Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency, Pharmacokinetics, and Metabolic Properties to Obtain Atropisomeric Quinolinone (AM-0466) that Affords Robust in Vivo Activity.
Russell F. Graceffa, A. Boezio, J. Able, S. Altmann +40 more
2017Journal of Medicinal Chemistry62 citations Open access
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