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P. Cotelle · SciRah

Researcher profile · Semantic Scholar

P. Cotelle

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P. Cotelle — researcher profile on SciRah

h-index: 28
Works: 121
Citations: 2,328

Most-cited papers

Oleuropein and derivatives from olives as Tau aggregation inhibitors.
Anthony Daccache, C. Lion, N. Sibille, M. Gérard +3 more
2011Neurochemistry International166 citations
Semantic Scholar
Magnesium chelating 2-hydroxyisoquinoline-1,3(2H,4H)-diones, as inhibitors of HIV-1 integrase and/or the HIV-1 reverse transcriptase ribonuclease H domain: discovery of a novel selective inhibitor of the ribonuclease H function.
M. Billamboz, Fabrice Bailly, C. Lion, Nadia Touati +6 more
2011Journal of Medicinal Chemistry121 citations Open access
Semantic Scholar
Design, synthesis, and biological evaluation of a series of 2-hydroxyisoquinoline-1,3(2H,4H)-diones as dual inhibitors of human immunodeficiency virus type 1 integrase and the reverse transcriptase RNase H domain.
M. Billamboz, Fabrice Bailly, M. L. Barreca, L. De Luca +7 more
2008Journal of Medicinal Chemistry115 citations Open access
Semantic Scholar
Targeting Transcriptional Enhanced Associate Domains (TEADs).
Floriane Gibault, M. Sturbaut, Fabrice Bailly, Patricia Melnyk +1 more
2017Journal of Medicinal Chemistry93 citations Open access
Semantic Scholar
Non-Photoinduced Biological Properties of Verteporfin.
Floriane Gibault, Matthieu Corvaisier, Fabrice Bailly, G. Huet +2 more
2016Current Medicinal Chemistry91 citations
Semantic Scholar
Reaction of rosmarinic acid with nitrite ions in acidic conditions: discovery of nitro- and dinitrorosmarinic acids as new anti-HIV-1 agents.
M. Dubois, Fabrice Bailly, G. Mbemba, J. Mouscadet +3 more
2008Journal of Medicinal Chemistry83 citations Open access
Semantic Scholar
Molecular Features of the YAP Inhibitor Verteporfin: Synthesis of Hexasubstituted Dipyrrins as Potential Inhibitors of YAP/TAZ, the Downstream Effectors of the Hippo Pathway
Floriane Gibault, Fabrice Bailly, Matthieu Corvaisier, Mathilde Coevoet +3 more
2017ChemMedChem72 citations
Semantic Scholar
Anti-HIV activities of natural antioxidant caffeic acid derivatives: toward an antiviral supplementation diet.
Fabrice Bailly, P. Cotelle
2005Current Medicinal Chemistry72 citations
Semantic Scholar
Bistramides A, B, C, D, and K: a new class of bioactive cyclic polyethers from Lissoclinum bistratum.
J. Biard, C. Roussakis, J. Kornprobst, D. Gouiffes-Barbin +5 more
1994Journal of Natural Products64 citations
Semantic Scholar
Antioxidant properties of 3-hydroxycoumarin derivatives.
Fabrice Bailly, C. Maurin, E. Teissier, H. Vezin +1 more
2004Bioorganic & Medicinal Chemistry59 citations
Semantic Scholar
2-hydroxyisoquinoline-1,3(2H,4H)-diones as inhibitors of HIV-1 integrase and reverse transcriptase RNase H domain: influence of the alkylation of position 4.
M. Billamboz, Fabrice Bailly, C. Lion, C. Calmels +7 more
2011European journal of medicinal chemistry58 citations Open access
Semantic Scholar
Inhibition of hepatitis B virus replication by N-hydroxyisoquinolinediones and related polyoxygenated heterocycles
Tiffany C. Edwards, E. Lomonosova, Jenny A. Patel, Qi-Lan Li +8 more
2017Antiviral Research54 citations Open access
Semantic Scholar
Progress with YAP/TAZ-TEAD inhibitors: a patent review (2018-present)
Benjamin Zagiel, Patricia Melnyk, P. Cotelle
2022Expert Opinion on Therapeutic Patents51 citations
Semantic Scholar
The NSP14/NSP10 RNA repair complex as a Pan-coronavirus therapeutic target
G. Róna, A. Zeke, Bearach Miwatani-Minter, Maren de Vries +13 more
2021Cell Death and Differentiation50 citations Open access
Semantic Scholar
4-Substituted 2-Hydroxyisoquinoline-1,3(2H,4H)-diones as a Novel Class of HIV-1 Integrase Inhibitors.
M. Billamboz, Virginie Suchaud, Fabrice Bailly, C. Lion +6 more
2013ACS Medicinal Chemistry Letters45 citations Open access
Semantic Scholar
Improved preparation and structural investigation of 4-aryl-4-oxo-2-hydroxy-2-butenoic acids and methyl esters
C. Maurin, Fabrice Bailly, P. Cotelle
200444 citations
Semantic Scholar
Toward the Discovery of a Novel Class of YAP–TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP–TEAD Protein–Protein Interface
Floriane Gibault, Mathilde Coevoet, M. Sturbaut, A. Farce +13 more
2018Cancers42 citations Open access
Semantic Scholar
Patented HIV-1 integrase inhibitors (1998-2005).
P. Cotelle
2006Recent Patents on Anti-Infective Drug Discovery42 citations
Semantic Scholar
Crosstalk between the Hippo Pathway and the Wnt Pathway in Huntington’s Disease and Other Neurodegenerative Disorders
Pasquale Sileo, C. Simonin, Patricia Melnyk, M. Chartier-Harlin +1 more
2022Cells40 citations Open access
Semantic Scholar
Development of a series of 3-hydroxyquinolin-2(1H)-ones as selective inhibitors of HIV-1 reverse transcriptase associated RNase H activity.
Virginie Suchaud, Fabrice Bailly, C. Lion, E. Tramontano +5 more
2012Bioorganic & Medicinal Chemistry Letters40 citations Open access
Semantic Scholar
Discovery of a cryptic site at the interface 2 of TEAD - Towards a new family of YAP/TAZ-TEAD inhibitors.
M. Sturbaut, Fabrice Bailly, Mathilde Coevoet, Pasquale Sileo +10 more
2021European journal of medicinal chemistry37 citations Open access
Semantic Scholar
Spectroscopic studies of diketoacids-metal interactions. A probing tool for the pharmacophoric intermetallic distance in the HIV-1 integrase active site.
C. Maurin, Fabrice Bailly, E. Buisine, H. Vezin +3 more
2004Journal of Medicinal Chemistry35 citations Open access
Semantic Scholar
Synthesis and biological activities of a series of 4,5-diaryl-3-hydroxy-2(5H)-furanones.
Fabrice Bailly, C. Queffélec, G. Mbemba, J. Mouscadet +4 more
2008European journal of medicinal chemistry29 citations Open access
Semantic Scholar
Synthesis and antiviral properties of some polyphenols related to Salvia genus.
C. Queffélec, Fabrice Bailly, G. Mbemba, J. Mouscadet +4 more
2008Bioorganic & Medicinal Chemistry Letters28 citations Open access
Semantic Scholar
Synthesis and HIV-1 integrase inhibitory activities of caffeic acid dimers derived from Salvia officinalis.
Fabrice Bailly, C. Queffélec, G. Mbemba, J. Mouscadet +1 more
2005Bioorganic & Medicinal Chemistry Letters28 citations Open access
Semantic Scholar
Nitration of Electron-Rich Aromatic Compounds by Cerium Ammonium Nitrate Coated on Silica
Jean-Luc Grenier, J. Catteau, P. Cotelle
199928 citations
Semantic Scholar
Synthesis and antioxidant properties of a new lipophilic ascorbic acid analogue.
P. Cotelle, N. Cotelle, E. Teissier, H. Vezin
2003Bioorganic & Medicinal Chemistry27 citations
Semantic Scholar
2-Hydroxyisoquinoline-1,3(2H,4H)-diones (HIDs), novel inhibitors of HIV integrase with a high barrier to resistance.
Belete A. Desimmie, J. Demeulemeester, Virginie Suchaud, O. Taltynov +7 more
2013ACS Chemical Biology25 citations
Semantic Scholar
Reaction of caffeic acid derivatives with acidic nitrite
P. Cotelle, H. Vezin
200125 citations
Semantic Scholar
The total synthesis of salvianolic acid F
V. Dalla, P. Cotelle
199924 citations
Semantic Scholar
Chemocontrolled reduction of aromatic α-ketoesters by NaBH4: Selective synthesis of α-hydroxy esters or 1,2-diols
V. Dalla, P. Cotelle, J. Catteau
199724 citations
Semantic Scholar
Toward the Design of Ligands Selective for the C-Terminal Domain of TEADs.
Maxime Liberelle, Florine Toulotte, N. Renault, M. Gelin +4 more
2022Journal of Medicinal Chemistry23 citations Open access
Semantic Scholar
Investigation of a novel series of 2-hydroxyisoquinoline-1,3(2H,4H)-diones as human immunodeficiency virus type 1 integrase inhibitors.
Virginie Suchaud, Fabrice Bailly, C. Lion, C. Calmels +4 more
2014Journal of Medicinal Chemistry22 citations Open access
Semantic Scholar
A Convenient Synthesis of Substituted 2-Phenylnaphthalenes From Phenylacetones
P. Cotelle, J. Catteau
199721 citations
Semantic Scholar
General Synthesis of 2,3-Substituted 5-Membered Heterocyclic Quinones
M. Cherif, P. Cotelle, J. Catteau
199219 citations Open access
Semantic Scholar
Design, synthesis, and anti-integrase activity of catechol-DKA hybrids.
C. Maurin, Fabrice Bailly, G. Mbemba, J. Mouscadet +1 more
2006Bioorganic & Medicinal Chemistry18 citations
Semantic Scholar
An expeditious synthesis of polyhydroxylated 2-arylbenzo[b]furans
R. Dupont, P. Cotelle
200118 citations
Semantic Scholar
New bis-catechols 5-lipoxygenase inhibitors.
R. Dupont, J. Goossens, N. Cotelle, L. Vrielynck +3 more
2001Bioorganic & Medicinal Chemistry17 citations
Semantic Scholar
Antiproliferative and apoptotic effects of the oxidative dimerization product of methyl caffeate on human breast cancer cells.
Fabrice Bailly, R. Toillon, Olympe Tomavo, N. Jouy +2 more
2013Bioorganic & Medicinal Chemistry Letters16 citations
Semantic Scholar
Ceric Ammonium Nitrate in Organic Synthesis. II. Oxidation of N,N-Dimethyl Methoxyphenylmethylamines to Methoxybenzaldehydes
I. Badea, P. Cotelle, J. Catteau
199416 citations
Semantic Scholar
Lissoclimides, Cytotoxic Diterpenes from Lissoclinum voeltzkowi Michaelsen
Jean-François Biard, C. Malochet-Grivois, C. Roussakis, P. Cotelle +3 more
199415 citations
Semantic Scholar
The preclinical discovery and development of dolutegravir for the treatment of HIV
Fabrice Bailly, P. Cotelle
2015Expert Opinion on Drug Discovery14 citations
Semantic Scholar
Reaction of aryl-2-hydroxypropenoic derivatives with boron tribromide
R. Dupont, P. Cotelle
200114 citations
Semantic Scholar
Design, Synthesis and Evaluation of a Series of 1,5‐Diaryl‐1,2,3‐triazole‐4‐carbohydrazones as Inhibitors of the YAP‐TAZ/TEAD Complex
Floriane Gibault, M. Sturbaut, Mathilde Coevoet, M. Pugnière +9 more
2021ChemMedChem13 citations
Semantic Scholar
Evaluation of aldose reductase inhibition and docking studies of 6'-nitro and 6',6''-dinitrorosmarinic acids.
Catherine Koukoulitsa, Fabrice Bailly, K. Pegklidou, V. Demopoulos +1 more
2010European journal of medicinal chemistry13 citations Open access
Semantic Scholar
NMR study of five N-terminal peptide fragments of the vasoactive intestinal peptide: crucial role of aromatic residues.
J. Goossens, P. Cotelle, P. Chavatte, J. Hénichart
1996Peptide research13 citations
Semantic Scholar
2-hydroxyisoquinoline-1,3(2H,4H)-diones (HIDs) as human immunodeficiency virus type 1 integrase inhibitors: Influence of the alkylcarboxamide substitution of position 4.
M. Billamboz, Virginie Suchaud, Fabrice Bailly, C. Lion +4 more
2016European journal of medicinal chemistry12 citations Open access
Semantic Scholar
Reaction of arylethanals with boron tribromide
R. Dupont, P. Cotelle
199812 citations
Semantic Scholar
Towards the first synthesis of salvianolic acid F: An unexpected intramolecular Diels-Alder cyclisation
V. Dalla, P. Cotelle
199812 citations
Semantic Scholar
Development of LM-41 and AF-2112, two flufenamic acid-derived TEAD inhibitors obtained through the replacement of the trifluoromethyl group by aryl rings.
Ahmed Fnaiche, L. Mélin, N. G. Suárez, A. Paquin +15 more
2023Bioorganic & Medicinal Chemistry Letters11 citations Open access
Semantic Scholar

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Fabrice Bailly×28
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Fabrice Bailly — researcher profile on SciRah
Z. Debyser×10
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Patricia Melnyk×9
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Patricia Melnyk — researcher profile on SciRah
C. Lion×8
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F. Christ — researcher profile on SciRah

J. Mouscadet×7

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M. Billamboz×6

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M. Billamboz — researcher profile on SciRah

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H. Vezin — researcher profile on SciRah

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M. Andreola — researcher profile on SciRah

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G. Mbemba — researcher profile on SciRah

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C. Calmels — researcher profile on SciRah

Floriane Gibault×5

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