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M. Waelbroeck · SciRah

Researcher profile · Semantic Scholar

M. Waelbroeck

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M. Waelbroeck — researcher profile on SciRah

h-index: 36
Works: 142
Citations: 4,172

Most-cited papers

Ghrelin degradation by serum and tissue homogenates: identification of the cleavage sites.
C. De Vriese, F. Grégoire, Roger Lema-Kisoka, M. Waelbroeck +2 more
2004Endocrinology311 citations Open access
Semantic Scholar
Binding of selective antagonists to four muscarinic receptors (M1 to M4) in rat forebrain.
M. Waelbroeck, M. Tastenoy, J. Camus, J. Christophe
1990Molecular Pharmacology237 citations Open access
Semantic Scholar
Development of high affinity selective VIP1 receptor agonists.
P. Gourlet, A. Vandermeers, P. Vertongen, J. Rathé +4 more
1997Peptides207 citations
Semantic Scholar
In vitro properties of a high affinity selective antagonist of the VIP1 receptor.
P. Gourlet, P. de Neef, Johnny Cnudde, M. Waelbroeck +1 more
1997Peptides188 citations
Semantic Scholar
Molecular cloning and functional characterization of a human VIP receptor from SUP-T1 lymphoblasts.
Michal Svoboda, M. Tastenoy, J. Vanrampelbergh, J. Goossens +3 more
1994Biochemical and Biophysical Research Communications - BBRC160 citations
Semantic Scholar
The long-acting vasoactive intestinal polypeptide agonist RO 25-1553 is highly selective of the VIP2 receptor subclass.
P. Gourlet, P. Vertongen, A. Vandermeers, M. Vandermeers-piret +4 more
1997Peptides152 citations
Semantic Scholar
Techniques: promiscuous Galpha proteins in basic research and drug discovery.
E. Kostenis, M. Waelbroeck, G. Milligan
2005TIPS - Trends in Pharmacological Sciences135 citations
Semantic Scholar
Affinity profiles of hexahydro-sila-difenidol analogues at muscarinic receptor subtypes.
G. Lambrecht, R. Feifel, Monika Wagner-Röder, C. Strohmann +6 more
1989European Journal of Pharmacology100 citations Open access
Semantic Scholar
Development of selective agonists and antagonists for the human vasoactive intestinal polypeptide VPAC(2) receptor.
D. Moreno, P. Gourlet, P. de Neef, Johnny Cnudde +2 more
2000Peptides86 citations
Semantic Scholar
The C-terminus ends of secretin and VIP interact with the N-terminal domains of their receptors.
P. Gourlet, Jean-Pierre Vilardaga, P. de Neef, M. Waelbroeck +2 more
1996Peptides83 citations
Semantic Scholar
Two Basic Residues of the h-VPAC1 Receptor Second Transmembrane Helix Are Essential for Ligand Binding and Signal Transduction*
R. Solano, I. Langer, J. Perret, P. Vertongen +3 more
2001Journal of Biological Chemistry80 citations Open access
Semantic Scholar
Properties of chimeric secretin and VIP receptor proteins indicate the importance of the N-terminal domain for ligand discrimination.
Jean-Pierre Vilardaga, P. Deneef, E. Di Paolo, Alex Bollen +2 more
1995Biochemical and Biophysical Research Communications - BBRC78 citations
Semantic Scholar
The pituitary adenylate cyclase activating polypeptide (PACAP I) and VIP (PACAP II VIP1) receptors stimulate inositol phosphate synthesis in transfected CHO cells through interaction with different G proteins.
J. van Rampelbergh, P. Poloczek, Isabelle Françoys, C. Delporte +3 more
1997Biochimica et Biophysica Acta76 citations Open access
Semantic Scholar
A new type of functional VIP receptor has an affinity for helodermin in human SUP‐T1 lymphoblasts
P. Robberecht, M. Waelbroeck, P. de Neef, M. Tastenoy +3 more
1988FEBS Letters63 citations
Semantic Scholar
Properties of the VIP-PACAP type II receptor stably expressed in CHO cells.
Ernesto Ciccarelli, Jean-Pierre Vilardaga, P. de Neef, E. Di Paolo +3 more
1994Regulatory Peptides58 citations Open access
Semantic Scholar
Contribution of the second transmembrane helix of the secretin receptor to the positioning of secretin
E. Di Paolo, P. de Neef, N. Moguilevsky, H. Petry +3 more
1998FEBS Letters49 citations Open access
Semantic Scholar
New functionally selective muscarinic agonists.
G. Lambrecht, U. Moser, Ulrike Grimm, O. Pfaff +5 more
1993Life Science48 citations
Semantic Scholar
G protein activation by G protein coupled receptors: ternary complex formation or catalyzed reaction?
D. J. Roberts, M. Waelbroeck
2004Biochemical Pharmacology45 citations
Semantic Scholar
Propiverine and metabolites: differences in binding to muscarinic receptors and in functional models of detrusor contraction
M. Wuest, Anke Weiss, M. Waelbroeck, M. Braeter +3 more
2006Naunyn-Schmiedeberg's Archives of Pharmacology44 citations
Semantic Scholar
Binding and functional properties of antimuscarinics of the hexocyclium/sila‐hexocyclium and hexahydro‐diphenidol/hexahydro‐sila‐diphenidol type to muscarinic receptor subtypes
M. Waelbroeck, M. Tastenoy, J. Camus, J. Christophe +6 more
1989British Journal of Pharmacology43 citations Open access
Semantic Scholar
Selective labeling and localization of the M4 (m4) muscarinic receptor subtype.
G. Ferrari-DiLeo, M. Waelbroeck, Deborah C. Mash, D. D. Flynn
1994Molecular Pharmacology41 citations
Semantic Scholar
Mutational analysis of the glucagon receptor: similarities with the vasoactive intestinal peptide (VIP)/pituitary adenylate cyclase-activating peptide (PACAP)/secretin receptors for recognition of the ligand's third residue.
J. Perret, M. Van Craenenbroeck, I. Langer, P. Vertongen +3 more
2002Biochemical Journal38 citations Open access
Semantic Scholar
Interaction of amino acid residues at positions 8-15 of secretin with the N-terminal domain of the secretin receptor.
P. Gourlet, Jean-Pierre Vilardaga, P. de Neef, A. Vandermeers +3 more
1996European Journal of Biochemistry38 citations Open access
Semantic Scholar
Secretin Receptors in Human Pancreatic Membranes
P. Robberecht, P. de Neef, M. Waelbroeck, J. Camus +5 more
1988Pancreas38 citations
Semantic Scholar
Analogues of VIP, Helodermin, and PACAP Discriminate between Rat and Human VIP1 and VIP2 Receptors a
P. Gourlet, A. Vandermeers, J. Rampelbergh, P. Neef +3 more
1998Annals of the New York Academy of Sciences36 citations
Semantic Scholar
Different vasoactive intestinal polypeptide receptor domains are involved in the selective recognition of two VPAC(2)-selective ligands.
M. Juarranz, J. van Rampelbergh, P. Gourlet, P. de Neef +3 more
1999Molecular Pharmacology35 citations
Semantic Scholar
CCK and gastrin inhibit adenylate cyclase activity through a pertussis toxin‐sensitive mechanism in the tumoral rat pancreatic acinar cell line AR 4‐2J
Jean Luc Scemama, P. Robberecht, M. Waelbroeck, P. de Neef +3 more
1988FEBS Letters35 citations Open access
Semantic Scholar
DNA immunization combined with scFv phage display identifies antagonistic GCGR specific antibodies and reveals new epitopes on the small extracellular loops
B. van der Woning, G. De Boeck, C. Blanchetot, V. Bobkov +7 more
2016mAbs33 citations Open access
Semantic Scholar
Biological recognition of enantiomeric silanes: Syntheses and antimuscarinic properties of optically active (2-aminoethyl)cyclohexyl(hydroxymethyl)phenylsilanes and related quaternary ammonium derivatives
R. Tacke, D. Reichel, Martin Kropfgans, P. Jones +5 more
199531 citations
Semantic Scholar
80% of muscarinic receptors expressed by the NB‐OK 1 human neuroblastoma cell line show high affinity for pirenzepine and are comparable to rat hippocampus M1 receptors
M. Waelbroeck, J. Camus, M. Tastenoy, J. Christophe
1988FEBS Letters31 citations
Semantic Scholar
Vasoactive intestinal peptide modification at position 22 allows discrimination between receptor subtypes.
P. Gourlet, M. Vandermeers-piret, J. Rathé, P. de Neef +3 more
1998European Journal of Pharmacology29 citations
Semantic Scholar
Vasoactive intestinal polypeptide VPAC1 and VPAC2 receptor chimeras identify domains responsible for the specificity of ligand binding and activation.
M. Juarranz, J. van Rampelbergh, P. Gourlet, Phillippe De Neef +3 more
1999European Journal of Biochemistry28 citations Open access
Semantic Scholar
Vasoactive intestinal peptide (VIP) stimulates [Ca2+]iand cyclic AMPin CHO cells expressing Gα16
I. Langer, J. Perret, P. Vertongen, M. Waelbroeck +1 more
200126 citations
Semantic Scholar
Stereoselective inhibition of muscarinic receptor subtypes by the enantiomers of hexahydro‐difenidol and acetylenic analogues
R. Feifel, Monika Wagner-Röder, Carsten Strohmann, R. Tacke +4 more
1990British Journal of Pharmacology24 citations Open access
Semantic Scholar
Stereoselective recognition of the enantiomers of phenglutarimide and of six related compounds by four muscarinic receptor subtypes
M. Waelbroeck, S. Lazareno, O. Pfaff, T. Friebe +3 more
1996British Journal of Pharmacology23 citations Open access
Semantic Scholar
The (S)-(+)-enantiomer of dimethindene: a novel M2-selective muscarinic receptor antagonist.
Otmar Pfaff, Caren Hildebrandt, M. Waelbroeck, Xue-Sen Hou +3 more
1995European Journal of Pharmacology23 citations
Semantic Scholar
Motilin and erythromycin-A share a common binding site in the third transmembrane segment of the motilin receptor
Luo Xu, I. Depoortere, P. Vertongen, M. Waelbroeck +2 more
200521 citations
Semantic Scholar
Purification and sequence determination of a new muscarinic toxin (MT4) from the venom of the green mamba (Dendroaspis angusticeps).
A. Vandermeers, M. Vandermeers-piret, J. Rathé, M. Waelbroeck +3 more
1995Toxicon21 citations
Semantic Scholar
Vasoactive Intestinal Peptide Receptors in Pancreas and Liver. Structure‐Function Relationship a
J. Christophe, M. Svoboda, M. Waelbroeck, J. Winand +1 more
1988Annals of the New York Academy of Sciences21 citations
Semantic Scholar
Pharmacological discrimination between enantiomeric germanes by muscarinic receptors: a study on germanium/silicon bioisosterism
R. Tacke, D. Reichel, P. Jones, Xue-Sen Hou +4 more
199620 citations
Semantic Scholar
Mutational and Cysteine Scanning Analysis of the Glucagon Receptor N-terminal Domain*
M. Prévost, P. Vertongen, V. Raussens, D. J. Roberts +3 more
2010Journal of Biological Chemistry19 citations Open access
Semantic Scholar
Analysis of the glucagon receptor first extracellular loop by the substituted cysteine accessibility method.
D. J. Roberts, P. Vertongen, M. Waelbroeck
2011Peptides17 citations Open access
Semantic Scholar
Molecular cloning and in vitro properties of the recombinant rabbit secretin receptor.
M. Svoboda, M. Tastenoy, P. de Neef, C. Delporte +2 more
1998Peptides16 citations
Semantic Scholar
The design and pharmacology of novel selective muscarinic agonists and antagonists.
G. Lambrecht, J. Gross, Uli Hacksell, Ulrike Hermanni +8 more
1995Life Science15 citations
Semantic Scholar
Motilin and erythromycin-A share a common binding site in the third transmembrane segment of the motilin receptor.
Luo Xu, I. Depoortere, P. Vertongen, L. Thielemans +4 more
2003Biochemical Pharmacology13 citations Open access
Semantic Scholar
A Critical View of the Methods for Characterization of the VIP/PACAP Receptor Subclasses a
P. Robberecht, M. Waelbroeck
1998Annals of the New York Academy of Sciences13 citations
Semantic Scholar
Functional characterization of muscarinic receptors in rat duodenum
O. Pfaff, J. Gross, M. Waelbroeck, E. Mutschler +1 more
199513 citations
Semantic Scholar
Binding and functional properties of hexocyclium and sila‐hexocyclium derivatives to muscarinic receptor subtypes
M. Waelbroeck, J. Camus, M. Tastenoy, R. Feifel +6 more
1994British Journal of Pharmacology13 citations Open access
Semantic Scholar
Influence of monovalent cations on the binding of a charged and an uncharged (‘carbo’‐)muscarinic antagonist to muscarinic receptors
Xue-Sen Hou, J. Wehrle, W. Menge, Ernesto Ciccarelli +5 more
1996British Journal of Pharmacology12 citations Open access
Semantic Scholar
Allosteric Drugs Acting at Muscarinic Acetylcholine Receptors
M. Waelbroeck
2003Neurochemical Research10 citations
Semantic Scholar

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R. Tacke — researcher profile on SciRah