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B. Szczepankiewicz · SciRah

Researcher profile · Semantic Scholar

B. Szczepankiewicz

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B. Szczepankiewicz — researcher profile on SciRah

h-index: 22
Works: 43
Citations: 1,956

Most-cited papers

Discovery of a potent, selective protein tyrosine phosphatase 1B inhibitor using a linked-fragment strategy.
B. Szczepankiewicz, Gang Liu, P. Hajduk, C. Abad-Zapatero +11 more
2003Journal of the American Chemical Society211 citations Open access
Semantic Scholar
Crystallographic structure of a small molecule SIRT1 activator-enzyme complex
H. Dai, A. Case, T. Riera, Thomas Considine +29 more
2014Nature Communications200 citations Open access
Semantic Scholar
Aminopyridine-based c-Jun N-terminal kinase inhibitors with cellular activity and minimal cross-kinase activity.
B. Szczepankiewicz, Christi Kosogof, L. Nelson, Gang Liu +22 more
2006Journal of Medicinal Chemistry164 citations Open access
Semantic Scholar
SIRT1 Activation by Small Molecules
H. Dai, Lauren Kustigian, David P. Carney, A. Case +7 more
2010Journal of Biological Chemistry119 citations Open access
Semantic Scholar
Selective protein tyrosine phosphatase 1B inhibitors: targeting the second phosphotyrosine binding site with non-carboxylic acid-containing ligands.
Gang Liu, Z. Xin, Heng Liang, C. Abad-Zapatero +12 more
2003Journal of Medicinal Chemistry102 citations Open access
Semantic Scholar
Inhibition of MptpB phosphatase from Mycobacterium tuberculosis impairs mycobacterial survival in macrophages.
Nicola J. Beresford, Debbie C. Mulhearn, B. Szczepankiewicz, Gang Liu +5 more
2009Journal of Antimicrobial Chemotherapy87 citations
Semantic Scholar
Potential drug targets and progress towards pharmacologic inhibition of hepatic glucose production.
Ravi Kurukulasuriya, J. T. Link, David J. Madar, Z. Pei +4 more
2003Current Medicinal Chemistry86 citations
Semantic Scholar
Isoxazole carboxylic acids as protein tyrosine phosphatase 1B (PTP1B) inhibitors.
Hongyu Zhao, Gang Liu, Z. Xin, Michael D. Serby +12 more
2004Bioorganic & Medicinal Chemistry Letters79 citations Open access
Semantic Scholar
Synthesis of carba-NAD and the structures of its ternary complexes with SIRT3 and SIRT5.
B. Szczepankiewicz, H. Dai, Karsten J. Koppetsch, Dong-Ming Qian +3 more
2012Journal of Organic Chemistry73 citations
Semantic Scholar
Discovery of piperidine-aryl urea-based stearoyl-CoA desaturase 1 inhibitors.
Z. Xin, Hongyu Zhao, Michael D. Serby, Bo Liu +12 more
2008Bioorganic & Medicinal Chemistry Letters70 citations Open access
Semantic Scholar
Discovery of potent, highly selective, and orally bioavailable pyridine carboxamide c-Jun NH2-terminal kinase inhibitors.
Hongyu Zhao, Michael D. Serby, Z. Xin, B. Szczepankiewicz +16 more
2006Journal of Medicinal Chemistry69 citations Open access
Semantic Scholar
New antimitotic agents with activity in multi-drug-resistant cell lines and in vivo efficacy in murine tumor models.
B. Szczepankiewicz, Gang Liu, H. Jae, A. Tasker +18 more
2001Journal of Medicinal Chemistry67 citations
Semantic Scholar
Inhibition of protein tyrosine phosphatase 1B as a potential treatment of diabetes and obesity.
Z. Pei, Gang Liu, T. Lubben, B. Szczepankiewicz
2004Current pharmaceutical design63 citations
Semantic Scholar
Discovery and structure-activity relationship of oxalylarylaminobenzoic acids as inhibitors of protein tyrosine phosphatase 1B.
Gang Liu, B. Szczepankiewicz, Z. Pei, D. Janowick +13 more
2003Journal of Medicinal Chemistry63 citations Open access
Semantic Scholar
Identification of a monoacid-based, cell permeable, selective inhibitor of protein tyrosine phosphatase 1B.
Z. Xin, Gang Liu, C. Abad-Zapatero, Z. Pei +10 more
2003Bioorganic & Medicinal Chemistry Letters54 citations Open access
Semantic Scholar
Prospects for pharmacologic inhibition of hepatic glucose production.
Ravi Kurukulasuriya, J. T. Link, David J. Madar, Z. Pei +4 more
2003Current Medicinal Chemistry50 citations
Semantic Scholar
Discovery and pharmacological evaluation of growth hormone secretagogue receptor antagonists.
Z. Xin, Michael D. Serby, Hongyu Zhao, Christi Kosogof +21 more
2006Journal of Medicinal Chemistry46 citations Open access
Semantic Scholar
Potent, selective inhibitors of protein tyrosine phosphatase 1B.
Z. Xin, T. Oost, C. Abad-Zapatero, P. Hajduk +9 more
2003Bioorganic & Medicinal Chemistry Letters45 citations Open access
Semantic Scholar
2,4-diaminopyrimidine derivatives as potent growth hormone secretagogue receptor antagonists.
Michael D. Serby, Hongyu Zhao, B. Szczepankiewicz, Christi Kosogof +19 more
2006Journal of Medicinal Chemistry39 citations Open access
Semantic Scholar
Potent and selective non-cysteine-containing inhibitors of protein farnesyltransferase.
David Augeri, Stephen J. O'Connor, Dave Janowick, B. Szczepankiewicz +10 more
1998Journal of Medicinal Chemistry36 citations Open access
Semantic Scholar
Synthesis of purines and other fused imidazoles from acyclic amidines and guanidines.
B. Szczepankiewicz, Jeffrey J. Rohde, Ravi Kurukulasuriya
2005Organic Letters35 citations Open access
Semantic Scholar
The Synthesis of Bromomethyltrifluoroborates through Continuous Flow Chemistry
T. Broom, M. Hughes, B. Szczepankiewicz, K. Ace +12 more
201426 citations
Semantic Scholar
A novel method for suppression of the abnormal Fischer indole synthesis
B. Szczepankiewicz, C. Heathcock
199722 citations
Semantic Scholar
Electrochemical Properties of Some Biologically Active Quinone Derivatives: Furanquinones, Pyridoquinones, and Diplamine, a Cytotoxic Pyridoacridine Alkaloid
P. W. Crawford, J. Gross, K. Lawson, C.-C. Cheng +5 more
199721 citations Open access
Semantic Scholar
Aminopyridine carboxamides as c-Jun N-terminal kinase inhibitors: targeting the gatekeeper residue and beyond.
Gang Liu, Hongyu Zhao, Bo Liu, Z. Xin +9 more
2006Bioorganic & Medicinal Chemistry Letters20 citations Open access
Semantic Scholar
Xanthine mimetics as potent dipeptidyl peptidase IV inhibitors.
Ravi Kurukulasuriya, Jeffrey J. Rohde, B. Szczepankiewicz, F. Basha +9 more
2006Bioorganic & Medicinal Chemistry Letters17 citations Open access
Semantic Scholar
Total Synthesis of Diplamine, a Cytotoxic Pyridoacridine Alkaloid from a Pacific Tunicate
B. Szczepankiewicz, C. Heathcock
199417 citations
Semantic Scholar
Structure-activity relationship studies on tetralin carboxamide growth hormone secretagogue receptor antagonists.
Hongyu Zhao, Z. Xin, J. Patel, L. Nelson +8 more
2005Bioorganic & Medicinal Chemistry Letters16 citations
Semantic Scholar
Sirtuin modulators: targets for metabolic diseases and beyond.
B. Szczepankiewicz, P. Ng
2008Current Topics in Medicinal Chemistry15 citations
Semantic Scholar
Optimization of 2,4-diaminopyrimidines as GHS-R antagonists: side chain exploration.
Bo Liu, Mei Liu, Z. Xin, Hongyu Zhao +11 more
2006Bioorganic & Medicinal Chemistry Letters13 citations Open access
Semantic Scholar
Frontiers in Medicinal Chemistry
Atta-ur-rahman, A. Reitz, M. Choudhary, C. P. Kordik +95 more
201612 citations Open access
Semantic Scholar
Aromatic heterocycle-based DPP-IV inhibitors: xanthines and related structural types.
B. Szczepankiewicz, Ravi Kurukulasuriya
2007Current Topics in Medicinal Chemistry10 citations
Semantic Scholar
One-step, nonenzymatic synthesis of O-acetyl-ADP-ribose and analogues from NAD and carboxylates.
B. Szczepankiewicz, Karsten J. Koppetsch, R. Perni
2011Journal of Organic Chemistry8 citations
Semantic Scholar
Total Synthesis of Diplamine, a Cytotoxic Pyridoacridine Alkaloid from a Pacific Tunicate.
B. Szczepankiewicz, C. Heathcock
19942 citations
Semantic Scholar
Potent, Selective Protein Tyrosine Phosphatase 1B Inhibitor Compound 12 Using a Linked-Fragment Strategy
B. Szczepankiewicz, G. Liu, P. Hajduk, C. Abad-Zapatero +11 more
20031 citations
Semantic Scholar
rat DPP-IV with xanthine mimetic inhibitor #7
Ravi Kurukulasuriya, Jeffrey J. Rohde, B. Szczepankiewicz, F. Basha +8 more
20060 citations
Semantic Scholar
Inhibition of Protein Tyrosine Phosphatase 1B for the Treatment of Diabetes and Obesity
Z. Pei, Gang Liu, T. Lubben, B. Szczepankiewicz
20060 citations
Semantic Scholar
PTP1B complexed with Isoxazole Carboxylic Acid
Hongyu Zhao, Gang Liu, Z. Xin, Michael D. Serby +12 more
20040 citations
Semantic Scholar
Pharmaceutical composition and their use as inhibitors of dipeptidyl peptidase IV (DPP-IV)
S. Djuric, H. Kopecká, Xiao-Fen Li, K. Longenecker +9 more
20030 citations
Semantic Scholar
DUAL-SITE POTENT, SELECTIVE PROTEIN TYROSINE PHOSPHATASE 1B INHIBITOR USING A LINKED FRAGMENT STRATEGY AND A MALONATE HEAD ON THE FIRST SITE
B. Szczepankiewicz, Gang Liu, P. Hajduk, C. Abad-Zapatero +6 more
20030 citations
Semantic Scholar
Oxalyl-Aryl-Amino Benzoic Acid inhibitors of PTP1B, compound 17
Gang Liu, B. Szczepankiewicz, Z. Pei, D. A. Janowich +13 more
20030 citations
Semantic Scholar
Non-carboxylic Acid-Containing Inhibitor of PTP1B Targeting the Second Phosphotyrosine Site
Gang Liu, Z. Xin, Heng Liang, C. Abad-Zapatero +6 more
20030 citations
Semantic Scholar
A Novel Method for Suppression of the Abnormal Fischer Indole Synthesis.
B. Szczepankiewicz, C. Heathcock
19970 citations
Semantic Scholar

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