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P. Arimondo · SciRah

Researcher profile · Semantic Scholar

P. Arimondo

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P. Arimondo — researcher profile on SciRah

h-index: 36
Works: 166
Citations: 5,408

Most-cited papers

Towards the sustainable discovery and development of new antibiotics
M. Miethke, M. Pieroni, T. Weber, M. Brönstrup +50 more
2021Nature Reviews Chemistry944 citations Open access
Semantic Scholar
The timeline of epigenetic drug discovery: from reality to dreams
A. Ganesan, P. Arimondo, M. Rots, C. Jerónimo +1 more
2019Clinical Epigenetics287 citations Open access
Semantic Scholar
DNA Methylation Targeting: The DNMT/HMT Crosstalk Challenge
O. Castillo-Aguilera, P. Depreux, L. Halby, P. Arimondo +1 more
2017Biomolecules145 citations Open access
Semantic Scholar
Targeting DNA methylation with small molecules: what's next?
A. Erdmann, L. Halby, J. Fahy, P. Arimondo
2015Journal of Medicinal Chemistry122 citations Open access
Semantic Scholar
DNA methyltransferase inhibitors in cancer: From pharmacology to translational studies.
Dany Pechalrieu, C. Etiévant, P. Arimondo
2017Biochemical Pharmacology106 citations Open access
Semantic Scholar
Identification of novel quinazoline derivatives as potent antiplasmodial agents.
Anne Bouchut, D. Rotili, C. Pierrot, S. Valente +13 more
2019European journal of medicinal chemistry55 citations Open access
Semantic Scholar
Non-canonical functions of UHRF1 maintain DNA methylation homeostasis in cancer cells
Kosuke Yamaguchi, Xiaoying Chen, Brianna Rodgers, F. Miura +19 more
2023bioRxiv54 citations Open access
Semantic Scholar
Microtubule-Driven Stress Granule Dynamics Regulate Inhibitory Immune Checkpoint Expression in T Cells.
Don-Marc Franchini, Olivia Lanvin, M. Tosolini, Emilie Patras de Campaigno +14 more
2019Cell Reports52 citations Open access
Semantic Scholar
Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells.
L. Halby, Yoann Menon, Elodie Rilova, Dany Pechalrieu +13 more
2017Journal of Medicinal Chemistry51 citations Open access
Semantic Scholar
Combined analysis of DNA methylation and cell cycle in cancer cells
C. Desjobert, M. El Maï, Tom Gérard-Hirne, D. Guianvarc’h +4 more
2015Epigenetics49 citations Open access
Semantic Scholar
The DNMT3A R882H mutant displays altered flanking sequence preferences
Max Emperle, A. Rajavelu, Stefan Kunert, P. Arimondo +3 more
2018Nucleic Acids Research46 citations Open access
Semantic Scholar
Malaria Parasite Stress Tolerance Is Regulated by DNMT2-Mediated tRNA Cytosine Methylation
Elie Hammam, Ameya Sinha, S. Baumgarten, F. Nardella +9 more
2021mBio37 citations Open access
Semantic Scholar
Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells
Clemens Zwergel, M. Schnekenburger, Federica Sarno, Cecilia Battistelli +17 more
2019Clinical Epigenetics37 citations Open access
Semantic Scholar
A Quinoline-Based DNA Methyltransferase Inhibitor as a Possible Adjuvant in Osteosarcoma Therapy
M. Manara, S. Valente, C. Cristalli, G. Nicoletti +12 more
2018Molecular Cancer Therapeutics35 citations Open access
Semantic Scholar
Synergistic chromatin repression of the tumor suppressor gene RARB in human prostate cancers
Céline Moison, Fanny Assemat, Antoine Daunay, J. Tost +2 more
2014Epigenetics33 citations Open access
Semantic Scholar
Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity
D. Rotili, D. Tarantino, B. Marrocco, Christina Gros +15 more
2014PLoS ONE33 citations Open access
Semantic Scholar
Cytisine-like alkaloids from Ormosia hosiei Hemsl. & E.H. Wilson.
Isabelle Pouny, Muriel Batut, L. Vendier, Bruno David +4 more
2014Phytochemistry30 citations
Semantic Scholar
DNA Methylation Bisubstrate Inhibitors Are Fast-Acting Drugs Active against Artemisinin-Resistant Plasmodium falciparum Parasites
F. Nardella, L. Halby, Elie Hammam, Diane Erdmann +7 more
2019ACS Central Science29 citations Open access
Semantic Scholar
Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors
L. Halby, N. Marechal, Dany Pechalrieu, V. Cura +15 more
2018Philosophical Transactions of the Royal Society B: Biological Sciences29 citations Open access
Semantic Scholar
Inhibition studies of DNA methyltransferases by maleimide derivatives of RG108 as non-nucleoside inhibitors.
G. Rondelet, L. Fleury, C. Faux, V. Masson +4 more
2017Future Medicinal Chemistry28 citations
Semantic Scholar
Synthesis of novel 3-halo-3-nitroflavanones and their activities as DNA methyltransferase inhibitors in cancer cells.
Dany Pechalrieu, D. Dauzonne, P. Arimondo, Marie Lopez
2019European journal of medicinal chemistry27 citations Open access
Semantic Scholar
Wandering along the epigenetic timeline
Clémence Topart, Emilie Werner, P. Arimondo
2020Clinical Epigenetics26 citations Open access
Semantic Scholar
DNA Methyltransferase Inhibitors: Development and Applications.
Marie Lopez, L. Halby, P. Arimondo
2016Advances in Experimental Medicine and Biology25 citations
Semantic Scholar
Procainamide-SAHA Fused Inhibitors of hHDAC6 Tackle Multidrug-Resistant Malaria Parasites.
F. Nardella, L. Halby, Irina Dobrescu, Johanna Viluma +13 more
2021Journal of Medicinal Chemistry24 citations Open access
Semantic Scholar
The past and presence of gene targeting: from chemicals and DNA via proteins to RNA
T. M. Geel, M. H. Ruiters, R. Cool, L. Halby +5 more
2018Philosophical Transactions of the Royal Society B: Biological Sciences23 citations Open access
Semantic Scholar
Design and synthesis of new non nucleoside inhibitors of DNMT3A.
A. Erdmann, Yoann Menon, Christina Gros, Nicolas Molinier +7 more
2015Bioorganic & Medicinal Chemistry23 citations Open access
Semantic Scholar
Natural Products and Chemical Biology Tools: Alternatives to Target Epigenetic Mechanisms in Cancers.
Santiago Lascano, Marie Lopez, P. Arimondo
2018The chemical record22 citations Open access
Semantic Scholar
Identification of epigenetic factors regulating the mesenchyme to epithelium transition by RNA interference screening in breast cancer cells
Jean-Marc Gregoire, L. Fleury, Clara Salazar-Cardozo, Frédéric Alby +3 more
2016BMC Cancer22 citations Open access
Semantic Scholar
Disruptor of telomeric silencing 1-like (DOT1L): disclosing a new class of non-nucleoside inhibitors by means of ligand-based and structure-based approaches
Manuela Sabatino, D. Rotili, A. Patsilinakos, M. Forgione +5 more
2018Journal of Computer-Aided Molecular Design20 citations
Semantic Scholar
Consequences of combining siRNA-mediated DNA methyltransferase 1 depletion with 5-aza-2′-deoxycytidine in human leukemic KG1 cells
S. Vispé, A. Deroide, Emeline L. Davoine, C. Desjobert +11 more
2015OncoTarget18 citations Open access
Semantic Scholar
Inhibitors of DNA Methylation.
Marie Lopez, Julie Gilbert, Jean-Marie Contreras, L. Halby +1 more
2022Advances in Experimental Medicine and Biology17 citations
Semantic Scholar
Identification and optimization of hydrazone-gallate derivatives as specific inhibitors of DNA methyltransferase 3A.
A. Erdmann, Yoann Menon, Christina Gros, V. Masson +6 more
2016Future Medicinal Chemistry15 citations
Semantic Scholar
Targeting Germ Cell Tumors with the Newly Synthesized Flavanone-Derived Compound MLo1302 Efficiently Reduces Tumor Cell Viability and Induces Apoptosis and Cell Cycle Arrest
J. Lobo, A. Cardoso, V. Miranda-Gonçalves, L. Looijenga +4 more
2021Pharmaceutics13 citations Open access
Semantic Scholar
The methylome of Biomphalaria glabrata and other mollusks: enduring modification of epigenetic landscape and phenotypic traits by a new DNA methylation inhibitor
N. Luviano, Marie Lopez, F. Gawehns, C. Chaparro +6 more
2020Epigenetics & Chromatin13 citations Open access
Semantic Scholar
Challenges in developing novel DNA methyltransferases inhibitors for cancer therapy.
D. Guianvarc’h, P. Arimondo
2014Future Medicinal Chemistry13 citations
Semantic Scholar
Towards the sustainable discovery and development of new antibiotics.
M. Miethke, M. Pieroni, T. Weber, M. Brönstrup +50 more
2021Nature Reviews Chemistry12 citations Open access
Semantic Scholar
Demethylation by low-dose 5-aza-2′-deoxycytidine impairs 3D melanoma invasion partially through miR-199a-3p expression revealing the role of this miR in melanoma
C. Desjobert, Arnaud Carrier, Audrey Delmas, D. Marzese +8 more
2019Clinical Epigenetics12 citations Open access
Semantic Scholar
Epidrugs as Promising Tools to Eliminate Plasmodium falciparum Artemisinin-Resistant and Quiescent Parasites
Thibaud Reyser, L. Paloque, Michel Nguyen, J. Augereau +7 more
2023Pharmaceutics11 citations Open access
Semantic Scholar
Synthesis and Biological Activity of a Cytostatic Inhibitor of MLLr Leukemia Targeting the DOT1L Protein
Corentin Bon, Y. Si, Mélanie Pernak, Magdalena Barbachowska +9 more
2021Molecules11 citations Open access
Semantic Scholar
A genetic screen identifies BEND3 as a regulator of bivalent gene expression and global DNA methylation
L. Yakhou, Anaelle Azogui, Nikhil Gupta, Julien Richard Albert +14 more
2023Nucleic Acids Research10 citations Open access
Semantic Scholar
Novel Quinoline Compounds Active in Cancer Cells through Coupled DNA Methyltransferase Inhibition and Degradation
Clemens Zwergel, R. Fioravanti, G. Stazi, Federica Sarno +15 more
2020Cancers10 citations Open access
Semantic Scholar
To target or not to target? The role of DNA and histone methylation in bacterial infections
Magdalena Barbachowska, P. Arimondo
2023Epigenetics9 citations Open access
Semantic Scholar
Structure-Guided Optimization of DNA Methyltransferase Inhibitors
A. Erdmann, P. Arimondo, D. Guianvarc’h
20168 citations
Semantic Scholar
Pioneering first-in-class HDAC-ROCK inhibitors as potential multitarget anticancer agents.
M. Beljkaš, D. Ružić, Ana Djurić, Ana Vuletic +9 more
2025Future Medicinal Chemistry7 citations Open access
Semantic Scholar
Hemisynthetic alkaloids derived from trilobine are antimalarials with sustained activity in multidrug-resistant Plasmodium falciparum
F. Nardella, Irina Dobrescu, Haitham Hassan, F. Rodrigues +19 more
2023iScience7 citations Open access
Semantic Scholar
Epigenetically regulated PCDHB15 impairs aggressiveness of metastatic melanoma cells
Arnaud Carrier, C. Desjobert, V. Lobjois, Lise Rigal +11 more
2022Clinical Epigenetics7 citations Open access
Semantic Scholar
Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic 'writers'.
Corentin Bon, L. Halby, P. Arimondo
2020Epigenomics7 citations Open access
Semantic Scholar
Plasmodium falciparum Eukaryotic Translation Initiation Factor 3 is Stabilized by Quinazoline-Quinoline Bisubstrate Inhibitors
Irina Dobrescu, Elie Hammam, J. Dziekan, Aurélie Claës +6 more
2023ACS Infectious Diseases6 citations Open access
Semantic Scholar
Bisubstrate-Type Chemical Probes Identify GRP94 as a Potential Target of Cytosine-Containing Adenosine Analogs
Dany Pechalrieu, Fanny Assemat, L. Halby, M. Marcellin +7 more
2020ACS Chemical Biology6 citations Open access
Semantic Scholar
DNA methylome combined with chromosome cluster-oriented analysis provides an early signature for cutaneous melanoma aggressiveness
Arnaud Carrier, C. Desjobert, L. Ponger, L. Lamant +14 more
2022bioRxiv5 citations Open access
Semantic Scholar

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