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A. Farce · SciRah

Researcher profile · Semantic Scholar

A. Farce

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A. Farce — researcher profile on SciRah

h-index: 26
Works: 90
Citations: 2,349

Most-cited papers

Intestinal antiinflammatory effect of 5-aminosalicylic acid is dependent on peroxisome proliferator–activated receptor-γ
C. Rousseaux, B. Lefebvre, L. Dubuquoy, P. Lefebvre +12 more
2005Journal of Experimental Medicine541 citations Open access
Semantic Scholar
Targeting peroxisome proliferator-activated receptors (PPARs): development of modulators.
Céline Pirat, A. Farce, N. Lebègue, N. Renault +7 more
2012Journal of Medicinal Chemistry180 citations Open access
Semantic Scholar
Novel 4-oxo-1,4-dihydroquinoline-3-carboxamide derivatives as new CB2 cannabinoid receptors agonists: synthesis, pharmacological properties and molecular modeling.
E. Stern, G. Muccioli, R. Millet, J. Goossens +6 more
2006Journal of Medicinal Chemistry81 citations Open access
Semantic Scholar
Switching invariant natural killer T (iNKT) cell response from anticancerous to anti-inflammatory effect: molecular bases.
Xavier Laurent, B. Bertin, N. Renault, A. Farce +6 more
2014Journal of Medicinal Chemistry68 citations Open access
Semantic Scholar
Impact of aryloxy-linked quinazolines: a novel series of selective VEGFR-2 receptor tyrosine kinase inhibitors.
A. Garofalo, L. Goossens, Perrine Six, A. Lemoine +3 more
2011Bioorganic & Medicinal Chemistry Letters67 citations Open access
Semantic Scholar
[4-(6,7-Disubstituted quinazolin-4-ylamino)phenyl] carbamic acid esters: a novel series of dual EGFR/VEGFR-2 tyrosine kinase inhibitors
A. Garofalo, L. Goossens, A. Lemoine, Séverine Ravez +4 more
201158 citations
Semantic Scholar
Synthesis and structure-activity relationships of (aryloxy)quinazoline ureas as novel, potent, and selective vascular endothelial growth factor receptor-2 inhibitors.
A. Garofalo, A. Farce, Séverine Ravez, A. Lemoine +4 more
2012Journal of Medicinal Chemistry53 citations Open access
Semantic Scholar
Functional genomics uncovers the transcription factor BNC2 as required for myofibroblastic activation in fibrosis
Marie Bobowski-Gérard, Clémence Boulet, F. P. Zummo, Julie Dubois-Chevalier +34 more
2022Nature Communications44 citations Open access
Semantic Scholar
Structural Insight into PPAR? Ligands Binding
A. Farce, N. Renault, P. Chavatte
200944 citations
Semantic Scholar
Journal of Enzyme Inhibition and Medicinal Chemistry
A. Durand, A. Farce, P. Carato, Sebastien Dilly Said Yous +2 more
44 citations
Semantic Scholar
In vitro and in silico hormonal activity studies of di‐(2‐ethylhexyl)terephthalate, a di‐(2‐ethylhexyl)phthalate substitute used in medical devices, and its metabolites
N. Kambia, I. Séverin, A. Farce, E. Moreau +5 more
2019Journal of Applied Toxicology43 citations Open access
Semantic Scholar
Toward the Discovery of a Novel Class of YAP–TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP–TEAD Protein–Protein Interface
Floriane Gibault, Mathilde Coevoet, M. Sturbaut, A. Farce +13 more
2018Cancers42 citations Open access
Semantic Scholar
Studies on indolizines. Evaluation of their biological properties as microtubule-interacting agents and as melanoma targeting compounds.
A. Ghinet, Cristina-Maria Abuhaie, P. Gautret, B. Rigo +4 more
2015European journal of medicinal chemistry40 citations
Semantic Scholar
Docking Study of Ligands into the Colchicine Binding Site of Tubulin
A. Farce, C. Logé, S. Gallet, N. Lebègue +4 more
2004Journal of Enzyme Inhibition and Medicinal Chemistry39 citations Open access
Semantic Scholar
Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel Disease.
Germain Homerin, S. Jawhara, X. Dezitter, Davy Baudelet +18 more
2020Journal of Medicinal Chemistry35 citations Open access
Semantic Scholar
New farnesyltransferase inhibitors in the phenothiazine series.
Dalila Belei, Carmen Dumea, Alexandrina Samson, A. Farce +3 more
2012Bioorganic & Medicinal Chemistry Letters35 citations Open access
Semantic Scholar
Synthesis and anticancer activity of analogues of phenstatin, with a phenothiazine A-ring, as a new class of microtubule-targeting agents.
Cristina-Maria Abuhaie, E. Bîcu, B. Rigo, P. Gautret +4 more
2013Bioorganic & Medicinal Chemistry Letters32 citations
Semantic Scholar
Molecular modelling of phthalates – PPARs interactions
N. Kambia, N. Renault, S. Dilly, A. Farce +5 more
2008Journal of Enzyme Inhibition and Medicinal Chemistry32 citations Open access
Semantic Scholar
New piperazine multi-effect drugs prevent neurofibrillary degeneration and amyloid deposition, and preserve memory in animal models of Alzheimer's disease.
N. Sergeant, V. Vingtdeux, S. Eddarkaoui, Marion Gay +17 more
2019Neurobiology of Disease29 citations Open access
Semantic Scholar
New indolizine-chalcones as potent inhibitors of human farnesyltransferase: Design, synthesis and biological evaluation.
Iuliana-Monica Moise, A. Ghinet, Dalila Belei, J. Dubois +2 more
2016Bioorganic & Medicinal Chemistry Letters28 citations Open access
Semantic Scholar
Synthesis and biological evaluation of fluoro analogues of antimitotic phenstatin.
A. Ghinet, A. Tourteau, B. Rigo, Vivien Stocker +4 more
2013Bioorganic & Medicinal Chemistry28 citations
Semantic Scholar
Synthesis and radioligand binding studies of bis-isoquinolinium derivatives as small conductance Ca(2+)-activated K(+) channel blockers.
Amaury Graulich, S. Dilly, A. Farce, J. Scuvée-Moreau +5 more
2007Journal of Medicinal Chemistry28 citations Open access
Semantic Scholar
Design, synthesis and biological evaluation of substituted dioxodibenzothiazepines and dibenzocycloheptanes as farnesyltransferase inhibitors.
P. Gilleron, Nicolas Wlodarczyk, R. Houssin, A. Farce +6 more
2007Bioorganic & Medicinal Chemistry Letters28 citations Open access
Semantic Scholar
Studies on phenothiazines: New microtubule-interacting compounds with phenothiazine A-ring as potent antineoplastic agents.
A. Ghinet, Iuliana-Monica Moise, B. Rigo, Germain Homerin +3 more
2016Bioorganic & Medicinal Chemistry26 citations Open access
Semantic Scholar
Quinazoline-urea, new protein kinase inhibitors in treatment of prostate cancer
A. Garofalo, L. Goossens, A. Lemoine, A. Farce +2 more
2010Journal of Enzyme Inhibition and Medicinal Chemistry26 citations Open access
Semantic Scholar
Homology modeling of MT1 and MT2 receptors.
A. Farce, A. Chugunov, C. Logé, Ahmed Sabaouni +7 more
2008European journal of medicinal chemistry26 citations
Semantic Scholar
Comparative Effects of Di-(2-ethylhexyl)phthalate and Di-(2-ethylhexyl)terephthalate Metabolites on Thyroid Receptors: In Vitro and In Silico Studies
N. Kambia, I. Séverin, A. Farce, L. Dahbi +4 more
2021Metabolites25 citations Open access
Semantic Scholar
Novel indolizine derivatives with unprecedented inhibitory activity on human farnesyltransferase.
Carmen Dumea, Dalila Belei, A. Ghinet, J. Dubois +2 more
2014Bioorganic & Medicinal Chemistry Letters24 citations Open access
Semantic Scholar
Synthesis and biological evaluation of a new series of phenothiazine-containing protein farnesyltransferase inhibitors.
Cristina-Maria Abuhaie, A. Ghinet, A. Farce, J. Dubois +4 more
2013European journal of medicinal chemistry24 citations Open access
Semantic Scholar
2,6-Diphenylthiazolo[3,2-b][1,2,4]triazoles as telomeric G-quadruplex stabilizers.
Jamal El Bakali, Frédérique Klupsch, A. Guédin, B. Brassart +9 more
2009Bioorganic & Medicinal Chemistry Letters24 citations
Semantic Scholar
Chlorinated and brominated bisphenol A derivatives: Synthesis, characterization and determination in water samples.
Manon Doumas, Steeve Rouillon, N. Venisse, Cédric Nadeau +6 more
2018Chemosphere22 citations
Semantic Scholar
Docking study: PPARs interaction with the selected alternative plasticizers to di(2-ethylhexyl) phthalate
N. Kambia, A. Farce, K. Belarbi, B. Gressier +3 more
2015Journal of Enzyme Inhibition and Medicinal Chemistry22 citations Open access
Semantic Scholar
Synthesis, antiproliferative activity and tubulin targeting effect of acridinone and dioxophenothiazine derivatives.
V. Vérones, N. Flouquet, M. Lecoeur, A. Lemoine +8 more
2013European journal of medicinal chemistry22 citations
Semantic Scholar
Intestinal antiinﬂammatory effect of 5-aminosalicylic acid is dependent on peroxisome proliferator–activated receptor- (cid:1)
C. Rousseaux, B. Lefebvre, L. Dubuquoy, P. Lefebvre +12 more
200521 citations
Semantic Scholar
Indolizine-phenothiazine hybrids as the first dual inhibitors of tubulin polymerization and farnesyltransferase with synergistic antitumor activity.
Iuliana-Monica Moise, E. Bîcu, A. Farce, J. Dubois +1 more
2020Bioorganic chemistry (Print)20 citations
Semantic Scholar
Synthesis and biological evaluation of thiophene and benzo[b]thiophene analogs of combretastatin A-4 and isocombretastatin A-4: A comparison between the linkage positions of the 3,4,5-trimethoxystyrene unit.
Cong Viet Do, Abdelfattah Faouzi, Caroline Barette, A. Farce +7 more
2016Bioorganic & Medicinal Chemistry Letters20 citations
Semantic Scholar
Virtual Screening of CB2 Receptor Agonists from Bayesian Network and High‐Throughput Docking: Structural Insights into Agonist‐Modulated GPCR Features
N. Renault, Xavier Laurent, A. Farce, Jamal El Bakali +6 more
2013Chemical Biology and Drug Design20 citations Open access
Semantic Scholar
Synthesis and biological evaluation of new phenothiazine derivatives bearing a pyrazole unit as protein farnesyltransferase inhibitors.
Lavinia Baciu-Atudosie, A. Ghinet, A. Farce, J. Dubois +2 more
2012Bioorganic & Medicinal Chemistry Letters19 citations Open access
Semantic Scholar
Identification of a pharmacophore of SKCa channel blockers
S. Dilly, Amaury Graulich, A. Farce, V. Seutin +2 more
2005Journal of Enzyme Inhibition and Medicinal Chemistry19 citations Open access
Semantic Scholar
Novel 1,3-dicarbonyl compounds having 2(3H)-benzazolonic heterocycles as PPARgamma agonists.
Elodie Blanc-Delmas, N. Lebègue, V. Wallez, V. Leclerc +20 more
2006Bioorganic & Medicinal Chemistry18 citations
Semantic Scholar
Potent farnesyltransferase inhibitors with 1,4-diazepane scaffolds as novel destabilizing microtubule agents in hormone-resistant prostate cancer.
Nicolas Wlodarczyk, Delphine Le Broc-Ryckewaert, P. Gilleron, A. Lemoine +7 more
2011Journal of Medicinal Chemistry17 citations
Semantic Scholar
Differences in Binding Sites of Two Melatonin Receptors Help to Explain Their Selectivity to Some Melatonin Analogs: A Molecular Modeling Study
A. Chugunov, A. Farce, P. Chavatte, R. Efremov
2006Journal of Biomolecular Structure and Dynamics17 citations
Semantic Scholar
Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3.
V. Leclerc, M. Ettaoussi, Marouan Rami, A. Farce +6 more
2011European journal of medicinal chemistry16 citations Open access
Semantic Scholar
Genetic polymorphism of CYP4A11 and CYP4A22 genes and in silico insights from comparative 3D modelling in a French population.
C. L. Lino Cardenas, N. Renault, A. Farce, C. Cauffiez +6 more
2011Gene15 citations
Semantic Scholar
Ultrasounds-mediated 10-seconds synthesis of chalcones as potential farnesyltransferase inhibitors.
Germain Homerin, A. Nica, A. Farce, J. Dubois +1 more
2020Bioorganic & Medicinal Chemistry Letters13 citations Open access
Semantic Scholar
Phenothiazine-based CaaX competitive inhibitors of human farnesyltransferase bearing a cysteine, methionine, serine or valine moiety as a new family of antitumoral compounds.
Gina-Mirabela Dumitriu, E. Bîcu, Dalila Belei, B. Rigo +3 more
2015Bioorganic & Medicinal Chemistry Letters13 citations Open access
Semantic Scholar
Synthesis and biological evaluation of a new series of N-ylides as protein farnesyltransferase inhibitors.
Cristina-Maria Abuhaie, A. Ghinet, A. Farce, J. Dubois +2 more
2013Bioorganic & Medicinal Chemistry Letters13 citations Open access
Semantic Scholar
Structural insight into PPARgamma ligands binding.
A. Farce, N. Renault, P. Chavatte
2009Current Medicinal Chemistry13 citations
Semantic Scholar
Quantitative structure-activity relationships studies of antioxidant hexahydropyridoindoles and flavonoid derivatives
A. Durand, A. Farce, P. Carato, S. Dilly +3 more
2007Journal of Enzyme Inhibition and Medicinal Chemistry13 citations Open access
Semantic Scholar
Polycyclic nitrogen heterocycles as potential thymidine phosphorylase inhibitors: synthesis, biological evaluation, and molecular docking study
Karen Aknin, Alexis Bontemps, A. Farce, Éric Merlet +6 more
2021Journal of Enzyme Inhibition and Medicinal Chemistry12 citations Open access
Semantic Scholar

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J. Dubois×14
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E. Bîcu×11
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