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P. Falson · SciRah

Researcher profile · Semantic Scholar

P. Falson

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P. Falson — researcher profile on SciRah

h-index: 29
Works: 122
Citations: 2,795

Most-cited papers

A new method for the reconstitution of membrane proteins into giant unilamellar vesicles.
P. Girard, J. Pécréaux, G. Lenoir, P. Falson +2 more
2004Biophysical Journal256 citations Open access
Semantic Scholar
Structures of P-glycoprotein reveal its conformational flexibility and an epitope on the nucleotide-binding domain
A. Ward, P. Szewczyk, Vinciane Grimard, Chang-wook Lee +12 more
2013Proceedings of the National Academy of Sciences of the United States of America246 citations Open access
Semantic Scholar
ABCG2 Transports and Transfers Heme to Albumin through Its Large Extracellular Loop*
Élodie Desuzinges-Mandon, Ophélie Arnaud, L. Martínez, F. Huché +2 more
2010Journal of Biological Chemistry91 citations Open access
Semantic Scholar
Structuring Detergents for Extracting and Stabilizing Functional Membrane Proteins
Rima Matar-Merheb, M. Rhimi, A. Leydier, F. Huché +10 more
2011PLoS ONE80 citations Open access
Semantic Scholar
Quantification of Detergents Complexed with Membrane Proteins
V. Chaptal, F. Delolme, A. Kilburg, S. Magnard +16 more
2017Scientific Reports71 citations Open access
Semantic Scholar
UNDERSTANDING POLYSPECIFICITY WITHIN THE SUBSTRATE-BINDING CAVITY OF THE HUMAN MULTIDRUG RESISTANCE P-GLYCOPROTEIN
L. Martínez, Ophélie Arnaud, E. Hénin, Hou-Chao Tao +9 more
2014The FEBS Journal66 citations Open access
Semantic Scholar
Hepatitis C Virus Envelope Glycoprotein E1 Forms Trimers at the Surface of the Virion
P. Falson, B. Bartosch, K. Alsaleh, B. Tews +11 more
2015Journal of Virology65 citations Open access
Semantic Scholar
Methoxy stilbenes as potent, specific, untransported, and noncytotoxic inhibitors of breast cancer resistance protein.
G. Valdameri, Luciana Pereira Rangel, C. Spatafora, J. Guitton +8 more
2012ACS Chemical Biology57 citations
Semantic Scholar
Unprecedented inhibition of P-gp activity by a novel rutheniumcyclopentadienyl compound bearing a bipyridine-biotin ligand
L. Côrte-Real, B. F. Karas, Patrícia Gírio, Alexis Moreno +8 more
2018European journal of medicinal chemistry44 citations Open access
Semantic Scholar
5‐Oxo‐hexahydroquinoline derivatives as modulators of P‐gp, MRP1 and BCRP transporters to overcome multidrug resistance in cancer cells
S. Ranjbar, Ruttiros Khonkarn, Alexis Moreno, H. Baubichon-Cortay +6 more
2019Toxicology and Applied Pharmacology43 citations
Semantic Scholar
Substrate-bound and substrate-free outward-facing structures of a multidrug ABC exporter
V. Chaptal, V. Zampieri, B. Wiseman, C. Orelle +16 more
2022Science Advances41 citations Open access
Semantic Scholar
The acridone derivative MBLI-87 sensitizes breast cancer resistance protein-expressing xenografts to irinotecan
O. Arnaud, A. Boumendjel, A. Gèze, M. Honorat +8 more
2011European Journal of Cancer41 citations Open access
Semantic Scholar
Targeting the multidrug ABCG2 transporter with flavonoidic inhibitors: in vitro optimization and in vivo validation.
A. Boumendjel, S. Macalou, G. Valdameri, A. Pozza +9 more
2011Current Medicinal Chemistry41 citations
Semantic Scholar
Molecular analysis of the massive GSH transport mechanism mediated by the human Multidrug Resistant Protein 1/ABCC1
Rachad Nasr, Doriane Lorendeau, Ruttiros Khonkarn, Lauriane Dury +6 more
2020Scientific Reports39 citations Open access
Semantic Scholar
Methyl-cyclopentadienyl Ruthenium Compounds with 2,2'-Bipyridine Derivatives Display Strong Anticancer Activity and Multidrug Resistance Potential.
L. Côrte-Real, Ricardo G. Teixeira, Patrícia Gírio, Elisabeta Comsa +11 more
2018Inorganic Chemistry35 citations Open access
Semantic Scholar
MRP1-dependent Collateral Sensitivity of Multidrug-resistant Cancer Cells: Identifying Selective Modulators Inducing Cellular Glutathione Depletion.
Doriane Lorendeau, Lauriane Dury, Rachad Nasr, A. Boumendjel +5 more
2017Current Medicinal Chemistry35 citations
Semantic Scholar
PDR-like ABC systems in pathogenic fungi.
Alexis Moreno, A. Banerjee, R. Prasad, P. Falson
2019Research in Microbiology34 citations Open access
Semantic Scholar
Functional Properties of Sarcoplasmic Reticulum Ca2+-ATPase after Proteolytic Cleavage at Leu119-Lys120, Close to the A-domain
G. Lenoir, M. Picard, Carole Gauron, C. Montigny +5 more
2004Journal of Biological Chemistry34 citations Open access
Semantic Scholar
The first ADC bearing the ferroptosis inducer RSL3 as a payload with conservation of the fragile electrophilic warhead.
K. Nguyen, L. Conilh, P. Falson, C. Dumontet +1 more
2022European journal of medicinal chemistry32 citations Open access
Semantic Scholar
Flavonoid dimers are highly potent killers of multidrug resistant cancer cells overexpressing MRP1
Lauriane Dury, Rachad Nasr, Doriane Lorendeau, Elisabeta Comsa +8 more
2017Biochemical Pharmacology31 citations
Semantic Scholar
Potent and fully noncompetitive peptidomimetic inhibitor of multidrug resistance P-glycoprotein.
Ophélie Arnaud, Ali Koubeissi, L. Ettouati, R. Terreux +6 more
2010Journal of Medicinal Chemistry30 citations Open access
Semantic Scholar
The multidrug resistance half-transporter ABCG2 is purified as a tetramer upon selective extraction from membranes.
Manuela Dezi, Pierre-Frédéric Fribourg, Aurélie Di Cicco, Ophélie Arnaud +4 more
2010Biochimica et Biophysica Acta30 citations Open access
Semantic Scholar
Optimizing the flavanone core toward new selective nitrogen-containing modulators of ABC transporters.
Ricardo J. Ferreira, Rafael Baptista, Alexis Moreno, P. G. Madeira +5 more
2018Future Medicinal Chemistry29 citations
Semantic Scholar
Monoterpene indole alkaloid azine derivatives as MDR reversal agents.
Angela Paterna, Ruttiros Khonkarn, S. Mulhovo, Alexis Moreno +4 more
2018Bioorganic & Medicinal Chemistry28 citations Open access
Semantic Scholar
Directed Mutational Strategies Reveal Drug Binding and Transport by the MDR Transporters of Candida albicans
A. Banerjee, Jorgaq Pata, S. Sharma, B. Monk +2 more
2021Journal of Fungi27 citations Open access
Semantic Scholar
Efficient and stable reconstitution of the ABC transporter BmrA for solid-state NMR studies
Britta Kunert, C. Gardiennet, Denis Lacabanne, Daniel Calles-Garcia +5 more
2014Frontiers in Molecular Biosciences26 citations Open access
Semantic Scholar
Polymer "ruthenium-cyclopentadienyl" conjugates - New emerging anti-cancer drugs.
Tiago Moreira, Rita Francisco, Elisabeta Comsa, Sophie Duban-Deweer +12 more
2019European journal of medicinal chemistry24 citations Open access
Semantic Scholar
Glycosyl-Substituted Dicarboxylates as Detergents for the Extraction, Overstabilization, and Crystallization of Membrane Proteins.
K. Nguyen, Marine Peuchmaur, S. Magnard, R. Haudecoeur +9 more
2018Angewandte Chemie24 citations
Semantic Scholar
Structure, function, and inhibition of catalytically asymmetric ABC transporters: Lessons from the PDR subfamily.
A. Banerjee, Jorgaq Pata, V. Chaptal, A. Boumendjel +2 more
2023Drug resistance updates23 citations Open access
Semantic Scholar
Synthesis and Anticancer Cytotoxicity of Azaaurones Overcoming Multidrug Resistance
S. Tóth, Áron Szepesi, Viet-Khoa Tran-Nguyen, B. Sarkadi +5 more
2020Molecules22 citations Open access
Semantic Scholar
2-Indolylmethylenebenzofuranones as first effective inhibitors of ABCC2.
Elisabeta Baiceanu, K. Nguyen, L. Gonzalez-Lobato, Rachad Nasr +7 more
2016European journal of medicinal chemistry22 citations Open access
Semantic Scholar
Mammalian membrane protein expression in baculovirus-infected insect cells.
Céline Trometer, P. Falson
2010Methods in molecular biology22 citations
Semantic Scholar
Cdr1p highlights the role of the non-hydrolytic ATP-binding site in driving drug translocation in asymmetric ABC pumps.
A. Banerjee, Alexis Moreno, M. Khan, Remya Nair +7 more
2019Biochimica et Biophysica Acta - Biomembranes21 citations Open access
Semantic Scholar
Involvement of the L6–7 Loop in SERCA1a Ca2+-ATPase Activation by Ca2+ (or Sr2+) and ATP*
G. Lenoir, M. Picard, J. Møller, M. le Maire +2 more
2004Journal of Biological Chemistry21 citations Open access
Semantic Scholar
Ovarian cancer cells cisplatin sensitization agents selected by mass cytometry target ABCC2 inhibition.
Elisabeta Comsa, K. Nguyen, F. Loghin, A. Boumendjel +3 more
2018Future Medicinal Chemistry20 citations
Semantic Scholar
Molecular Basis of Substrate Polyspecificity of the Candida albicans Mdr1p Multidrug/H+ Antiporter.
A. K. Redhu, A. Banerjee, A. H. Shah, Alexis Moreno +4 more
2018Journal of Molecular Biology20 citations
Semantic Scholar
Atomic modelling and systematic mutagenesis identify residues in multiple drug binding sites that are essential for drug resistance in the major Candida transporter Cdr1.
Shweta Nim, L. Lobato, Alexis Moreno, V. Chaptal +3 more
2016Biochimica et Biophysica Acta20 citations Open access
Semantic Scholar
Modulators of the human ABCC2: hope from natural sources?
Elisabeta Baiceanu, G. Crișan, F. Loghin, P. Falson
2015Future Medicinal Chemistry20 citations
Semantic Scholar
Stubborn Contaminants: Influence of Detergents on the Purity of the Multidrug ABC Transporter BmrA
B. Wiseman, A. Kilburg, V. Chaptal, Gina Catalina Reyes-Mejia +3 more
2014PLoS ONE20 citations Open access
Semantic Scholar
Identification of pyrrolopyrimidine derivative PP-13 as a novel microtubule-destabilizing agent with promising anticancer properties
P. Gilson, F. Josa-Prado, C. Beauvineau, Delphine Naud-Martin +10 more
2017Scientific Reports19 citations Open access
Semantic Scholar
Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2.
Nathalie Guragossian, B. Belhani, Alexis Moreno, M. Nunes +13 more
2020European journal of medicinal chemistry18 citations Open access
Semantic Scholar
Peroxisomal ATP-binding cassette transporters form mainly tetramers
F. Geillon, C. Gondcaille, Q. Raas, Alexandre M. M. Dias +7 more
2017Journal of Biological Chemistry18 citations Open access
Semantic Scholar
W1038 near D-loop of NBD2 is a focal point for inter-domain communication in multidrug transporter Cdr1 of Candida albicans.
A. Banerjee, A. H. Shah, A. K. Redhu, Alexis Moreno +2 more
2018Biochimica et Biophysica Acta - Biomembranes17 citations Open access
Semantic Scholar
Trianionic calix[4]arene monoalkoxy derivatives : synthesis, solid-state structures and self-assembly properties
K. Suwińska, O. Shkurenko, C. Mbemba, A. Leydier +4 more
200817 citations
Semantic Scholar
The Binding Mechanism of the Yeast F1-ATPase Inhibitory Peptide
Vincent Corvest, C. Sigalat, R. Venard, P. Falson +2 more
2005Journal of Biological Chemistry17 citations Open access
Semantic Scholar
Structural insight into the cooperativity between catalytic and noncatalytic sites of F1-ATPase.
P. Falson, A. Goffeau, M. Boutry, J. Jault
2004Biochimica et Biophysica Acta17 citations Open access
Semantic Scholar
Chromones bearing amino acid residues: Easily accessible and potent inhibitors of the breast cancer resistance protein ABCG2.
Emile Roussel, Alexis Moreno, Nicolas Altounian, C. Philouze +5 more
2020European journal of medicinal chemistry16 citations Open access
Semantic Scholar
Stoichiometry of the MexA‐OprM binding, as investigated by blue native gel electrophoresis
Y. Ferrandez, L. Monlezun, G. Phan, H. Benabdelhak +6 more
2012Electrophoresis16 citations
Semantic Scholar
Multidrug resistance ABC transporter structure predictions by homology modeling approaches.
Myléne Honorat, P. Falson, R. Terreux, A. di Pietro +2 more
2011Current drug metabolism16 citations
Semantic Scholar
Modulators of the Efflux Pump Cdr1p of Candida albicans: Mechanisms of Action and Chemical Features.
Viet-Khoa Tran-Nguyen, R. Prasad, P. Falson, A. Boumendjel
2017Current Medicinal Chemistry15 citations
Semantic Scholar

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