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A. Rampa · SciRah

Researcher profile · Semantic Scholar

A. Rampa

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A. Rampa — researcher profile on SciRah

h-index: 35
Works: 106
Citations: 3,711

Most-cited papers

3-(4-[[Benzyl(methyl)amino]methyl]phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced beta-amyloid aggregation: a dual function lead for Alzheimer's disease therapy.
Lorna Piazzi, A. Rampa, A. Bisi, S. Gobbi +6 more
2003Journal of Medicinal Chemistry237 citations Open access
Semantic Scholar
Multi-target-directed coumarin derivatives: hAChE and BACE1 inhibitors as potential anti-Alzheimer compounds.
Lorna Piazzi, A. Cavalli, Francesco Colizzi, Federica Belluti +5 more
2008Bioorganic & Medicinal Chemistry Letters205 citations Open access
Semantic Scholar
Benzofuran-based hybrid compounds for the inhibition of cholinesterase activity, beta amyloid aggregation, and abeta neurotoxicity.
S. Rizzo, C. Rivière, Lorna Piazzi, A. Bisi +7 more
2008Journal of Medicinal Chemistry178 citations Open access
Semantic Scholar
SAR of 9-amino-1,2,3,4-tetrahydroacridine-based acetylcholinesterase inhibitors: synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues.
M. Recanatini, Andrea Cavalli, Federica Belluti, Lorna Piazzi +7 more
2000Journal of Medicinal Chemistry148 citations Open access
Semantic Scholar
Phytoestrogens in Postmenopause: The State of the Art from a Chemical, Pharmacological and Regulatory Perspective
E. Poluzzi, C. Piccinni, E. Raschi, A. Rampa +2 more
2013Current Medicinal Chemistry138 citations Open access
Semantic Scholar
A new class of nonsteroidal aromatase inhibitors: design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17 alpha-hydroxylase/C17,20-lyase.
M. Recanatini, A. Bisi, A. Cavalli, Federica Belluti +6 more
2001Journal of Medicinal Chemistry113 citations Open access
Semantic Scholar
Versatility of the Curcumin Scaffold: Discovery of Potent and Balanced Dual BACE-1 and GSK-3β Inhibitors.
R. Di Martino, A. De Simone, V. Andrisano, P. Bisignano +10 more
2016Journal of Medicinal Chemistry104 citations Open access
Semantic Scholar
Targeting Alzheimer's disease: Novel indanone hybrids bearing a pharmacophoric fragment of AP2238.
S. Rizzo, M. Bartolini, L. Ceccarini, Lorna Piazzi +5 more
2010Bioorganic & Medicinal Chemistry94 citations Open access
Semantic Scholar
Lead optimization providing a series of flavone derivatives as potent nonsteroidal inhibitors of the cytochrome P450 aromatase enzyme.
S. Gobbi, A. Cavalli, A. Rampa, Federica Belluti +5 more
2006Journal of Medicinal Chemistry88 citations Open access
Semantic Scholar
Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation.
Federica Belluti, A. Rampa, Lorna Piazzi, A. Bisi +6 more
2005Journal of Medicinal Chemistry87 citations Open access
Semantic Scholar
Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives.
A. Rampa, A. Bisi, Federica Belluti, S. Gobbi +5 more
2000Bioorganic & Medicinal Chemistry84 citations Open access
Semantic Scholar
Extensive SAR and computational studies of 3-{4-[(benzylmethylamino)methyl]phenyl}-6,7-dimethoxy-2H-2-chromenone (AP2238) derivatives.
Lorna Piazzi, A. Cavalli, Federica Belluti, A. Bisi +6 more
2007Journal of Medicinal Chemistry75 citations Open access
Semantic Scholar
Synthesis and biological activity of some rigid analogues of flavone-8-acetic acid.
P. Valenti, A. Bisi, A. Rampa, Federica Belluti +3 more
2000Bioorganic & Medicinal Chemistry75 citations
Semantic Scholar
Coumarin derivatives as potential antitumor agents: Growth inhibition, apoptosis induction and multidrug resistance reverting activity.
A. Bisi, C. Cappadone, A. Rampa, G. Farruggia +7 more
2017European journal of medicinal chemistry73 citations Open access
Semantic Scholar
Fatty Acid Amide Hydrolase (FAAH), Acetylcholinesterase (AChE), and Butyrylcholinesterase (BuChE): Networked Targets for the Development of Carbamates as Potential Anti-Alzheimer's Disease Agents.
S. Montanari, L. Scalvini, M. Bartolini, Federica Belluti +8 more
2016Journal of Medicinal Chemistry71 citations Open access
Semantic Scholar
Acetylcholinesterase inhibitors: synthesis and structure-activity relationships of omega-[N-methyl-N-(3-alkylcarbamoyloxyphenyl)- methyl]aminoalkoxyheteroaryl derivatives.
A. Rampa, A. Bisi, Piero Valenti, M. Recanatini +6 more
1998Journal of Medicinal Chemistry65 citations Open access
Semantic Scholar
Cholinesterase inhibitors: SAR and enzyme inhibitory activity of 3-[omega-(benzylmethylamino)alkoxy]xanthen-9-ones.
Lorna Piazzi, Federica Belluti, A. Bisi, S. Gobbi +5 more
2007Bioorganic & Medicinal Chemistry63 citations Open access
Semantic Scholar
Enantioselective nonsteroidal aromatase inhibitors identified through a multidisciplinary medicinal chemistry approach.
A. Cavalli, A. Bisi, C. Bertucci, C. Rosini +9 more
2005Journal of Medicinal Chemistry63 citations Open access
Semantic Scholar
Small-molecule inhibitors/modulators of amyloid-β peptide aggregation and toxicity for the treatment of Alzheimer's disease: a patent review (2010 – 2012)
Federica Belluti, A. Rampa, S. Gobbi, A. Bisi
2013Expert Opinion on Therapeutic Patents62 citations
Semantic Scholar
Identification of chalcone-based antileishmanial agents targeting trypanothione reductase.
M. Ortalli, A. Ilari, G. Colotti, Ilenia De Ionna +8 more
2018European journal of medicinal chemistry61 citations Open access
Semantic Scholar
Multidrug resistance reverting activity and antitumor profile of new phenothiazine derivatives.
A. Bisi, M. Meli, S. Gobbi, A. Rampa +2 more
2008Bioorganic & Medicinal Chemistry60 citations
Semantic Scholar
Acetylcholinesterase inhibitors: SAR and kinetic studies on omega-[N-methyl-N-(3-alkylcarbamoyloxyphenyl)methyl]aminoalkoxyaryl derivatives.
A. Rampa, Lorna Piazzi, Federica Belluti, S. Gobbi +7 more
2001Journal of Medicinal Chemistry60 citations Open access
Semantic Scholar
2-Arylbenzofuran-based molecules as multipotent Alzheimer's disease modifying agents.
S. Rizzo, A. Tarozzi, M. Bartolini, G. da Costa +10 more
2012European journal of medicinal chemistry57 citations Open access
Semantic Scholar
Hybrid-based multi-target ligands for the treatment of Alzheimer's disease.
A. Rampa, Federica Belluti, S. Gobbi, A. Bisi
2011Current Topics in Medicinal Chemistry56 citations
Semantic Scholar
Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson’s Disease
R. Di Martino, L. Pruccoli, A. Bisi, S. Gobbi +9 more
2020ACS Chemical Neuroscience51 citations Open access
Semantic Scholar
Novel highly potent and selective nonsteroidal aromatase inhibitors: synthesis, biological evaluation and structure-activity relationships investigation.
S. Gobbi, Christina Zimmer, Federica Belluti, A. Rampa +3 more
2010Journal of Medicinal Chemistry51 citations Open access
Semantic Scholar
From the dual function lead AP2238 to AP2469, a multi-target-directed ligand for the treatment of Alzheimer's disease
A. Tarozzi, M. Bartolini, Lorna Piazzi, L. Valgimigli +6 more
2014Pharmacology Research & Perspectives47 citations Open access
Semantic Scholar
Benzophenone-based derivatives: a novel series of potent and selective dual inhibitors of acetylcholinesterase and acetylcholinesterase-induced beta-amyloid aggregation.
Federica Belluti, M. Bartolini, G. Bottegoni, A. Bisi +3 more
2011European journal of medicinal chemistry47 citations Open access
Semantic Scholar
Recent progress on curcumin-based therapeutics: a patent review (2012-2016). Part II: curcumin derivatives in cancer and neurodegeneration
R. Di Martino, A. Bisi, A. Rampa, S. Gobbi +1 more
2017Expert Opinion on Therapeutic Patents45 citations
Semantic Scholar
The First Dual ChE/FAAH Inhibitors: New Perspectives for Alzheimer's Disease?
A. Rampa, M. Bartolini, A. Bisi, Federica Belluti +4 more
2012ACS Medicinal Chemistry Letters39 citations Open access
Semantic Scholar
Synthesis and biological evaluation of 3-alkoxy analogues of flavone-8-acetic acid.
S. Gobbi, A. Rampa, A. Bisi, Federica Belluti +5 more
2003Journal of Medicinal Chemistry39 citations
Semantic Scholar
Discovery of novel benzofuran-based compounds with neuroprotective and immunomodulatory properties for Alzheimer's disease treatment.
S. Montanari, Ali Mokhtar Mahmoud, L. Pruccoli, Alessandro Rabbito +13 more
2019European journal of medicinal chemistry38 citations Open access
Semantic Scholar
1,4-Dihydropyridine derivatives as calcium channel modulators: the role of 3-methoxy-flavone moiety.
R. Budriesi, A. Bisi, Pierfranco Ioan, A. Rampa +5 more
2005Bioorganic & Medicinal Chemistry38 citations
Semantic Scholar
Modulation of cytochromes P450 with xanthone-based molecules: from aromatase to aldosterone synthase and steroid 11β-hydroxylase inhibition.
S. Gobbi, Qingzhong Hu, M. Negri, Christina Zimmer +4 more
2013Journal of Medicinal Chemistry37 citations Open access
Semantic Scholar
Multi-target strategy to address Alzheimer's disease: design, synthesis and biological evaluation of new tacrine-based dimers.
S. Rizzo, A. Bisi, M. Bartolini, F. Mancini +4 more
2011European journal of medicinal chemistry36 citations Open access
Semantic Scholar
From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold.
A. Rampa, F. Mancini, A. De Simone, Federico Falchi +8 more
2015Bioorganic & Medicinal Chemistry Letters34 citations Open access
Semantic Scholar
Nonsteroidal aromatase inhibitors for the treatment of breast cancer: an update.
S. Gobbi, A. Rampa, Federica Belluti, A. Bisi
2014Anti-Cancer Agents in Medicinal Chemistry34 citations
Semantic Scholar
Design, synthesis, and biological and crystallographic evaluation of novel inhibitors of Plasmodium falciparum enoyl-ACP-reductase (PfFabI).
Federica Belluti, R. Perozzo, L. Lauciello, Francesco Colizzi +9 more
2013Journal of Medicinal Chemistry34 citations Open access
Semantic Scholar
Design, synthesis, and evaluation of benzophenone derivatives as novel acetylcholinesterase inhibitors.
Federica Belluti, Lorna Piazzi, A. Bisi, S. Gobbi +4 more
2009European journal of medicinal chemistry34 citations Open access
Semantic Scholar
Reconsidering Aromatase for Breast Cancer Treatment: New Roles for an Old Target
Jessica Caciolla, A. Bisi, Federica Belluti, A. Rampa +1 more
2020Molecules33 citations Open access
Semantic Scholar
Recent progress on curcumin-based therapeutics: a patent review (2012-2016). Part I: Curcumin
R. Di Martino, B. Luppi, A. Bisi, S. Gobbi +3 more
2017Expert Opinion on Therapeutic Patents33 citations
Semantic Scholar
Multitarget Strategy to Address Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and Computational Studies of Coumarin‐Based Derivatives
S. Montanari, M. Bartolini, P. Neviani, Federica Belluti +10 more
2016ChemMedChem30 citations Open access
Semantic Scholar
Cardiovascular hybrid drugs: new benzazepinone derivatives as bradycardic agents endowed with selective beta1-non-competitive antagonism.
A. Bisi, A. Rampa, R. Budriesi, S. Gobbi +5 more
2003Bioorganic & Medicinal Chemistry30 citations
Semantic Scholar
Acetylcholinesterase inhibition by tacrine analogues
P. Valenti, A. Rampa, A. Bisi, V. Andrisano +4 more
199730 citations
Semantic Scholar
Chalcone-based carbamates for Alzheimer's disease treatment.
A. Rampa, S. Montanari, L. Pruccoli, M. Bartolini +7 more
2017Future Medicinal Chemistry28 citations
Semantic Scholar
Structure–Activity Relationships and Binding Mode in the Human Acetylcholinesterase Active Site of Pseudo‐Irreversible Inhibitors Related to Xanthostigmine
S. Rizzo, A. Cavalli, L. Ceccarini, M. Bartolini +5 more
2009ChemMedChem27 citations
Semantic Scholar
Curcumin-1,2,3-Triazole Conjugation for Targeting the Cancer Apoptosis Machinery
Francesca Seghetti, R. Di Martino, E. Catanzaro, A. Bisi +8 more
2020Molecules26 citations Open access
Semantic Scholar
Dual BACE-1/GSK-3β Inhibitors to Combat Alzheimer's Disease: A Focused Review.
A. Rampa, S. Gobbi, Rita Maria Concetta Di Martino, Federica Belluti +1 more
2018Current Topics in Medicinal Chemistry26 citations
Semantic Scholar
Synthesis and antitumor activity of new derivatives of xanthen-9-one-4-acetic acid.
S. Gobbi, A. Rampa, A. Bisi, Federica Belluti +4 more
2002Journal of Medicinal Chemistry26 citations
Semantic Scholar
Naturally Inspired Coumarin Derivatives in Alzheimer’s Disease Drug Discovery: Latest Advances and Current Challenges
Rebecca Orioli, Federica Belluti, S. Gobbi, A. Rampa +1 more
2024Molecules25 citations Open access
Semantic Scholar

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A. Bisi×46
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A. Bisi — researcher profile on SciRah
S. Gobbi×43
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S. Gobbi — researcher profile on SciRah
Federica Belluti×43
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Federica Belluti — researcher profile on SciRah
V. Andrisano×22
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M. Bartolini — researcher profile on SciRah

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A. Cavalli — researcher profile on SciRah

M. Recanatini×17

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M. Recanatini — researcher profile on SciRah

Lorna Piazzi×15

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Lorna Piazzi — researcher profile on SciRah

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P. Valenti — researcher profile on SciRah

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A. Tarozzi — researcher profile on SciRah

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S. Rizzo — researcher profile on SciRah