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J. Pawluczyk · SciRah

Researcher profile · Semantic Scholar

J. Pawluczyk

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J. Pawluczyk — researcher profile on SciRah

h-index: 11
Works: 30
Citations: 532

Most-cited papers

Synthesis of Cyclobutane-Fused Tetracyclic Scaffolds via Visible-Light Photocatalysis for Building Molecular Complexity.
Martins S Oderinde, Edna Mao, Antonio Ramirez, J. Pawluczyk +10 more
2020Journal of the American Chemical Society99 citations Open access
Semantic Scholar
Photocatalytic Dearomative Intermolecular [2 + 2] Cycloaddition of Heterocycles for Building Molecular Complexity.
Martins S Oderinde, Antonio Ramirez, T. Dhar, Lyndon A. M. Cornelius +8 more
2020Journal of Organic Chemistry53 citations Open access
Semantic Scholar
1-(1-[4-[(N-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]piperidin-4- yl)-4H-3,1-benzoxazin-2(1H)-one (L-371,257): a new, orally bioavailable, non-peptide oxytocin antagonist.
P. D. Williams, B. Clineschmidt, J. M. Erb, R. Freidinger +6 more
1995Journal of Medicinal Chemistry49 citations Open access
Semantic Scholar
Development of orally active oxytocin antagonists: studies on 1-(1-[4-[1-(2-methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl]piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and related pyridines.
I. M. Bell, J. M. Erb, R. Freidinger, S. N. Gallicchio +15 more
1998Journal of Medicinal Chemistry48 citations Open access
Semantic Scholar
Design and synthesis of a pro-drug of vinblastine targeted at treatment of prostate cancer with enhanced efficacy and reduced systemic toxicity.
S. F. Brady, J. Pawluczyk, P. Lumma, D. Feng +9 more
2002Journal of Medicinal Chemistry47 citations
Semantic Scholar
A prostate-specific antigen (PSA)-activated vinblastine prodrug selectively kills PSA-secreting cells in vivo.
D. Defeo-jones, S. F. Brady, D. Feng, Brad Wong +16 more
2002Molecular Cancer Therapeutics46 citations
Semantic Scholar
Discovery of (S)-1-((2',6-Bis(difluoromethyl)-[2,4'-bipyridin]-5-yl)oxy)-2,4-dimethylpentan-2-amine (BMS-986176/LX-9211): A Highly Selective, CNS Penetrable, and Orally Active Adaptor Protein-2 Associated Kinase 1 Inhibitor in Clinical Trials for the Treatment of Neuropathic Pain.
Guang-Lin Luo, Ling Chen, W. Kostich, Brian D. Hamman +55 more
2022Journal of Medicinal Chemistry28 citations Open access
Semantic Scholar
Nanomolar-affinity, non-peptide oxytocin receptor antagonists.
B. E. Evans, G. F. Lundell, K. F. Gilbert, M. Bock +6 more
1993Journal of Medicinal Chemistry24 citations Open access
Semantic Scholar
Microwave-initiated living free radical polymerization: optimization of the preparative scale synthesis of Rasta resins
J. Pawluczyk, R. McClain, C. Denicola, James Mulhearn +2 more
200720 citations
Semantic Scholar
1-(((7,7-Dimethyl-2(S)-(2(S)-amino-4-(methylsulfonyl)butyramido) bicyclo(2.2.1)heptan-1(S)-yl)methyl)sulfonyl)-4-(2-methylphenyl) piperazine (L-368,899): An Orally Bioavailable, Non-Peptide Oxytocin Antagonist with Potential Utility for Managing Preterm Labor.
P. D. Williams, P. Anderson, R. Ball, M. Bock +15 more
199416 citations
Semantic Scholar
Intramolecular [2+2] Cycloaddition of N-Allylcinnamamines and N -Allylcinnamamides by Visible-Light Photocatalysis
Martins S Oderinde, J. Kempson, Daniel J. Smith, N. Meanwell +9 more
2019Annalen der Pharmacie15 citations
Semantic Scholar
Process Development of a Macrocyclic Peptide Inhibitor of PD-L1.
Subha Mukherjee, Amanda J. Rogers, Gardner S. Creech, Chao Hang +14 more
2024Journal of Organic Chemistry9 citations
Semantic Scholar
Applications of microwave-assisted organic synthesis on the multigram scale.
S. Wolkenberg, W. Shipe, C. Lindsley, J. Guare +1 more
2005Current opinion in drug discovery & development9 citations
Semantic Scholar
1‐(1‐(4‐((N‐Acetyl‐4‐piperidinyl)oxy)‐2‐methoxybenzoyl)piperidin‐4‐yl)‐ 4H‐3,1‐benzoxazin‐2(1H)‐one (L‐371,257): A New, Orally Bioavailable, Non‐Peptide Oxytocin Antagonist.
P. D. Williams, B. Clineschmidt, J. M. Erb, R. Freidinger +7 more
19969 citations
Semantic Scholar
Challenges with the Synthesis of a Macrocyclic Thioether Peptide: From Milligram to Multigram Using Solid Phase Peptide Synthesis (SPPS).
J. Kempson, Rulin Zhao, J. Pawluczyk, Bei Wang +17 more
2024Journal of Organic Chemistry7 citations
Semantic Scholar
A Stereocontrolled Synthesis of a Phosphorothioate Cyclic Dinucleotide-Based STING Agonist.
J. Kempson, Huiping Zhang, Xiaoping Hou, Lyndon A. M. Cornelius +20 more
2021Journal of Organic Chemistry7 citations
Semantic Scholar
Driving Potency with Rotationally Stable Atropisomers: Discovery of Pyridopyrimidinedione-Carbazole Inhibitors of BTK.
A. Srivastava, Soo S. Ko, Scott H. Watterson, M. Pattoli +31 more
2020ACS Medicinal Chemistry Letters7 citations Open access
Semantic Scholar
Synthesis of 1-(tert-Butyl) 4-Methyl (1R,2S,4R)-2-Methylcyclohexane-1,4-Dicarboxylate from Hagemann's tert-Butyl Ester for an Improved Synthesis of BMS-986251.
Lyndon A. M. Cornelius, Jianqing Li, Daniel J. Smith, Subramaniam Krishnananthan +10 more
2020Journal of Organic Chemistry7 citations
Semantic Scholar
Development of the Large-Scale Synthesis of Tetrahydropyran Glycine, a Precursor to the HCV NS5A Inhibitor BMS-986097.
A. Mathur, Bei Wang, Daniel J. Smith, Jianqing Li +22 more
2017Journal of Organic Chemistry7 citations
Semantic Scholar
Development of a Rapid Scale-Up Synthesis of (S)-N-(8-((2-Amino-2,4-dimethylpentyl)oxy)-5H-chromeno[3,4-c]pyridin-2-yl)acetamide, a Potent Adaptor-Associated Kinase 1 Inhibitor
Jianqing Li, Daniel J. Smith, J. Pawluczyk, Subramaniam Krishnananthan +13 more
2022Organic Process Research & Development6 citations
Semantic Scholar
Synthesis Optimization, Scale-Up, and Catalyst Screening Efforts toward the MGAT2 Clinical Candidate, BMS-963272
J. Kempson, Xiaoping Hou, Jung-Hui Sun, Michael K Wong +18 more
2022Organic Process Research & Development5 citations
Semantic Scholar
Long-Acting Tumor-Activated Prodrug of a TGFβR Inhibitor.
Yong Zhang, Karen E Parrish, D. Tortolani, M. Poss +17 more
2021Journal of Medicinal Chemistry5 citations
Semantic Scholar
A mild and readily scalable procedure for the N-1-difluoromethylation of ethyl 6-((tert-butyldiphenylsilyl)oxy)-1H-indazole-3-carboxylate and its applications to the N-difluoromethylation of indazole, benzotriazole, imidazole, indole and pyrazole derivatives
Zhenqiu Hong, Xiaoping Hou, Ru-Lin Zhao, Jianqing Li +7 more
2020Journal of fluorine chemistry4 citations
Semantic Scholar
Route evaluation and development of a practical synthesis of methyl (S)-2-chloro-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine-7-carboxylate
J. Pawluczyk, J. Kempson, A. Mathur, Martins S Oderinde
20202 citations
Semantic Scholar
Orally active, non-peptide oxytocin antagonists
P. D. Williams, R. Ball, M. Bock, L. Carroll +17 more
19942 citations
Semantic Scholar
Discovery of BMS-986449: A Potent, Selective Degrader of the Transcription Factors IKZF2 (Helios) and IKZF4 (Eos) to Target Regulatory T Cells in Solid Tumors.
E. Cherney, S. Nair, Suresh Babu Viswa Krishna Penmetsa, Bharat Shimpukade +75 more
2026Journal of Medicinal Chemistry1 citations
Semantic Scholar
Efficient and Scalable Diastereoselective Synthesis of ((2R,7aS)-2-fluorotetrahydro-1H-pyrrolizin-7a(5H)-yl)methanol Hydrochloride
Rulin Zhao, Zhenqiu Hong, Bei Wang, Daniel J. Smith +11 more
2025Organic Process Research & Development1 citations
Semantic Scholar
Large-scale purification of a deprotected macrocyclic peptide by supercritical fluid chromatography (SFC) integrated with liquid chromatography in discovery chemistry.
Peng Li, Dauh-Rurng Wu, S. Yip, Dawn Sun +4 more
2024Journal of Chromatography A1 citations
Semantic Scholar
Cover Feature: Intramolecular [2+2] Cycloaddition of N-Allylcinnamamines and N -Allylcinnamamides by Visible-Light Photocatalysis (Eur. J. Org. Chem. 1/2020)
Martins S Oderinde, J. Kempson, Daniel J. Smith, N. Meanwell +9 more
2019Annalen der Pharmacie0 citations
Semantic Scholar
Antagonistes recepteurs d'oxytocine tocolytique
Ben E. Evans, D. W. Hobbs, J. Pawluczyk, Douglas J. Pettibone +2 more
19930 citations
Semantic Scholar

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