Skip to content

Home Search Authors Pakistan News Saved

SciRah

SciRah does not host or store research papers. Results come live from free, official scholarly APIs, and every paper links back to its original source.

Data sources

OpenAlex
Semantic Scholar
Crossref
CORE
arXiv
PubMed

Privacy policy Terms of service

Ciro Milite · SciRah

Researcher profile · Semantic Scholar

Ciro Milite

Share profile

Ciro Milite — researcher profile on SciRah

h-index: 22
Works: 69
Citations: 1,342

Most-cited papers

NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors
A. Cipriano, M. Viviano, Alessandra Feoli, Ciro Milite +3 more
2023Journal of Medicinal Chemistry165 citations Open access
Semantic Scholar
Highly enantioselective organocatalytic α-amination reactions of aryl oxindoles: developing designer multifunctional alkaloid catalysts.
Tommy Bui, Gloria Hernández-Torres, Ciro Milite, C. Barbas
2010Organic Letters106 citations
Semantic Scholar
p300/CBP-associated factor selectively regulates the extinction of conditioned fear
Wei Wei, C. Coelho, Xiang Li, R. Marek +13 more
2012Journal of Neuroscience95 citations Open access
Semantic Scholar
The emerging role of lysine methyltransferase SETD8 in human diseases
Ciro Milite, Alessandra Feoli, M. Viviano, Donatella Rescigno +5 more
2016Clinical Epigenetics87 citations Open access
Semantic Scholar
Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines.
M. Sala, A. Chimento, C. Saturnino, I. Gomez-Monterrey +10 more
2013Bioorganic & Medicinal Chemistry Letters68 citations Open access
Semantic Scholar
Nutraceutical properties and polyphenolic profile of berry skin and wine of Vitis vinifera L. (cv. Aglianico).
M. De Nisco, M. Manfra, A. Bolognese, A. Sofo +5 more
2013Food Chemistry68 citations
Semantic Scholar
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI‐1)
S. Castellano, Ciro Milite, R. Ragno, S. Simeoni +9 more
2010ChemMedChem64 citations
Semantic Scholar
A novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach.
Ciro Milite, Alessandra Feoli, K. Sasaki, V. La Pietra +7 more
2015Journal of Medicinal Chemistry54 citations Open access
Semantic Scholar
Discovery of a Novel Chemotype of Histone Lysine Methyltransferase EHMT1/2 (GLP/G9a) Inhibitors: Rational Design, Synthesis, Biological Evaluation, and Co-crystal Structure
Ciro Milite, Alessandra Feoli, J. Horton, Donatella Rescigno +10 more
2019Journal of Medicinal Chemistry51 citations Open access
Semantic Scholar
Structure-activity relationship refinement and further assessment of 4-phenylquinazoline-2-carboxamide translocator protein ligands as antiproliferative agents in human glioblastoma tumors.
S. Castellano, Sabrina Taliani, M. Viviano, Ciro Milite +11 more
2014Journal of Medicinal Chemistry45 citations Open access
Semantic Scholar
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells
E. Miele, S. Valente, Vincenzo Alfano, M. Silvano +16 more
2017OncoTarget44 citations Open access
Semantic Scholar
Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.
S. Castellano, Sabrina Taliani, Ciro Milite, Isabella Pugliesi +11 more
2012Journal of Medicinal Chemistry39 citations Open access
Semantic Scholar
Modulation of the activity of histone acetyltransferases by long chain alkylidenemalonates (LoCAMs).
Ciro Milite, S. Castellano, R. Benedetti, A. Tosco +7 more
2011Bioorganic & Medicinal Chemistry33 citations Open access
Semantic Scholar
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation
Tara H. W. Dobson, R. Hatcher, Jyothishmathi Swaminathan, C. Das +7 more
2017Molecular Cancer Research32 citations Open access
Semantic Scholar
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies
Ciro Milite, Giorgio Amendola, A. Nocentini, Silvia Bua +9 more
2019Journal of Enzyme Inhibition and Medicinal Chemistry30 citations Open access
Semantic Scholar
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach.
M. G. Chini, N. Malafronte, M. Vaccaro, M. Gualtieri +8 more
2016Chemistry30 citations
Semantic Scholar
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction–Reconstruction and Fragment-Growing Approach
Giulia Iannelli, Ciro Milite, N. Marechal, V. Cura +11 more
2022Journal of Medicinal Chemistry28 citations Open access
Semantic Scholar
Lysine methyltransferase inhibitors: where we are now
Alessandra Feoli, M. Viviano, A. Cipriano, Ciro Milite +2 more
2021RSC Chemical Biology28 citations Open access
Semantic Scholar
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1
S. Castellano, Astrid Spannhoff, Ciro Milite, F. Dal Piaz +12 more
2012Journal of Medicinal Chemistry27 citations Open access
Semantic Scholar
Reverse transcriptase inhibitors promote the remodeling of nuclear architecture and induce autophagy in prostate cancer cells.
Cristina Bellisai, I. Sciamanna, P. Rovella, D. Giovannini +12 more
2020Cancer Letters25 citations
Semantic Scholar
Identification of Structural Features of 2‐Alkylidene‐1,3‐Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF
S. Castellano, Ciro Milite, Alessandra Feoli, M. Viviano +4 more
2015ChemMedChem24 citations
Semantic Scholar
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors.
Silvia Salerno, E. Barresi, Giorgio Amendola, E. Berrino +7 more
2018Journal of Medicinal Chemistry22 citations Open access
Semantic Scholar
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans.
E. C. Calabrese, S. Castellano, Marisabella Santoriello, C. Sgherri +11 more
2013Journal of Antimicrobial Chemotherapy21 citations
Semantic Scholar
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors.
Gianluca Sbardella, A. Mai, Sara Bartolini, S. Castellano +9 more
2011Journal of Medicinal Chemistry19 citations
Semantic Scholar
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery
M. Viviano, Ciro Milite, Donatella Rescigno, S. Castellano +1 more
201517 citations
Semantic Scholar
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO).
Ciro Milite, E. Barresi, E. Da Pozzo, B. Costa +10 more
2017Journal of Medicinal Chemistry16 citations Open access
Semantic Scholar
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors
Ciro Milite, Alessandra Feoli, M. Viviano, Donatella Rescigno +3 more
2016ChemMedChem16 citations
Semantic Scholar
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor
Alessandra Feoli, Giulia Iannelli, A. Cipriano, Ciro Milite +14 more
2023Journal of Medicinal Chemistry13 citations Open access
Semantic Scholar
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli.
M. Franek, S. Legartová, J. Suchánková, Ciro Milite +4 more
2015Physiological Research11 citations Open access
Semantic Scholar
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization
L. Fattore, D. Malpicci, Ciro Milite, S. Castellano +5 more
2020Cell communication and signaling : CCS8 citations Open access
Semantic Scholar
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice
S. Creighton, Kristen H. Jardine, Alexa Desimone, Megan Zmetana +4 more
2022Learning & memory (Cold Spring Harbor, N.Y.)7 citations Open access
Semantic Scholar
Discovery of Benzo[d]imidazole‐6‐sulfonamides as Bromodomain and Extra‐Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain
A. Cipriano, Ciro Milite, Alessandra Feoli, M. Viviano +10 more
2022ChemMedChem7 citations Open access
Semantic Scholar
Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases.
Silvia Salerno, V. La Pietra, M. Hyeraci, Sabrina Taliani +10 more
2019European journal of medicinal chemistry6 citations Open access
Semantic Scholar
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids
S. Castellano, Ciro Milite, P. Campiglia, Gianluca Sbardella
20076 citations
Semantic Scholar
New Pyridobenothiazolone Derivatives Display Nanomolar Pan‐Serotype Anti‐Dengue Virus Activity
Tommaso Felicetti, C. P. Gwee, K. Chan, G. Pepe +10 more
2025ChemMedChem5 citations
Semantic Scholar
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review
M. Viviano, Alessandra Cipriano, Emanuele Fabbrizi, Alessandra Feoli +5 more
2024Expert Opinion on Therapeutic Patents5 citations
Semantic Scholar
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors
Ermelinda Vernieri, I. Gomez-Monterrey, Ciro Milite, P. Grieco +9 more
2013Journal of Amino Acids5 citations Open access
Semantic Scholar
Straightforward, metal-free, and stereoselective synthesis of 9-oxo- and 10-hydroxy-2(E)-decenoic acids, important components of honeybee (Apis mellifera) secretions
Ciro Milite, M. Viviano, Marisabella Santoriello, F. Aricò +2 more
20125 citations Open access
Semantic Scholar
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype
Yi Zhang, Paolo Zanotti Fregonara, J. Kimberly, Robert L. Gladding +9 more
20133 citations Open access
Semantic Scholar
2‐Phenylquinolines Exhibit Anti‐Severe Acute Respiratory Syndrome Coronavirus‐2 Activity Through the Nonstructural Protein 13 Helicase Inhibition
Giada Cernicchi, Maria Giulia Nizi, Roberta Emmolo, L. Persoons +21 more
2026ChemMedChem2 citations Open access
Semantic Scholar
Prodrug Approach to Exploit (S)‐Alanine Amide as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors
Ciro Milite, Giuliana Sarno, Ida Pacilio, Agostino Cianciulli +9 more
2024ChemMedChem2 citations Open access
Semantic Scholar
The Lysine Acetyltransferase PCAF Functionally Interacts with Estrogen Receptor Alpha in the Hippocampus of Gonadally Intact Male—But Not Female—Rats to Enhance Short-Term Memory
K. Mitchnick, Kate Nicholson, Cassidy E. Wideman, Kristen H. Jardine +9 more
2024Journal of Neuroscience2 citations Open access
Semantic Scholar
Inside Cover: Identification of Structural Features of 2‐Alkylidene‐1,3‐Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015)
S. Castellano, Ciro Milite, Alessandra Feoli, M. Viviano +4 more
20152 citations Open access
Semantic Scholar
Targeting Copper in Cancer: Chelators to Counteract Cuproplasia and Ionophores to Promote Cuproptosis
Sabrina Castellano, A. Tosco, Ciro Milite, M. Viviano +3 more
2026Journal of Medicinal Chemistry1 citations Open access
Semantic Scholar
Coactivator-associated arginine methyltransferase 1 (CARM1) inhibitors: a patenting perspective (2018-present)
M. Viviano, Alessandra Cipriano, Alessandra Feoli, Ciro Milite +2 more
2025Expert Opinion on Therapeutic Patents1 citations
Semantic Scholar
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization
L. Fattore, D. Malpicci, Ciro Milite, S. Castellano +5 more
2020Cell Communication and Signaling1 citations Open access
Semantic Scholar
Patent evaluation of WO2019209182 (A1) 2019-10-31 (Conjugated Oligoelectrolytes as Antimicrobial Agents)
Ciro Milite
2020Expert Opinion on Therapeutic Patents1 citations
Semantic Scholar
Sulfonyl Anthranilic Acid Analogues Display Pan-Serotype Anti-Dengue Activity by Downregulating the Expression of Ribosomal Proteins Encoded by 5′-Terminal Oligopyrimidine Motif-Containing mRNA
C. P. Gwee, Tommaso Felicetti, K. Chan, M. Tan +21 more
2026Journal of Medicinal Chemistry0 citations Open access
Semantic Scholar
Discovery of High-Affinity Peptide Ligands Targeting the SPIN1 Tudor 3 Domain Via a Minimalist Pruning Strategy
Alessandra Feoli, Giulio Esposito, M. Grimaldi, M. Viviano +8 more
2026ACS Medicinal Chemistry Letters0 citations Open access
Semantic Scholar
Targeting PRMTs with small-molecule inhibitors: a comprehensive review
M. Viviano, Alessandra Cipriano, Benito D'Ascoli, Ciro Milite +2 more
2026RSC Medicinal Chemistry0 citations Open access
Semantic Scholar

Frequent co-authors

Invite them to SciRah by sharing their profile.

Gianluca Sbardella×39
Invite
Gianluca Sbardella — researcher profile on SciRah
S. Castellano×32
Invite
S. Castellano — researcher profile on SciRah
M. Viviano×21
Invite
M. Viviano — researcher profile on SciRah
Alessandra Feoli×16
Invite
Alessandra Feoli — researcher profile on SciRah

×14

Invite

E. Novellino — researcher profile on SciRah

Invite

A. Mai — researcher profile on SciRah

Invite

A. Cipriano — researcher profile on SciRah

S. Cosconati×7

Invite

S. Cosconati — researcher profile on SciRah

Sabrina Taliani×7

Invite

Sabrina Taliani — researcher profile on SciRah

F. Da Settimo×7

Invite

F. Da Settimo — researcher profile on SciRah

Sabrina Castellano×7

Invite

Sabrina Castellano — researcher profile on SciRah

Invite

A. Tosco — researcher profile on SciRah