélie Descheemaeker, Karine Hérault, F. Giraud +5 more
2021European journal of medicinal chemistry2 citations Open access
Semantic Scholar
Synthesis and kinase inhibitory potencies of new pyrido[3,4-g]quinazolines substituted at the 8-position
Y. Esvan, B. Josselin, B. Baratte, S. Bach +4 more
2020ARKIVOC1 citations Open access
Semantic Scholar
Synthesis and Biological Activities of 4‐Substituted Pyrrolo[2,3‐a]carbazole Pim Kinase Inhibitors.
F. Giraud, Rufine Akué-Gédu, L. Nauton, N. Candelon +4 more
20131 citations
Semantic Scholar
Recent developments in Haspin kinase inhibitors: Structure, synthesis and activities.
Killian Malosse, Elisabeth Pereira, F. Giraud, F. Anizon +1 more
2026Bioorganic & Medicinal Chemistry0 citations Open access
Semantic Scholar
Synthesis, anti-cancer activity, Pim-3 inhibitory potency and zebrafish larvae toxicity evaluation of indolopyrazolocarbazole derivatives
Théo Frazier, Elisabeth Pereira, Reidun Aesoy, A. Trentani +4 more
2026European Journal of Medicinal Chemistry Reports0 citations Open access
Semantic Scholar
Synthesis of 1H-Pyrrolo[3,2-g]isoquinoline Derivatives as Ligands Targeting Haspin Kinase
Killian Malosse, B. Josselin, S. Ruchaud, F. Anizon +2 more
2025Molecules0 citations
Semantic Scholar
Improved Synthesis and Preparation of Analogues of a Pain-Relieving Pyridin-2(1 H )-one
Théo Frazier, Pauline Murail, F. Giraud, A. Artola +3 more
2024Synthesis0 citations Open access
Semantic Scholar
Synthesis of diversely substituted pyridin-2(1H)-ones and in vivo evaluation of their anti-allodynic effect on cutaneous inflammatory mechanical allodynia.
Théo Frazier, Pauline Murail, Arthur Boulangé, Nazim Chalane +5 more
2024RSC Medicinal Chemistry0 citations Open access
Semantic Scholar
Synthesis of (2-Aminopyrimidin-4-yl)(pyridin-4-yl)methanone and Derivatives
F. Giraud, B. Josselin, S. Ruchaud, F. Anizon +1 more
2023Synthesis0 citations Open access
Semantic Scholar
CLK1 with bound pyridoquinazoline
M. Schroeder, H. Tazarki, Wael Zeinyeh, Y. Esvan +11 more
20190 citations
Semantic Scholar
Design and synthesis of new nitrogen-containing heterocycles for the treatment of mechanical allodynia.
A. Visseq, A. Descheemaeker, L. Nauton, V. Thery +5 more
20190 citations
Semantic Scholar
Structure of CLK1 with bound N-methyl-10-nitropyrido[3,4-g]quinazolin-2-amine
A. Joerger, D. Chatterjee, M. Schroeder, H. Tazarki +11 more
20190 citations
Semantic Scholar
Crystal structure of human CLK1 in complex with pyrido[3,4-g]quinazoline derivative ZW31 (compound 14)
A. Chaikuad, Y. Esvan, Wael Zeinyeh, T. Boibessot +12 more
20160 citations
Semantic Scholar
Crystal structure of human CLK1 in complex with pyrido[3,4-g]quinazoline derivative ZW29 (compound 13)
A. Chaikuad, Y. Esvan, Wael Zeinyeh, T. Boibessot +12 more
20160 citations
Semantic Scholar

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F. Anizon×39
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L. Nauton×14
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