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L. Winneroski · SciRah

Researcher profile · Semantic Scholar

L. Winneroski

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L. Winneroski — researcher profile on SciRah

h-index: 18
Works: 49
Citations: 1,363

Most-cited papers

(S)-13-[(dimethylamino)methyl]-10,11,14,15-tetrahydro-4,9:16, 21-dimetheno-1H, 13H-dibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecene-1,3(2H)-d ione (LY333531) and related analogues: isozyme selective inhibitors of protein kinase C beta.
M. Jirousek, James R. Gillig, C. Gonzalez, William F. Heath +11 more
1996Journal of Medicinal Chemistry311 citations Open access
Semantic Scholar
The Potent BACE1 Inhibitor LY2886721 Elicits Robust Central Aβ Pharmacodynamic Responses in Mice, Dogs, and Humans
P. May, B. Willis, S. Lowe, R. Dean +27 more
2015Journal of Neuroscience165 citations Open access
Semantic Scholar
A New, Efficient Method for the Synthesis of Bisindolylmaleimides.
M. Faul, L. Winneroski, C. A. Krumrich
1998Journal of Organic Chemistry126 citations
Semantic Scholar
Salt form selection and characterization of LY333531 mesylate monohydrate.
Gary Lowell Engel, N. A. Farid, M. Faul, Lori Ann Richardson +1 more
2000International journal of pharmaceutics106 citations
Semantic Scholar
Design and synthesis of 2-methyl-2-[4-(2-[5-methyl-2-aryloxazol-4-yl]ethoxy)phenoxy]propionic acids: a new class of dual PPARalpha/gamma agonists.
Dawn A. Brooks, Garret J. Etgen, C. J. Rito, Anthony John Shuker +13 more
2001Journal of Medicinal Chemistry60 citations Open access
Semantic Scholar
Synthesis of novel retinoid X receptor-selective retinoids.
M. Faul, A. M. Ratz, K. A. Sullivan, W. G. Trankle +1 more
2001Journal of Organic Chemistry59 citations
Semantic Scholar
SYNTHESIS OF REBECCAMYCIN AND 11-DECHLOROREBECCAMYCIN
M. Faul, L. Winneroski, C. A. Krumrich
199955 citations
Semantic Scholar
A new one step synthesis of maleimides by condensation of glyoxylate esters with acetamides
M. Faul, L. Winneroski, C. A. Krumrich
199952 citations
Semantic Scholar
Aryl[a]pyrrolo[3,4-c]carbazoles as selective cyclin D1-CDK4 inhibitors.
Concha Sánchez-Martínez, C. Shih, M. Faul, Guoxin Zhu +18 more
2003Bioorganic & Medicinal Chemistry Letters47 citations Open access
Semantic Scholar
A General Approach to the Synthesis of Bisindolylmaleimides: Synthesis of Staurosporine Aglycone
M. Faul, K. A. Sullivan, L. Winneroski
199544 citations
Semantic Scholar
Design and synthesis of alpha-aryloxy-alpha-methylhydrocinnamic acids: a novel class of dual peroxisome proliferator-activated receptor alpha/gamma agonists.
Yan-Ping Xu, C. J. Rito, G. Etgen, R. Ardecky +22 more
2004Journal of Medicinal Chemistry42 citations Open access
Semantic Scholar
Design and synthesis of dual peroxisome proliferator-activated receptors γ and δ agonists as novel euglycemic agents with a reduced weight gain profile
Yan-Ping Xu, G. Etgen, C. Broderick, Emily J. Canada +12 more
200627 citations Open access
Semantic Scholar
Discovery and Early Clinical Development of LY3202626, a Low-Dose, CNS-Penetrant BACE Inhibitor.
D. McKinzie, L. Winneroski, S. J. Green, E. Hembre +22 more
2021Journal of Medicinal Chemistry25 citations Open access
Semantic Scholar
Palladium-catalyzed acylation of a 1,2-disubstituted 3-indolylzinc chloride
M. Faul, L. Winneroski
199725 citations
Semantic Scholar
Macrocyclic Bisindolylmaleimides: Synthesis by Inter- and Intramolecular Alkylation
M. Faul, L. Winneroski, C. A. Krumrich, K. A. Sullivan +4 more
199824 citations
Semantic Scholar
Design and synthesis of a novel class of dual PPARγ/δ agonists
Isabel C. González, Lamar Jason Eric, Fatima Iradier, Yan-Ping Xu +9 more
200723 citations Open access
Semantic Scholar
Synthesis of 2′,3′-dideoxy-3′-hydroxymethylcytidine; a unique antiviral nucleoside
M. Faul, B. Huff, S. Dunlap, Scott A. Frank +7 more
199720 citations
Semantic Scholar
Preparation and biological evaluation of conformationally constrained BACE1 inhibitors.
L. Winneroski, M. A. Schiffler, J. Erickson, P. May +15 more
2015Bioorganic & Medicinal Chemistry18 citations Open access
Semantic Scholar
Preparation and biological evaluation of BACE1 inhibitors: Leveraging trans-cyclopropyl moieties as ligand efficient conformational constraints.
L. Winneroski, J. Erickson, S. J. Green, J. E. Lopez +22 more
2019Bioorganic & Medicinal Chemistry16 citations Open access
Semantic Scholar
Synthesis of indolo[2,3-a]carbazole glycoside analogs of rebeccamycin: inhibitors of cyclin D1-CDK4
M. Faul, K. A. Sullivan, J. Grutsch, L. Winneroski +3 more
200416 citations
Semantic Scholar
Conversion of human-selective PPARalpha agonists to human/mouse dual agonists: a molecular modeling analysis.
Minmin Wang, L. Winneroski, R. Ardecky, R. Babine +17 more
2004Bioorganic & Medicinal Chemistry Letters12 citations Open access
Semantic Scholar
Synthesis of bisindolylmaleimide macrocycles
M. Jirousek, G. Ronald, D. A. Neel, C. J. Rito +9 more
199512 citations
Semantic Scholar
Synthesis, Optimization, and Large-Scale Preparation of the Low-Dose Central Nervous System-Penetrant BACE1 Inhibitor LY3202626 via a [3 + 2] Nitrone Cycloaddition
P. García-Losada, A. C. DeBaillie, J. Eugenio de Diego, S. J. Green +18 more
202010 citations
Semantic Scholar
Peroxisome proliferator activated receptor agonists
T. Gibson, R. Johnston, N. Mantlo, R. Thompson +3 more
199710 citations
Semantic Scholar
Practical Asymmetric Fluorination Approach to the Scalable Synthesis of New Fluoroaminothiazine BACE Inhibitors
P. García-Losada, M. Barberis, Yuan Shi, E. Hembre +7 more
20189 citations
Semantic Scholar
Design and synthesis of dual peroxisome proliferator-activated receptors gamma and delta agonists as novel euglycemic agents with a reduced weight gain profile.
Yan-Ping Xu, G. Etgen, C. Broderick, Emily J. Canada +12 more
2006Journal of Medicinal Chemistry8 citations Open access
Semantic Scholar
P1‐080: Nonclinical Pharmacological Characterization of the Bace1 Inhibitor LY3202626
David L. Mckinzie, Patrick C. May, L. Boggs, Zhi-Xiang Yang +7 more
20167 citations
Semantic Scholar
Two complementary approaches toward 2-alkoxy carboxylic acid synthesis from 1,3-dioxolan-4-ones.
L. Winneroski, Yan-Ping Xu
2004Journal of Organic Chemistry6 citations
Semantic Scholar
Synthesis of 2-Phenyloxazole Derivatives Containing Amino Acids as Insulin Sensitivity Enhancers for Treatment of Type II Diabetes.
M. Faul, L. Winneroski, J. York, Matt R. Reinhard +3 more
20016 citations Open access
Semantic Scholar
Design and synthesis of a novel class of dual PPARgamma/delta agonists.
Isabel C. González, J. Lamar, Fatima Iradier, Yan-Ping Xu +9 more
2007Bioorganic & Medicinal Chemistry Letters5 citations
Semantic Scholar
Design and synthesis of novel and potent amide linked PPARγ/δ dual agonists
Qing Shi, Emily J. Canada, Yan-Ping Xu, Alan M. Warshawsky +14 more
20075 citations Open access
Semantic Scholar
Robust Pharmacodynamic Effect of LY3202626, a Central Nervous System Penetrant, Low Dose BACE1 Inhibitor, in Humans and Nonclinical Species
B. Willis, S. Lowe, S. Monk, Patrick J. Cocke +17 more
2022Journal of Alzheimer's disease reports4 citations Open access
Semantic Scholar
Inhibitor protein kinase c.
Gary Lowell Engel, N. A. Farid, M. Faul, M. Jirousek +2 more
19963 citations
Semantic Scholar
Cycloalkyllactamderivater as inhibitors of 11-beta hydroxysteroid dehydrogenase 1
T. Aicher, M. Chicarelli, R. Hinklin, H. Tian +7 more
20052 citations
Semantic Scholar
Macrocyclic Bisindolylmaleimides: Synthesis by Inter- and Intramolecular Alkylation.
M. Faul, L. Winneroski, C. A. Krumrich, K. A. Sullivan +4 more
19982 citations
Semantic Scholar
Synthesis of 2′,3′-Dideoxy-3′-hydroxymethylcytidine; a Unique Antiviral Nucleoside.
M. Faul, B. Huff, S. Dunlap, Scott A. Frank +7 more
19971 citations
Semantic Scholar
Discovery and Structure–Activity Relationship Optimization of a Novel Rv1625c Agonist Chemotype with Antitubercular Activity
Han Xie, Paridhi Sukheja, Kirsten T. Tolentino, J. Webb +13 more
2026bioRxiv0 citations Open access
Semantic Scholar
P3‐035: A Correlational Analysis of Exposure and Pharmacodynamic Effects of the Bace1 Inhibitor LY3202626 in PDAPP Mice Following Acute Oral Dosing
L. Boggs, Patrick C. May, Zhi-Xiang Yang, R. Brier +6 more
20160 citations Open access
Semantic Scholar
Design and synthesis of novel and potent amide linked PPARgamma/delta dual agonists.
Qing Shi, Emily J. Canada, Yan-Ping Xu, Alan M. Warshawsky +14 more
2007Bioorganic & Medicinal Chemistry Letters0 citations
Semantic Scholar
derivatives and agonists Oxazolylarylpropionsäure their use as PPAR
R. Ardecky, Dawn A. Brooks, A. Godfrey, S. Jones +7 more
20010 citations
Semantic Scholar
Synthesis of Novel Retinoid X Receptor‐Selective Retinoids.
M. Faul, A. M. Ratz, K. A. Sullivan, W. G. Trankle +1 more
20010 citations
Semantic Scholar
derivatives and agonists Oxazolylaryloxyessigsäure their use as PPAR
Dawn A. Brooks, S. Connor, S. J. Dominianni, A. Godfrey +6 more
20010 citations
Semantic Scholar
Oxazolyl-derivatives ariloxiacetico acid and their use as PPAR agonists.
Dawn A. Brooks, S. Connor, S. J. Dominianni, A. Godfrey +6 more
20010 citations
Semantic Scholar
A New, Efficient Method for the Synthesis of Bisindolylmaleimides.
M. Faul, L. Winneroski, C. A. Krumrich
19990 citations
Semantic Scholar
A New One-Step Synthesis of Maleimides by Condensation of Glyoxylate Esters with Acetamides.
M. Faul, L. Winneroski, C. A. Krumrich
19990 citations
Semantic Scholar
Palladium-Catalyzed Acylation of a 1,2-Disubstituted 3-Indolylzinc Chloride.
M. Faul, L. Winneroski
19970 citations
Semantic Scholar
A General Approach to the Synthesis of Bisindolylmaleimides: Synthesis of Staurosporine Aglycone.
M. Faul, K. A. Sullivan, L. Winneroski
19960 citations
Semantic Scholar
Synthesis of Bisindolylmaleimide Macrocycles.
M. Jirousek, G. Ronald, D. A. Neel, C. J. Rito +9 more
19960 citations
Semantic Scholar
Intermediates and their use to prepare bisindolylmaleimides bridge n, n '.
M. Faul, C. A. Krumrich, L. Winneroski
19960 citations
Semantic Scholar

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