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Giorgio Amendola · SciRah

Researcher profile · Semantic Scholar

Giorgio Amendola

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Giorgio Amendola — researcher profile on SciRah

h-index: 15
Works: 28
Citations: 503

Most-cited papers

Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs).
S. Previti, R. Ettari, S. Cosconati, Giorgio Amendola +12 more
2017Journal of Medicinal Chemistry56 citations Open access
Semantic Scholar
PyRMD: A New Fully Automated AI-Powered Ligand-Based Virtual Screening Tool
Giorgio Amendola, S. Cosconati
2021Journal of Chemical Information and Modeling54 citations Open access
Semantic Scholar
Discovery of a Novel Chemotype of Histone Lysine Methyltransferase EHMT1/2 (GLP/G9a) Inhibitors: Rational Design, Synthesis, Biological Evaluation, and Co-crystal Structure
Ciro Milite, Alessandra Feoli, J. Horton, Donatella Rescigno +10 more
2019Journal of Medicinal Chemistry51 citations Open access
Semantic Scholar
Lead Discovery of SARS-CoV-2 Main Protease Inhibitors through Covalent Docking-Based Virtual Screening
Giorgio Amendola, R. Ettari, S. Previti, C. Di Chio +8 more
2021Journal of Chemical Information and Modeling41 citations
Semantic Scholar
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies
Ciro Milite, Giorgio Amendola, A. Nocentini, Silvia Bua +9 more
2019Journal of Enzyme Inhibition and Medicinal Chemistry30 citations Open access
Semantic Scholar
Optimization strategy of novel peptide-based Michael acceptors for the treatment of Human African Trypanosomiasis.
R. Ettari, S. Previti, Santina Maiorana, Giorgio Amendola +5 more
2019Journal of Medicinal Chemistry26 citations Open access
Semantic Scholar
Dual MET and SMO Negative Modulators Overcome Resistance to EGFR Inhibitors in Human Nonsmall Cell Lung Cancer.
F. Morgillo, Giorgio Amendola, C. D. Della Corte, C. Giacomelli +11 more
2017Journal of Medicinal Chemistry25 citations Open access
Semantic Scholar
Discovery of the first dual G-triplex/G-quadruplex stabilizing compound: a new opportunity in the targeting of G-rich DNA structures?
J. Amato, Alessia Pagano, S. Cosconati, Giorgio Amendola +8 more
2017Biochimica et Biophysica Acta - General Subjects24 citations
Semantic Scholar
Pyrrolyl Pyrazoles as Non-Diketo Acid Inhibitors of the HIV-1 Ribonuclease H Function of Reverse Transcriptase.
A. Messore, A. Corona, V. N. Madia, Francesco Saccoliti +16 more
2020ACS Medicinal Chemistry Letters23 citations Open access
Semantic Scholar
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors.
Silvia Salerno, E. Barresi, Giorgio Amendola, E. Berrino +7 more
2018Journal of Medicinal Chemistry22 citations Open access
Semantic Scholar
FEPrepare: A Web-Based Tool for Automating the Setup of Relative Binding Free Energy Calculations
Stamatia Zavitsanou, Alexandros Tsengenes, Michail Papadourakis, Giorgio Amendola +4 more
2021Journal of Chemical Information and Modeling21 citations
Semantic Scholar
Development of novel dipeptide nitriles as inhibitors of rhodesain of Trypanosoma brucei rhodesiense.
C. Di Chio, S. Previti, Giorgio Amendola, R. Ravichandran +6 more
2022European journal of medicinal chemistry19 citations Open access
Semantic Scholar
Streamlining Large Chemical Library Docking with Artificial Intelligence: the PyRMD2Dock Approach
Michele Roggia, Benito Natale, Giorgio Amendola, S. Di Maro +1 more
2023Journal of Chemical Information and Modeling18 citations Open access
Semantic Scholar
Peptidyl Vinyl Ketones Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment.
Santina Maiorana, R. Ettari, S. Previti, Giorgio Amendola +5 more
2020ChemMedChem16 citations
Semantic Scholar
Identification of novel indole derivatives acting as inhibitors of the Keap1–Nrf2 interaction
B. Cosimelli, G. Greco, S. Laneri, E. Novellino +5 more
2019Journal of Enzyme Inhibition and Medicinal Chemistry16 citations Open access
Semantic Scholar
Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold.
Silvia Salerno, Giorgio Amendola, A. Angeli, Emma Baglini +10 more
2021European journal of medicinal chemistry13 citations Open access
Semantic Scholar
Development of Novel Benzodiazepine‐Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense
C. Di Chio, S. Previti, Giorgio Amendola, S. Cosconati +3 more
2020ChemMedChem11 citations
Semantic Scholar
Structure–Activity Relationship Studies on Oxazolo[3,4-a]pyrazine Derivatives Leading to the Discovery of a Novel Neuropeptide S Receptor Antagonist with Potent In Vivo Activity
Valentina Albanese, C. Ruzza, E. Marzola, T. Bernardi +12 more
2021Journal of Medicinal Chemistry9 citations Open access
Semantic Scholar
Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase
A. Messore, A. Corona, V. N. Madia, Francesco Saccoliti +15 more
2021Journal of Medicinal Chemistry8 citations Open access
Semantic Scholar
New insights in the structure-activity relationships of 2-phenylamino-substituted benzothiopyrano[4,3-d]pyrimidines as kinase inhibitors.
Silvia Salerno, A. García-Argáez, E. Barresi, Sabrina Taliani +9 more
2018European journal of medicinal chemistry8 citations Open access
Semantic Scholar
Discovery of Pyrido[3',2':5,6]thiopyrano[4,3-d]pyrimidine-Based Antiproliferative Multikinase Inhibitors.
Silvia Salerno, E. Barresi, A. García-Argáez, Sabrina Taliani +8 more
2019ACS Medicinal Chemistry Letters6 citations Open access
Semantic Scholar
Best Matching Protein Conformations and Docking Programs for a Virtual Screening Campaign Against SMO Receptor
Giorgio Amendola, D. Di Maio, V. La Pietra, S. Cosconati
2016Molecular Informatics4 citations
Semantic Scholar
Discovering Dually Active Anti-cancer Compounds with a Hybrid AI-structure-based Approach
Michele Roggia, Benito Natale, Giorgio Amendola, Nicola Grasso +7 more
2024Journal of Chemical Information and Modeling1 citations
Semantic Scholar
Discovery of N-substituted-2-oxoindolin benzoylhydrazines as c-MET/SMO modulators in EGFRi-resistant non-small cell lung cancer.
Stefano Tomassi, Benito Natale, Michele Roggia, Luisa Amato +13 more
2024RSC Medicinal Chemistry1 citations Open access
Semantic Scholar
Targeting the Tumor-Stroma Crosstalk: An AI-Based Virtual Screening Strategy for Dual MET/SMO Inhibitors in Pancreatic Cancer
Michele Roggia, U. Chianese, Giorgio Amendola, Valentina Albanese +13 more
2026bioRxiv0 citations Open access
Semantic Scholar
Repurposing of valproic acid and simvastatin as anticancer agents in pancreatic cancer: a new therapeutic approach in combination with chemotherapy. Tutor: Dott
A. Ametrano, M. Coscia, A. M. Campos, P. Italiani +29 more
20190 citations
Semantic Scholar
Standards, what passion] OSI, SNA, MAP
Giorgio Amendola
19870 citations
Semantic Scholar
Structure − Activity Relationship Studies on Oxazolo[3,4 ‑ a ]pyrazine Derivatives Leading to the Discovery of a Novel Neuropeptide S Receptor Antagonist with Potent In Vivo Activity
Valentina Albanese, Chiara Ruzza, E. Marzola, Tatiana Bernardi +12 more
0 citations
Semantic Scholar

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