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A. Bolasco · SciRah

Researcher profile · Semantic Scholar

A. Bolasco

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A. Bolasco — researcher profile on SciRah

h-index: 43
Works: 111
Citations: 4,256

Most-cited papers

Chalcones: a valid scaffold for monoamine oxidases inhibitors.
F. Chimenti, R. Fioravanti, A. Bolasco, P. Chimenti +6 more
2009Journal of Medicinal Chemistry191 citations Open access
Semantic Scholar
Synthesis, molecular modeling, and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins.
F. Chimenti, D. Secci, A. Bolasco, P. Chimenti +7 more
2009Journal of Medicinal Chemistry159 citations Open access
Semantic Scholar
A novel histone acetyltransferase inhibitor modulating Gcn5 network: cyclopentylidene-[4-(4'-chlorophenyl)thiazol-2-yl)hydrazone.
F. Chimenti, B. Bizzarri, E. Maccioni, D. Secci +9 more
2009Journal of Medicinal Chemistry141 citations
Semantic Scholar
Selective MAO-B inhibitors: a lesson from natural products
S. Carradori, Melissa D'Ascenzio, P. Chimenti, D. Secci +1 more
2013Molecular diversity136 citations
Semantic Scholar
Quercetin as the active principle of Hypericum hircinum exerts a selective inhibitory activity against MAO-A: extraction, biological analysis, and computational study.
F. Chimenti, F. Cottiglia, L. Bonsignore, L. Casu +13 more
2006Journal of Natural Products120 citations Open access
Semantic Scholar
Synthesis of some pyrazole derivatives and preliminary investigation of their affinity binding to P-glycoprotein.
F. Manna, F. Chimenti, R. Fioravanti, A. Bolasco +4 more
2005Bioorganic & Medicinal Chemistry Letters117 citations
Semantic Scholar
Synthesis and biological evaluation of N-substituted-3,5-diphenyl-2-pyrazoline derivatives as cyclooxygenase (COX-2) inhibitors.
R. Fioravanti, A. Bolasco, F. Manna, F. Rossi +4 more
2010European journal of medicinal chemistry113 citations Open access
Semantic Scholar
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)- pyrazole derivatives.
F. Chimenti, E. Maccioni, D. Secci, A. Bolasco +10 more
2005Journal of Medicinal Chemistry111 citations Open access
Semantic Scholar
Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides.
F. Chimenti, B. Bizzarri, A. Bolasco, D. Secci +7 more
2010Bioorganic & Medicinal Chemistry Letters108 citations
Semantic Scholar
The state of the art of pyrazole derivatives as monoamine oxidase inhibitors and antidepressant/anticonvulsant agents.
D. Secci, A. Bolasco, P. Chimenti, S. Carradori
2011Current Medicinal Chemistry106 citations
Semantic Scholar
Synthesis and selective inhibitory activity of 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives against monoamine oxidase.
F. Chimenti, A. Bolasco, F. Manna, D. Secci +7 more
2004Journal of Medicinal Chemistry99 citations Open access
Semantic Scholar
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives.
D. Secci, S. Carradori, A. Bolasco, P. Chimenti +3 more
2011European journal of medicinal chemistry95 citations Open access
Semantic Scholar
Inhibition of amine oxidases activity by 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives.
F. Manna, F. Chimenti, A. Bolasco, D. Secci +6 more
2002Bioorganic & Medicinal Chemistry Letters93 citations Open access
Semantic Scholar
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors.
F. Chimenti, R. Fioravanti, A. Bolasco, P. Chimenti +9 more
2010Bioorganic & Medicinal Chemistry92 citations Open access
Semantic Scholar
Inhibition of monoamine oxidases by coumarin-3-acyl derivatives: biological activity and computational study.
F. Chimenti, D. Secci, A. Bolasco, P. Chimenti +5 more
2004Bioorganic & Medicinal Chemistry Letters92 citations Open access
Semantic Scholar
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents.
F. Chimenti, B. Bizzarri, A. Bolasco, D. Secci +6 more
2011European journal of medicinal chemistry88 citations
Semantic Scholar
Homoisoflavonoids: natural scaffolds with potent and selective monoamine oxidase-B inhibition properties.
N. Desideri, A. Bolasco, R. Fioravanti, Luca Proietti Monaco +4 more
2011Journal of Medicinal Chemistry87 citations Open access
Semantic Scholar
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives.
F. Chimenti, S. Carradori, D. Secci, A. Bolasco +5 more
2010European journal of medicinal chemistry87 citations Open access
Semantic Scholar
Selective inhibitory activity against MAO and molecular modeling studies of 2-thiazolylhydrazone derivatives.
F. Chimenti, E. Maccioni, D. Secci, A. Bolasco +8 more
2007Journal of Medicinal Chemistry87 citations Open access
Semantic Scholar
Synthesis, stereochemical identification, and selective inhibitory activity against human monoamine oxidase-B of 2-methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones.
F. Chimenti, E. Maccioni, D. Secci, A. Bolasco +10 more
2008Journal of Medicinal Chemistry86 citations Open access
Semantic Scholar
Anti-inflammatory, analgesic and antipyretic 4,6-disubstituted 3-cyano-2-aminopyridines
F. Manna, F. Chimenti, A. Bolasco, B. Bizzarri +3 more
199985 citations
Semantic Scholar
Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp.
F. Chimenti, B. Bizzarri, E. Maccioni, D. Secci +9 more
2007Bioorganic & Medicinal Chemistry Letters82 citations
Semantic Scholar
Investigations on the 2-thiazolylhydrazyne scaffold: synthesis and molecular modeling of selective human monoamine oxidase inhibitors.
F. Chimenti, A. Bolasco, D. Secci, P. Chimenti +6 more
2010Bioorganic & Medicinal Chemistry80 citations Open access
Semantic Scholar
Focusing on new monoamine oxidase inhibitors
A. Bolasco, S. Carradori, R. Fioravanti
2010Expert Opinion on Therapeutic Patents73 citations
Semantic Scholar
Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitors.
D. Secci, S. Carradori, B. Bizzarri, A. Bolasco +6 more
2014Bioorganic & Medicinal Chemistry65 citations
Semantic Scholar
Monoamine oxidase isoform-dependent tautomeric influence in the recognition of 3,5-diaryl pyrazole inhibitors.
F. Chimenti, R. Fioravanti, A. Bolasco, F. Manna +6 more
2007Journal of Medicinal Chemistry61 citations Open access
Semantic Scholar
Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii.
Melissa D'Ascenzio, B. Bizzarri, C. De Monte, S. Carradori +6 more
2014European journal of medicinal chemistry59 citations
Semantic Scholar
CPTH6, a Thiazole Derivative, Induces Histone Hypoacetylation and Apoptosis in Human Leukemia Cells
D. Trisciuoglio, Ylenia Ragazzoni, A. Pelosi, M. Desideri +13 more
2011Clinical Cancer Research58 citations
Semantic Scholar
Synthesis, biological evaluation and 3D-QSAR of 1,3,5-trisubstituted-4,5-dihydro-(1H)-pyrazole derivatives as potent and highly selective monoamine oxidase A inhibitors.
F. Chimenti, A. Bolasco, F. Manna, D. Secci +9 more
2006Current Medicinal Chemistry54 citations
Semantic Scholar
Synthesis and in vitro selective anti-Helicobacter pylori activity of pyrazoline derivatives.
F. Chimenti, B. Bizzarri, F. Manna, A. Bolasco +7 more
2005Bioorganic & Medicinal Chemistry Letters53 citations
Semantic Scholar
Anti-inflammatory, analgesic and antipyretic N-acetyl-Δ2-pyrazolines and dihydrothienocoumarines
F. Manna, F. Chimenti, A. Bolasco, Cenicola Ml +4 more
199253 citations
Semantic Scholar
Anti-inflammatory, analgesic and antipyretic 4,6-disubstituted 3-cyanopyridine-2-ones and 3-cyano-2-aminopyridines
F. Manna, F. Chimenti, A. Bolasco, A. Filippelli +4 more
199253 citations
Semantic Scholar
Analytical and semipreparative high performance liquid chromatography enantioseparation of new substituted 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazoles on polysaccharide-based chiral stationary phases in normal-phase, polar organic and reversed-phase conditions.
R. Cirilli, A. Simonelli, R. Ferretti, A. Bolasco +4 more
2006Journal of Chromatography A52 citations
Semantic Scholar
Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides.
F. Chimenti, B. Bizzarri, A. Bolasco, D. Secci +7 more
2006European journal of medicinal chemistry52 citations
Semantic Scholar
Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives.
C. De Monte, S. Carradori, B. Bizzarri, A. Bolasco +7 more
2016European journal of medicinal chemistry50 citations Open access
Semantic Scholar
Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives.
D. Secci, B. Bizzarri, A. Bolasco, S. Carradori +5 more
2012European journal of medicinal chemistry49 citations
Semantic Scholar
Synthesis and cytotoxicity of novel (thiazol-2-yl)hydrazine derivatives as promising anti-Candida agents.
S. Carradori, D. Secci, A. Bolasco, D. Rivanera +4 more
2013European journal of medicinal chemistry46 citations
Semantic Scholar
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential
S. Carradori, D. Secci, A. Bolasco, P. Chimenti +1 more
2012Expert Opinion on Therapeutic Patents46 citations
Semantic Scholar
Simple Extraction and HPLC Determination of UV-A and UV-B Filters in Sunscreen Products
D. Orsi, G. Giannini, L. Gagliardi, R. Porrà +4 more
200646 citations
Semantic Scholar
Synthesis and biological evaluation of novel conjugated coumarin‐thiazole systems
F. Chimenti, S. Carradori, D. Secci, A. Bolasco +3 more
200945 citations
Semantic Scholar
Recent advances in the development of selective human MAO-B inhibitors: (hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines.
D. Secci, A. Bolasco, S. Carradori, Melissa D'Ascenzio +2 more
2012European journal of medicinal chemistry44 citations Open access
Semantic Scholar
Conventional and Microwave-Assisted Synthesis of Benzimidazole Derivatives and Their In Vitro Inhibition of Human Cyclooxygenase
D. Secci, A. Bolasco, Melissa D'Ascenzio, F. Della Sala +2 more
201244 citations
Semantic Scholar
Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors.
D. Secci, S. Carradori, A. Bolasco, B. Bizzarri +2 more
2012Current Topics in Medicinal Chemistry43 citations
Semantic Scholar
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors.
F. Chimenti, D. Secci, A. Bolasco, P. Chimenti +13 more
2010Bioorganic & Medicinal Chemistry43 citations Open access
Semantic Scholar
Synthesis, molecular modeling studies and selective inhibitory activity against MAO of N1-propanoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives.
F. Chimenti, R. Fioravanti, A. Bolasco, F. Manna +7 more
2008European journal of medicinal chemistry42 citations Open access
Semantic Scholar
Synthesis, stereochemical separation, and biological evaluation of selective inhibitors of human MAO-B: 1-(4-arylthiazol-2-yl)-2-(3-methylcyclohexylidene)hydrazines.
F. Chimenti, D. Secci, A. Bolasco, P. Chimenti +7 more
2010Journal of Medicinal Chemistry41 citations Open access
Semantic Scholar
High-performance liquid chromatographic separation of enantiomers and diastereomers of 2-methylcyclohexanone thiosemicarbazone, and determination of absolute configuration and configurational stability.
Roberto Cirilli, R. Ferretti, F. la Torre, D. Secci +3 more
2007Journal of Chromatography A40 citations
Semantic Scholar
Synthesis and biological assessment of novel 2-thiazolylhydrazones and computational analysis of their recognition by monoamine oxidase B.
S. Distinto, M. Yáñez, S. Alcaro, M. Cardia +10 more
2012European journal of medicinal chemistry38 citations Open access
Semantic Scholar
A novel class of selective anti-Helicobacter pylori agents 2-oxo-2H-chromene-3-carboxamide derivatives.
F. Chimenti, B. Bizzarri, A. Bolasco, D. Secci +8 more
2007Bioorganic & Medicinal Chemistry Letters38 citations
Semantic Scholar
Simultaneous determination of triprolidine, pseudoephedrine, paracetamol and dextromethorphan by HPLC
D. De Orsi, L. Gagliardi, A. Bolasco, D. Tonelli
199637 citations
Semantic Scholar

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D. Secci×42
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D. Secci — researcher profile on SciRah
P. Chimenti×30
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P. Chimenti — researcher profile on SciRah
F. Chimenti×29
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F. Chimenti — researcher profile on SciRah
S. Carradori×28
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B. Bizzarri — researcher profile on SciRah

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