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J. A. Cisneros · SciRah

Researcher profile · Semantic Scholar

J. A. Cisneros

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J. A. Cisneros — researcher profile on SciRah

h-index: 17
Works: 23
Citations: 868

Most-cited papers

Identification of a Novel Endocannabinoid-Hydrolyzing Enzyme Expressed by Microglial Cells
G. Muccioli, Cong Xu, E. Odah, E. Cudaback +5 more
2007Journal of Neuroscience167 citations Open access
Semantic Scholar
The constitutive production of the endocannabinoid 2‐arachidonoylglycerol participates in oligodendrocyte differentiation
Ó. Gómez, A. Arevalo‐Martin, D. Garcia-Ovejero, S. Ortega-Gutiérrez +5 more
2010Glia93 citations
Semantic Scholar
Design, Synthesis, and Protein Crystallography of Biaryltriazoles as Potent Tautomerase Inhibitors of Macrophage Migration Inhibitory Factor
P. Dziedzic, J. A. Cisneros, M. Robertson, Alissa A. Hare +3 more
2015Journal of the American Chemical Society64 citations Open access
Semantic Scholar
Crystal Structures of HIV-1 Reverse Transcriptase with Picomolar Inhibitors Reveal Key Interactions for Drug Design
K. Frey, Mariela Bollini, A. Mislak, J. A. Cisneros +3 more
2012Journal of the American Chemical Society54 citations Open access
Semantic Scholar
Covalent inhibitors for eradication of drug-resistant HIV-1 reverse transcriptase: From design to protein crystallography
A. Chan, Won-Gil Lee, K. Spasov, J. A. Cisneros +5 more
2017Proceedings of the National Academy of Sciences of the United States of America47 citations Open access
Semantic Scholar
From in silico hit to long-acting late-stage preclinical candidate to combat HIV-1 infection
S. Kudalkar, J. Beloor, E. Quijano, K. Spasov +6 more
2017Proceedings of the National Academy of Sciences of the United States of America37 citations Open access
Semantic Scholar
Extension into the entrance channel of HIV-1 reverse transcriptase – crystallography and enhanced solubility
Mariela Bollini, K. Frey, J. A. Cisneros, K. Spasov +5 more
2013Bioorganic & Medicinal Chemistry Letters37 citations Open access
Semantic Scholar
Systematic Study of Effects of Structural Modifications on the Aqueous Solubility of Drug-like Molecules.
J. A. Cisneros, M. Robertson, Brandon Q. Mercado, W. L. Jorgensen
2017ACS Medicinal Chemistry Letters36 citations Open access
Semantic Scholar
Structural studies provide clues for analog design of specific inhibitors of Cryptosporidium hominis Thymidylate Synthase-Dihydrofolate Reductase
V. P. Kumar, J. A. Cisneros, K. Frey, Alejandro Castellanos-González +5 more
2014Bioorganic & Medicinal Chemistry Letters34 citations Open access
Semantic Scholar
A Fluorescence Polarization Assay for Binding to Macrophage Migration Inhibitory Factor and Crystal Structures for Complexes of Two Potent Inhibitors
J. A. Cisneros, M. Robertson, M. Valhondo, W. L. Jorgensen
2016Journal of the American Chemical Society33 citations Open access
Semantic Scholar
Optimization of diarylazines as anti-HIV agents with dramatically enhanced solubility
Mariela Bollini, J. A. Cisneros, K. Spasov, K. Anderson +1 more
2013Bioorganic & Medicinal Chemistry Letters33 citations Open access
Semantic Scholar
Structure-activity relationship of a new series of reversible dual monoacylglycerol lipase/fatty acid amide hydrolase inhibitors.
J. A. Cisneros, Emmelie Björklund, I. González-Gil, Yan-Ling Hu +6 more
2012Journal of Medicinal Chemistry33 citations Open access
Semantic Scholar
Dual Inhibition of α/β-Hydrolase Domain 6 and Fatty Acid Amide Hydrolase Increases Endocannabinoid Levels in Neurons*
William R. Marrs, Eric A. Horne, S. Ortega-Gutiérrez, J. A. Cisneros +5 more
2011Journal of Biological Chemistry31 citations Open access
Semantic Scholar
JAK2 JH2 Fluorescence Polarization Assay and Crystal Structures for Complexes with Three Small Molecules.
Ana S. Newton, L. Deiana, D. Puleo, J. A. Cisneros +3 more
2017ACS Medicinal Chemistry Letters28 citations Open access
Semantic Scholar
The medicinal chemistry of agents targeting monoacylglycerol lipase.
S. Ortega-Gutiérrez, A. Viso, J. A. Cisneros
2008Current Topics in Medicinal Chemistry26 citations
Semantic Scholar
Covalent Inhibition of Wild-Type HIV-1 Reverse Transcriptase Using a Fluorosulfate Warhead.
J. Ippolito, Haichan Niu, N. Bertoletti, Z. Carter +7 more
2021ACS Medicinal Chemistry Letters24 citations Open access
Semantic Scholar
Irregularities in enzyme assays: The case of macrophage migration inhibitory factor.
J. A. Cisneros, M. Robertson, M. Valhondo, W. L. Jorgensen
2016Bioorganic & Medicinal Chemistry Letters22 citations Open access
Semantic Scholar
Structural and Pharmacological Evaluation of a Novel Non-nucleoside Reverse Transcriptase Inhibitor as a Promising Long Acting Nanoformulation for Treating HIV
S. Kudalkar, Irfan Ullah, N. Bertoletti, Hanna K. Mandl +8 more
2019Antiviral Research17 citations Open access
Semantic Scholar
A nanotherapy strategy significantly enhances anticryptosporidial activity of an inhibitor of bifunctional thymidylate synthase-dihydrofolate reductase from Cryptosporidium
A. Mukerjee, P. Iyidogan, Alejandro Castellanos-González, J. A. Cisneros +6 more
2015Bioorganic & Medicinal Chemistry Letters16 citations Open access
Semantic Scholar
Optimization of Pyrazoles as Phenol Surrogates to Yield Potent Inhibitors of Macrophage Migration Inhibitory Factor
Vinay Trivedi-Parmar, M. Robertson, J. A. Cisneros, S. Krimmer +1 more
2018ChemMedChem14 citations Open access
Semantic Scholar
Structure-activity relationship of a series of inhibitors of monoacylglycerol hydrolysis--comparison with effects upon fatty acid amide hydrolase.
J. A. Cisneros, S. Vandevoorde, S. Ortega-Gutiérrez, C. Paris +2 more
2007Journal of Medicinal Chemistry13 citations Open access
Semantic Scholar
Adding a Hydrogen Bond May Not Help: Naphthyridinone vs Quinoline Inhibitors of Macrophage Migration Inhibitory Factor.
Thomas K Dawson, P. Dziedzic, M. Robertson, J. A. Cisneros +4 more
2017ACS Medicinal Chemistry Letters10 citations Open access
Semantic Scholar
Reply to Pandey et al.: Understanding the efficacy of a potential antiretroviral drug candidate in humanized mouse model of HIV infection
S. Kudalkar, J. Beloor, E. Quijano, K. Spasov +6 more
2018Proceedings of the National Academy of Sciences of the United States of America0 citations Open access
Semantic Scholar

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