Discovery of TBC11251, a potent, long acting, orally active endothelin receptor-A selective antagonist.
Cheng-De Wu, M. Chan, F. Stavros, B. Raju +6 more
Researcher profile · Semantic Scholar
Cheng-De Wu, M. Chan, F. Stavros, B. Raju +6 more
Jessica Jones, Schonna R. Manning, Morela Montoya, Karin M. Keller +1 more
H. Gong, B. Rambo, E. Karnas, V. Lynch +2 more
T. Kogan, B. Dupré, Karin M. Keller, I. L. Scott +6 more
Clint D. J. Tavares, J. O'Brien, O. Abramczyk, Ashwini K. Devkota +10 more
H. Gong, B. Rambo, V. Lynch, Karin M. Keller +1 more
Karin M. Keller, Junmei Zhang, Leon P. Oehlers, J. Brodbelt
Karin M. Keller, Megan M Breeden, Junmei Zhang, A. Ellington +1 more
B. Dupré, Huong Bui, I. L. Scott, Robert V. Market +3 more
Cheng-De Wu, E. Decker, N. Blok, Jian Li +9 more
H. Gong, B. Rambo, V. Lynch, Karin M. Keller +1 more
Y.-J. Xue, Brian Melo, M. Vallejo, Yuwen Zhao +3 more
Karin M. Keller, J. Brodbelt, R. Hettich, G. V. Van Berkel
Cheryl J. Bartleson, E. López, S. Unger, Karin M. Keller
Cheng-Du Wu, N. Blok, T. Kogan, Karin M. Keller +1 more
T. Kogan, B. Dupré, I. L. Scott, Huong Bui +3 more