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S. Denoyelle · SciRah

Researcher profile · Semantic Scholar

S. Denoyelle

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S. Denoyelle — researcher profile on SciRah

h-index: 18
Works: 45
Citations: 1,135

Most-cited papers

N-Terminal Liver-Expressed Antimicrobial Peptide 2 (LEAP2) Region Exhibits Inverse Agonist Activity toward the Ghrelin Receptor.
Céline M'kadmi, Agustina Cabral, Franco Barrile, Julien Giribaldi +12 more
2018Journal of Medicinal Chemistry165 citations Open access
Semantic Scholar
Chemical Genetics Identify eIF2α Kinase Heme Regulated Inhibitor as Anti-Cancer Target
Ting Chen, D. Ozel, Yuan Qiao, Fred Harbinski +8 more
2011Nature Chemical Biology112 citations Open access
Semantic Scholar
Tumor suppression by small molecule inhibitors of translation initiation
Limo Chen, B. Aktas, Yibo Wang, Xiao-Ying He +10 more
2012OncoTarget102 citations Open access
Semantic Scholar
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling*
Céline M'kadmi, Jean-Philippe Leyris, Lauriane Onfroy, C. Galés +11 more
2015Journal of Biological Chemistry94 citations Open access
Semantic Scholar
Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex
Marjorie Damian, Sophie Mary, Mathieu Maingot, Céline M'kadmi +16 more
2015Proceedings of the National Academy of Sciences of the United States of America74 citations Open access
Semantic Scholar
GHSR-D2R heteromerization modulates dopamine signaling through an effect on G protein conformation
Marjorie Damian, V. Pons, P. Renault, Céline M'kadmi +18 more
2018Proceedings of the National Academy of Sciences of the United States of America69 citations Open access
Semantic Scholar
The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist
A. Moulin, Luc Brunel, D. Boeglin, Luc Demange +5 more
2012Amino Acids67 citations
Semantic Scholar
In Vitro inhibition of translation initiation by N,N’-diarylureas – Potential anti-cancer agents
S. Denoyelle, Ting Chen, Limo Chen, Yibo Wang +4 more
2011Bioorganic & Medicinal Chemistry Letters49 citations Open access
Semantic Scholar
Allosteric modulation of ghrelin receptor signaling by lipids
Marjorie Damian, M. Louet, A. A. Gomes, Céline M'kadmi +8 more
2021Nature Communications45 citations Open access
Semantic Scholar
Circulating ghrelin crosses the blood-cerebrospinal fluid barrier via growth hormone secretagogue receptor dependent and independent mechanisms.
Maia Uriarte, P. D. De Francesco, Gimena Fernandez, D. Castrogiovanni +8 more
2021Molecular and Cellular Endocrinology42 citations Open access
Semantic Scholar
Development of a novel fluorescent ligand of growth hormone secretagogue receptor based on the N-Terminal Leap2 region.
Franco Barrile, Céline M'kadmi, P. D. De Francesco, Agustina Cabral +11 more
2019Molecular and Cellular Endocrinology38 citations Open access
Semantic Scholar
GHSR controls food deprivation-induced activation of CRF neurons of the hypothalamic paraventricular nucleus in a LEAP2-dependent manner
Gimena Fernandez, Agustina Cabral, P. D. De Francesco, Maia Uriarte +10 more
2022Cellular and Molecular Life Sciences34 citations Open access
Semantic Scholar
LEAP2 Impairs the Capability of the Growth Hormone Secretagogue Receptor to Regulate the Dopamine 2 Receptor Signaling
E. R. Mustafá, Santiago Cordisco González, Marjorie Damian, S. Cantel +7 more
2021Frontiers in Pharmacology31 citations Open access
Semantic Scholar
Selective C-acylation of 2-aminoimidazo[1,2-a]pyridine: application to the synthesis of imidazopyridine-fused [1,3]diazepinones.
Nicolas Masurier, Roberta Aruta, V. Gaumet, S. Denoyelle +4 more
2012Journal of Organic Chemistry31 citations
Semantic Scholar
Synthesis and preliminary biological studies of hemifluorinated bifunctional bolaamphiphiles designed for gene delivery
S. Denoyelle, A. Polidori, M. Brunelle, P. Vuillaume +3 more
200627 citations
Semantic Scholar
Synthesis and SAR study of novel 3,3-diphenyl-1,3-dihydroindol-2-one derivatives as potent eIF2·GTP·Met-tRNAiMet ternary complex inhibitors.
S. Denoyelle, Ting Chen, Hongwei Yang, Limo Chen +4 more
2013European journal of medicinal chemistry23 citations
Semantic Scholar
A structure–activity investigation of hemifluorinated bifunctional bolaamphiphiles designed for gene delivery
M. Brunelle, A. Polidori, S. Denoyelle, A. Fabiano +3 more
200923 citations Open access
Semantic Scholar
Growth hormone secretagogues modulate inflammation and fibrosis in mdx mouse model of Duchenne muscular dystrophy
Brigida Boccanegra, O. Cappellari, P. Mantuano, Daniela Trisciuzzi +17 more
2023Frontiers in Immunology20 citations Open access
Semantic Scholar
Design and synthesis of amidoxime derivatives for orally potent C-alkylamidine-based antimalarial agents.
M. Ouattara, S. Wein, S. Denoyelle, S. Ortial +4 more
2009Bioorganic & Medicinal Chemistry Letters17 citations
Semantic Scholar
Evaluation of amidoxime derivatives as prodrug candidates of potent bis-cationic antimalarials.
O. Berger, S. Ortial, S. Wein, S. Denoyelle +5 more
2019Bioorganic & Medicinal Chemistry Letters13 citations Open access
Semantic Scholar
A Novel Truncated Liver Enriched Antimicrobial Peptide-2 Palmitoylated at its N-Terminal Antagonizes Effects of Ghrelin
L. Holá, B. Železná, A. Karnošová, J. Kuneš +7 more
2022Journal of Pharmacology and Experimental Therapeutics12 citations Open access
Semantic Scholar
Development of non-peptidic inverse agonists of the ghrelin receptor (GHSR) based on the 1,2,4-triazole scaffold.
Khoubaib Ben Haj Salah, Mathieu Maingot, A. Blayo, Céline M'kadmi +13 more
2020Journal of Medicinal Chemistry11 citations Open access
Semantic Scholar
New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center.
Mathieu Maingot, A. Blayo, S. Denoyelle, Céline M'kadmi +13 more
2016Bioorganic & Medicinal Chemistry Letters7 citations Open access
Semantic Scholar
New trisubstituted 1,2,4-triazoles as ghrelin receptor antagonists.
A. Blayo, Mathieu Maingot, B. Aicher, Céline M'kadmi +8 more
2015Bioorganic & Medicinal Chemistry Letters7 citations Open access
Semantic Scholar
Synthesis and Evaluation of Hybrid Bis‐cationic Salts as Antimalarial Drugs
S. Ortial, S. Denoyelle, S. Wein, O. Berger +5 more
2010ChemMedChem7 citations
Semantic Scholar
Concerted conformational dynamics and water movements in the ghrelin G protein-coupled receptor
M. Louet, Marina Casiraghi, Marjorie Damian, Maurício G. S. Costa +14 more
2021eLife6 citations Open access
Semantic Scholar
Synthesis of [1,2,4]Triazolo[4,3- a]piperazin-6-ones: An Approach to the Triazole-Fused Ketopiperazine Scaffold.
Khoubaib Ben Haj Salah, Baptiste Legrand, Mathieu Bibian, E. Wenger +2 more
2018Organic Letters6 citations
Semantic Scholar
Synthesis of Thieno[3,2‐e][1,4]diazepin‐2‐ones: Application of an Uncatalysed Pictet–Spengler Reaction
S. Denoyelle, Guillaume Tambutet, Nicolas Masurier, L. Maillard +2 more
20155 citations
Semantic Scholar
Design and Characterization of a Triazole-Based Growth Hormone Secretagogue Receptor Modulator Inhibiting the Glucoregulatory and Feeding Actions of Ghrelin.
S. Péraldi-Roux, Morgane Bayle, Céline M'kadmi, Marjorie Damian +12 more
2022Biochemical Pharmacology3 citations Open access
Semantic Scholar
Novel insights into the effects of JMV2894, a growth hormone secretagogue, in Duchenne muscular dystrophy: A preclinical study in the D2-mdx mouse model.
P. Mantuano, Brigida Boccanegra, Manuel Marinelli, Enrica Cristiano +11 more
2025Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie1 citations Open access
Semantic Scholar
Role of Symmetry in 3,3-Diphenyl-1,3-dihydroindol-2-one Derivatives as Inhibitors of Translation Initiation
Hongwei Yang, Ting Chen, S. Denoyelle, Limo Chen +5 more
2022Bioorganic & Medicinal Chemistry Letters1 citations Open access
Semantic Scholar
CP-231 Implementation of medication reconciliation on admission in a psychiatric hospital: who comes first?
S. Denoyelle, O. Bureš, A. Fischer
20171 citations
Semantic Scholar
From Design to Outcome: The Role of Bi‐ and Multifunctional Ligands in Modern Therapeutics
Célia Bouacha, S. Denoyelle, S. Cantel
20250 citations Open access
Semantic Scholar
A novel truncated LEAP2 palmitoylated at its N-terminal antagonizes effects of ghrelin
L. Holá, B. Železná, A. Karnošová, J. Kuneš +7 more
20220 citations
Semantic Scholar
A novel truncated LEAP2 palmitoylated at its N-terminal antagonizes effects of ghrelin
L. Holá, B. Železná, A. Karnošová, J. Kuneš +7 more
20220 citations
Semantic Scholar
A novel truncated LEAP2 palmitoylated at its N-terminal antagonizes effects of ghrelin
L. Holá, B. Železná, A. Karnošová, J. Kuneš +7 more
20220 citations
Semantic Scholar
A novel truncated LEAP2 palmitoylated at its N-terminal antagonizes effects of ghrelin
L. Holá, B. Železná, A. Karnošová, J. Kuneš +7 more
20220 citations
Semantic Scholar
VP.84 Growth hormone secretagogues in Duchenne muscular dystrophy: a preclinical evaluation of potential benefits on muscle function and morphology
P. Mantuano, B. Boccanegra, O. Cappellari, S. Cirmi +8 more
2022Neuromuscular Disorders0 citations
Semantic Scholar
A novel truncated LEAP2 palmitoylated at its N-terminal antagonizes effects of ghrelin
L. Holá, B. Železná, A. Karnošová, J. Kuneš +7 more
20220 citations
Semantic Scholar
A novel truncated LEAP2 palmitoylated at its N-terminal antagonizes effects of ghrelin
L. Holá, B. Železná, A. Karnošová, J. Kuneš +7 more
20220 citations
Semantic Scholar
Author response: Concerted conformational dynamics and water movements in the ghrelin G protein-coupled receptor
M. Louet, Marina Casiraghi, Marjorie Damian, Maurício G. S. Costa +14 more
20210 citations Open access
Semantic Scholar
DMD – ANIMAL MODELS
P. Mantuano, B. Boccanegra, E. Bresciani, F. Sanarica +7 more
2021Neuromuscular Disorders0 citations Open access
Semantic Scholar
Ghrelin receptor ligands: from the bench to the drug on the market
J. Fehrentz, Céline M'kadmi, Marjorie Damian, Sophie Mary +8 more
20180 citations Open access
Semantic Scholar
Synthesis of Thieno[3,2‐e][1,4]diazepin‐2‐ones: Application of an Uncatalyzed Pictet—Spengler Reaction.
S. Denoyelle, Guillaume Tambutet, Nicolas Masurier, L. Maillard +2 more
20160 citations
Semantic Scholar
New cationic vectors bolaforms hemifluorocarbones and applications
Ange Polidor, B. Pucci, S. Denoyelle, J. Salles
20050 citations
Semantic Scholar

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J. Fehrentz×21
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S. Cantel×18
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Céline M'kadmi×14
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Marjorie Damian×13
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Khoubaib Ben Haj Salah×7

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