Mathieu Pizzonero

Most-cited papers

1. Discovery and optimization of an azetidine chemical series as a free fatty acid receptor 2 (FFA2) antagonist: from hit to clinic.

   Mathieu Pizzonero, S. Dupont, Marielle Babel, Stéphane Beaumont +27 more

   2014Journal of Medicinal Chemistry97 citations Open access

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2. The syntheses of rac-inthomycin A, (+)-inthomycin B and (+)-inthomycin C using a unified synthetic approach

   M. R. Webb, M. Addie, Catherine M. Crawforth, James W. Dale +4 more

   200840 citations

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3. Identification of GLPG/ABBV-2737, a Novel Class of Corrector, Which Exerts Functional Synergy With Other CFTR Modulators

   G. de Wilde, M. Gees, S. Musch, Katleen Verdonck +12 more

   2019Frontiers in Pharmacology36 citations Open access

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4. Recent Progress in the Discovery and Development of Small-Molecule Modulators of CFTR.

   P. Kym, Xue-Qing Wang, Mathieu Pizzonero, S. E. Van der Plas

   2018Progress in Medicinal Chemistry25 citations

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5. X-Ray crystal structures of potent opioid receptor ligands: etonitazene, cis-(+)-3-methylfentanyl, etorphine, diprenorphine, and buprenorphine

   Mathieu Pizzonero, J. Flippen-Anderson, C. George, Craing M. Bertha +1 more

   199417 citations Open access

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6. Discovery of Pyridones As Oral AMPK Direct Activators.

   O. Mirguet, S. Sautet, Catherine A Clément, Jérôme Toum +13 more

   2013ACS Medicinal Chemistry Letters15 citations Open access

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7. The asymmetric Michael-type alkylation of chiral β-enamino esters: critical role of a benzyl ester group in the racemization of adducts

   Mathieu Pizzonero, F. Hendra, Sandrine Delarue-Cochin, M. T. Huu-Dau +4 more

   20059 citations

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8. Enantioselective Synthesis of (R)-1-Azaspiro-[4.4]nonane-2,6-dione Ethylene Ketal, Key Chiral Intermediate in the Elaboration of (-)-Cephalotaxine

   J. d'Angelo, F. Dumas, Mathieu Pizzonero

   20057 citations Open access

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9. Crystallographic/experimental electron density characterizations and reactions with nucleophiles of beta-enaminonitriles possessing a pyrrolobenzazepine core.

   Mathieu Pizzonero, Laurent Keller, F. Dumas, M. Ourévitch +5 more

   2004Journal of Organic Chemistry6 citations Open access

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10. The Syntheses of rac-Inthomycin A, (+)-Inthomycin B and (+)-Inthomycin C Using a Unified Synthetic Approach.

    M. R. Webb, M. Addie, Catherine M. Crawforth, James W. Dale +4 more

    20083 citations

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11. Novel corrector-potentiator combinations for treating Cystic Fibrosis

    K. Conrath, C. Balut, S. Musch, A. Swensen +9 more

    20141 citations

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12. Reinvestigation of the fluoride-triggered condensation of allyltrimethylsilane with cinnamonitrile: ‘abnormal Sakurai’ and sequential ‘abnormal Sakurai’–Michael–Thorpe Ziegler side reactions

    Laurent Keller, F. Dumas, Mathieu Pizzonero, J. d'Angelo +2 more

    20021 citations

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13. Mo1234 The FFA2 Antagonist GLPG0974: A Promising Approach to Treat Neutrophil-Driven Inflammation

    F. Vanhoutte, F. Namour, S. Dupont, Mathieu Pizzonero +5 more

    20140 citations Open access

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14. CCDC 235835: Experimental Crystal Structure Determination

    Mathieu Pizzonero, Laurent Keller, F. Dumas, M. Ourévitch +5 more

    20040 citations

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15. CCDC 235834: Experimental Crystal Structure Determination

    Mathieu Pizzonero, Laurent Keller, F. Dumas, M. Ourévitch +5 more

    20040 citations

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