J. Coterón

Most-cited papers

1. Structure-guided lead optimization of triazolopyrimidine-ring substituents identifies potent Plasmodium falciparum dihydroorotate dehydrogenase inhibitors with clinical candidate potential

   J. Coterón, Maria Marco, J. Esquivias, Xiao-Yi Deng +21 more

   2011Journal of Medicinal Chemistry284 citations Open access

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2. Falcipain inhibitors: optimization studies of the 2-pyrimidinecarbonitrile lead series.

   J. Coterón, D. Catterick, Julia Castro, M. J. Chaparro +18 more

   2010Journal of Medicinal Chemistry105 citations

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3. An Invitation to Open Innovation in Malaria Drug Discovery: 47 Quality Starting Points from the TCAMS.

   Félix Calderón, David Barros, J. M. Bueno, J. Coterón +10 more

   2011ACS Medicinal Chemistry Letters74 citations Open access

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4. Glycophanes, cyclodextrin-cyclophane hybrid receptors for apolar binding in aqueous solutions. A stereoselective carbohydrate-carbohydrate interaction in water

   J. Coterón, Cristina Vicent, C. Bosso, S. Penadés

   199365 citations

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5. Falcipain inhibition as a promising antimalarial target.

   Maria Marco, J. Coterón

   2012Current Topics in Medicinal Chemistry64 citations

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6. A New Set of Chemical Starting Points with Plasmodium falciparum Transmission-Blocking Potential for Antimalarial Drug Discovery

   M. J. Almela, Sonia Lozano, J. Lelièvre, Gonzalo Colmenarejo +4 more

   2015PLoS ONE57 citations Open access

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7. Tetrahydro-2-naphthyl and 2-Indanyl Triazolopyrimidines Targeting Plasmodium falciparum Dihydroorotate Dehydrogenase Display Potent and Selective Antimalarial Activity

   Sreekanth Kokkonda, Xiao-Yi Deng, K. White, J. Coterón +22 more

   2016Journal of Medicinal Chemistry56 citations Open access

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8. A Replicative In Vitro Assay for Drug Discovery against Leishmania donovani

   Diana Tegazzini, Rosario Díaz, F. Aguilar, Imanol Peña +6 more

   2016Antimicrobial Agents and Chemotherapy51 citations Open access

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9. Interactions of Hydroxy Compounds and Sugars with Anions1

   J. Coterón, Frank Hacket, H. Schneider

   199650 citations

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10. Stereoselective synthesis of the antifungal GM222712

    J. M. Bueno, J. Coterón, J. Chiara, A. Fernández-Mayoralas +2 more

    200029 citations Open access

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11. Oligosaccharides Structurally Related to E-Selectin Ligands Are Inhibitors of Neural Cell Division: Synthesis, Conformational Analysis, and Biological Activity

    J. Coterón, Kamaljit Singh, J. L. Asensio, Maria Dominguez-Dalda +4 more

    199528 citations

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12. The complexation of glucose and other monosaccharides with cyclodextrins

    F. Hacket, J. Coterón, H. Schneider, V. Kazachenko

    199715 citations Open access

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13. Case Study of Small Molecules As Antimalarials: 2-Amino-1-phenylethanol (APE) Derivatives.

    M. J. Chaparro, J. Vidal, Iñigo Angulo-Barturen, J. M. Bueno +23 more

    2014ACS Medicinal Chemistry Letters14 citations Open access

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14. The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold.

    Elena Sandoval, M. Lafuente-Monasterio, M. J. Almela, Pablo Castañeda +35 more

    2017Journal of Medicinal Chemistry10 citations Open access

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15. A novel class of neutral chiral cyclophanes from α,α′-trehalose

    S. Penadés, J. Coterón

    19928 citations

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16. Stereocontrolled glycosylation of sordaricin in the presence of ammonium salts

    J. Coterón, J. Chiara, A. Fernández-Mayoralas, J. Fiandor +1 more

    20007 citations

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17. A new synthesis of 3,5-dihydroxy-7-(1-pyrrolyl)-6-heptenoic acids, a family of HMGCoA reductase inhibitors with antifungal activity

    Julia Castro, J. Coterón, M. T. Fraile, S. Garcı́a-Ochoa +2 more

    20025 citations

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18. Different reactivities of acetylated exo- and endo-cyanoethylidene derivatives in glycosylation reactions

    Cristina Vicent, J. Coterón, J. Jiménez-Barbero, M. Martín‐Lomas +1 more

    19895 citations

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19. Unravelling the rate of action of hits in the Leishmania donovani box using standard drugs amphotericin B and miltefosine

    Diana Tegazzini, J. Cantizani, Imanol Peña, Julio Martin +1 more

    2017PLoS Neglected Tropical Diseases4 citations Open access

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20. Correction to The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold.

    Elena Sandoval, M. Lafuente-Monasterio, M. J. Almela, Pablo Castañeda +35 more

    2017Journal of Medicinal Chemistry1 citations

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21. Stereoselective Synthesis of the Antifungal GM222712.

    J. M. Bueno, J. Coterón, J. Chiara, A. Fernández-Mayoralas +2 more

    20001 citations

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22. A replicative in vitro assay for drug discovery against Leishmania donovani 1

    Diana Tegazzini, Rosario Díaz, Fernando Aguilar, Imanol Peña +7 more

    20160 citations

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23. Corrections to Falcipain Inhibitors: Optimization Studies of the 2-Pyrimidinecarbonitrile Lead Series

    J. Coterón, D. Catterick, Julia Castro, M. J. Chaparro +18 more

    20100 citations

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24. A New Synthesis of 3,5-Dihydroxy-7-(1-pyrrolyl)-6-heptenoic Acids, a Family of HMGCoA Reductase Inhibitors with Antifungal Activity.

    Julia Castro, J. Coterón, M. T. Fraile, S. Garcı́a-Ochoa +2 more

    20020 citations

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25. A Novel Class of Neutral Chiral Cyclophanes from α,α′- Trehalose.

    S. Penadés, J. Coterón

    19920 citations

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