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C. G. Caldwell · SciRah

Researcher profile · Semantic Scholar

C. G. Caldwell

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C. G. Caldwell — researcher profile on SciRah

h-index: 21
Works: 43
Citations: 1,045

Most-cited papers

Binding of 2-aryl-4-(piperidin-1-yl)butanamines and 1,3,4-trisubstituted pyrrolidines to human CCR5: a molecular modeling-guided mutagenesis study of the binding pocket.
L. Castonguay, Youmin Weng, W. Adolfsen, J. di Salvo +10 more
2003Biochemistry90 citations
Semantic Scholar
Isoform-Selective and Stereoselective Inhibition of Hypoxia Inducible Factor-2.
T. H. Scheuermann, Daniel P. Stroud, Christopher E Sleet, Liela Bayeh +8 more
2015Journal of Medicinal Chemistry77 citations Open access
Semantic Scholar
The di--butylsilylene protecting group for diols
B. Trost, C. G. Caldwell
198168 citations
Semantic Scholar
Substituted 4,6-diaminoquinolines as inhibitors of C5a receptor binding.
T. Lanza, P. Durette, Thomas E. Rollins, S. Siciliano +5 more
1992Journal of Medicinal Chemistry67 citations Open access
Semantic Scholar
Sulfur-substituted dienes and the silylene protecting group in synthesis. Deoxypillaromycinone
B. Trost, C. G. Caldwell, E. Murayama, D. Heissler
198363 citations
Semantic Scholar
Fluoropyrrolidine amides as dipeptidyl peptidase IV inhibitors.
C. G. Caldwell, Ping Chen, Jiafang He, E. Parmee +10 more
2004Bioorganic & Medicinal Chemistry Letters48 citations Open access
Semantic Scholar
Discovery of human CCR5 antagonists containing hydantoins for the treatment of HIV-1 infection.
Dooseop Kim, Li-Ping Wang, C. G. Caldwell, Ping Chen +18 more
2001Bioorganic & Medicinal Chemistry Letters46 citations Open access
Semantic Scholar
Design, synthesis, and SAR of heterocycle-containing antagonists of the human CCR5 receptor for the treatment of HIV-1 infection.
Dooseop Kim, Li-Ping Wang, C. G. Caldwell, Ping Chen +18 more
2001Bioorganic & Medicinal Chemistry Letters42 citations Open access
Semantic Scholar
Photoisomerization mechanism of the rhodopsin chromophore: picosecond photolysis of pigment containing 11-cis-locked eight-membered ring retinal.
Taku Mizukami, Hideki Kandori, Yoshinori Shichida, Arh-Hwang Chen +5 more
1993Proceedings of the National Academy of Sciences of the United States of America40 citations Open access
Semantic Scholar
Novel tetrahydropyran analogs as dipeptidyl peptidase IV inhibitors: Profile of clinical candidate (2R,3S,5R)-2- (2,5-difluorophenyl)-5-(4,6-dihydropyrrolo [3,4-c]pyrazol-5-(1H)-yl)tetrahydro-2H-pyran-3-amine (23) [corrected].
T. Biftu, Xiaoxia Qian, Ping Chen, D. Feng +16 more
2013Bioorganic & Medicinal Chemistry Letters39 citations Open access
Semantic Scholar
Additions and Corrections - Bacteriorhodopsins Containing Cyanine Dye Chromophores. Support for the External Point-Charge Model
F. Derguini, C. G. Caldwell, M. Motto, V. Balogh‐Nair +1 more
198339 citations
Semantic Scholar
1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists: modifications of the arylpropylpiperidine side chains.
C. L. Lynch, C. A. Willoughby, J. Hale, Edward J Holson +26 more
2003Bioorganic & Medicinal Chemistry Letters38 citations Open access
Semantic Scholar
Total synthesis of 1-156,602, a novel cyclic hexadepsipeptide antibiotic
P. Durette, F. Baker, P. L. Barker, J. Boger +5 more
199034 citations
Semantic Scholar
A Convenient Synthesis of Enantiomerically Pure (2S,3S)- or (2R,3R)-3-Hydroxyleucine
C. G. Caldwell, S. Bondy
199032 citations
Semantic Scholar
2,3-Dihydro-5-benzofuranols as antioxidant-based inhibitors of leukotriene biosynthesis.
M. Hammond, I. Kopka, Robert A. Zambias, C. G. Caldwell +5 more
1989Journal of Medicinal Chemistry31 citations
Semantic Scholar
Synthesis of the lipophilic side chain of the cyclic hexadepsipeptide antibiotic L-156,602
C. G. Caldwell, K. Rupprecht, S. Bondy, Alita A. Davis
199030 citations
Semantic Scholar
METABOLIC ACTIVATION OF FLUOROPYRROLIDINE DIPEPTIDYL PEPTIDASE-IV INHIBITORS BY RAT LIVER MICROSOMES
S. Xu, Bing Zhu, Y. Teffera, Deborah E. Pan +5 more
2004Drug Metabolism And Disposition29 citations
Semantic Scholar
Substituted 2-aminopyridines as inhibitors of nitric oxide synthases.
W. Hagmann, C. G. Caldwell, Ping Chen, P. Durette +19 more
2000Bioorganic & Medicinal Chemistry Letters24 citations Open access
Semantic Scholar
Phosphinic acid inhibitors of matrix metalloproteinases
C. G. Caldwell, S. Sahoo, S. Polo, R. R. Eversole +11 more
199624 citations
Semantic Scholar
Confirmation of the secondary deuterium isotope effect for the peptidyl prolyl cis-trans isomerase activity of cyclophilin by a competitive, double-label technique
R. Harrison, C. G. Caldwell, A. Rosegay, D. Melillo +1 more
199023 citations
Semantic Scholar
Comparison of the structure of human recombinant short form stromelysin by multidimensional heteronuclear NMR and X-ray crystallography
P. Gooley, J. O'Connell, A. Marcy, G. C. Cuca +4 more
1996Journal of Biomolecular NMR21 citations
Semantic Scholar
Imidazopiperidine amides as dipeptidyl peptidase IV inhibitors for the treatment of diabetes.
Ping Chen, C. G. Caldwell, R. Mathvink, B. Leiting +7 more
2007Bioorganic & Medicinal Chemistry Letters18 citations Open access
Semantic Scholar
Synthesis of analogs of (1,4)-3- and 5-imino oxazepane, thiazepane, and diazepane as inhibitors of nitric oxide synthases.
K. Shankaran, K. Donnelly, Shrenik K. Shah, C. G. Caldwell +8 more
2004Bioorganic & Medicinal Chemistry Letters17 citations Open access
Semantic Scholar
Synthesis of optically active 3-diazoacetylretinals with triisopropylphenylsulfonylhydrazone
H. Ok, C. G. Caldwell, D. Schroeder, Anil Kumar Singh +1 more
198816 citations Open access
Semantic Scholar
A convenient synthesis of 4-tert-butyl-5-benzofuranols and dihydrobenzofuranols
R. Zambias, C. G. Caldwell, I. Kopka, M. Hammond
198815 citations
Semantic Scholar
Orally active inhibitors of stromelysin-1 (MMP-3)
K. Chapman, P. Durette, C. G. Caldwell, Kelly M. Sperow +8 more
199614 citations
Semantic Scholar
Synthesis and evaluation of [(1R)-1-amino-2-(2,5-difluorophenyl)ethyl]cyclohexanes and 4-[(1R)-1-amino-2-(2,5-difluorophenyl)ethyl]piperidines as DPP-4 inhibitors.
Ping Chen, C. G. Caldwell, W. Ashton, Joseph K. Wu +4 more
2011Bioorganic & Medicinal Chemistry Letters13 citations Open access
Semantic Scholar
CCR5 antagonists: 3-(pyrrolidin-1-yl)propionic acid analogues with potent anti-HIV activity.
C. L. Lynch, J. Hale, R. Budhu, Amy L Gentry +22 more
2003Organic Letters12 citations
Semantic Scholar
Syntheses and biological evaluation of 5-(piperidin-1-yl)-3-phenyl-pentylsulfones as CCR5 antagonists.
K. Shankaran, K. Donnelly, Shrenik K. Shah, C. G. Caldwell +21 more
2004Bioorganic & Medicinal Chemistry Letters11 citations Open access
Semantic Scholar
Synthesis of retinals with eight- and nine-membered rings in the side chain. Models for rhodopsin photobleaching intermediates
C. G. Caldwell, F. Derguini, C. Bigge, Arh-Hwang Chen +4 more
199311 citations
Semantic Scholar
Effects of Matrix Metalloproteinases on Cartilage Biophysical Properties in Vitro and in Vivo a
Lawrence J. Bonassar, Claribel G. Paguio, E. Frank, Kimberly A. Jeffries +5 more
1994Annals of the New York Academy of Sciences8 citations
Semantic Scholar
The inhibition of C5a receptor binding by analogs of L-156,602, a cyclic hexadepsipeptide antibiotic
P. Durette, I. Kopka, T. Lanza, Joung L. Goulet +12 more
19923 citations
Semantic Scholar
Corrigendum to “Novel tetrahydropyran analogs as dipeptidyl peptidase IV inhibitors: Profile of clinical candidate (2R,3S,5R)-2-(2,5-difluorophenyl)-5-(4,6-dihydropyrrolo[3,4-c]pyrazol-5-(1H)-yl)tetrahydro-2H-pyran-3-amine (23)” [Bioorg. Med. Chem. Lett. 23 (2013) 5361–5366]
T. Biftu, Xiaoxia Qian, Ping Chen, D. Feng +16 more
20142 citations Open access
Semantic Scholar
Inhibition of hif-2.alpha. heterodimerization with hif 1.beta. (arnt)
R. Bruick, C. G. Caldwell, D. Frantz, K. Gardner +3 more
20130 citations
Semantic Scholar
Pyrimidines bicycliques en tant qu'inhibiteurs de la dipeptidyl-peptidase-iv dans le traitement ou la prevention de diabetes
W. Ashton, C. G. Caldwell, H. Dong, Yinghong Gao +2 more
20060 citations
Semantic Scholar
Inhibiteurs de peptidase dipeptidyl destines au traitement ou a la prevention du diabete
W. Ashton, C. G. Caldwell, Hyun O. Ok, Emma R. Parmee +1 more
20020 citations
Semantic Scholar
6,6‐Dimethylfulvene
C. G. Caldwell
20010 citations
Semantic Scholar
Dibenzyl N,N‐Diethylphosphoramidite
C. G. Caldwell
20010 citations
Semantic Scholar
Synthesis of Retinals with Eight- and Nine-Membered Rings in the Side Chain. Models for Rhodopsin Photobleaching Intermediates.
C. G. Caldwell, F. Derguini, C. Bigge, Arh-Hwang Chen +4 more
19930 citations
Semantic Scholar
A Convenient Synthesis of Enantiomerically Pure (2S,3S)‐ or (2R,3R)‐3‐Hydroxyleucine.
C. G. Caldwell, S. Bondy
19900 citations
Semantic Scholar
A Convenient Synthesis of 4-tert-Butyl-5-benzofuranols and Dihydrobenzofuranols.
R. Zambias, C. G. Caldwell, I. Kopka, M. Hammond
19890 citations
Semantic Scholar
Synthesis of Optically Active 3-Diazoacetylretinals with Triisopropylphenylsulfonylhydrazone.
H. Ok, C. G. Caldwell, D. Schroeder, Anil Kumar Singh +1 more
19880 citations
Semantic Scholar
THE DI-TERT-BUTYLSILYLENE PROTECTING GROUP FOR DIOLS
B. Trost, C. G. Caldwell
19820 citations
Semantic Scholar

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